BR0211749B1 - processo para a preparação de derivados de 4-(imidazol-1- il)benzenossulfonamida - Google Patents
processo para a preparação de derivados de 4-(imidazol-1- il)benzenossulfonamidaInfo
- Publication number
- BR0211749B1 BR0211749B1 BRPI0211749-5B1A BR0211749A BR0211749B1 BR 0211749 B1 BR0211749 B1 BR 0211749B1 BR 0211749 A BR0211749 A BR 0211749A BR 0211749 B1 BR0211749 B1 BR 0211749B1
- Authority
- BR
- Brazil
- Prior art keywords
- imidazol
- formula
- preparation
- benzenesulfonamide derivatives
- chem
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/64—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C303/00—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides
- C07C303/36—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of amides of sulfonic acids
- C07C303/40—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of amides of sulfonic acids by reactions not involving the formation of sulfonamide groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C311/00—Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
- C07C311/30—Sulfonamides, the carbon skeleton of the acid part being further substituted by singly-bound nitrogen atoms, not being part of nitro or nitroso groups
- C07C311/37—Sulfonamides, the carbon skeleton of the acid part being further substituted by singly-bound nitrogen atoms, not being part of nitro or nitroso groups having the sulfur atom of at least one of the sulfonamide groups bound to a carbon atom of a six-membered aromatic ring
- C07C311/38—Sulfonamides, the carbon skeleton of the acid part being further substituted by singly-bound nitrogen atoms, not being part of nitro or nitroso groups having the sulfur atom of at least one of the sulfonamide groups bound to a carbon atom of a six-membered aromatic ring having sulfur atoms of sulfonamide groups and amino groups bound to carbon atoms of six-membered rings of the same carbon skeleton
- C07C311/39—Sulfonamides, the carbon skeleton of the acid part being further substituted by singly-bound nitrogen atoms, not being part of nitro or nitroso groups having the sulfur atom of at least one of the sulfonamide groups bound to a carbon atom of a six-membered aromatic ring having sulfur atoms of sulfonamide groups and amino groups bound to carbon atoms of six-membered rings of the same carbon skeleton having the nitrogen atom of at least one of the sulfonamide groups bound to hydrogen atoms or to an acyclic carbon atom
- C07C311/40—Sulfonamides, the carbon skeleton of the acid part being further substituted by singly-bound nitrogen atoms, not being part of nitro or nitroso groups having the sulfur atom of at least one of the sulfonamide groups bound to a carbon atom of a six-membered aromatic ring having sulfur atoms of sulfonamide groups and amino groups bound to carbon atoms of six-membered rings of the same carbon skeleton having the nitrogen atom of at least one of the sulfonamide groups bound to hydrogen atoms or to an acyclic carbon atom to an acyclic carbon atom of a hydrocarbon radical substituted by singly-bound oxygen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D233/68—Halogen atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Health & Medical Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Animal Behavior & Ethology (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pain & Pain Management (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Rheumatology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ES200101853A ES2184633B1 (es) | 2001-08-07 | 2001-08-07 | Procedimiento para la preparacion de derivados de 4-(imidazol-1-il) bencenosulfonamida. |
| PCT/ES2002/000385 WO2003016285A1 (es) | 2001-08-07 | 2002-08-01 | Procedimiento para la preparacion de derivados de 4-(imidazol-1-il)bencenosulfonamida |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| BR0211749A BR0211749A (pt) | 2004-10-13 |
| BR0211749B1 true BR0211749B1 (pt) | 2013-09-10 |
| BRPI0211749B8 BRPI0211749B8 (pt) | 2021-05-25 |
Family
ID=8498662
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BRPI0211749A BRPI0211749B8 (pt) | 2001-08-07 | 2002-08-01 | processo para a preparação de derivados de 4-(imidazol-1- il)benzenossulfonamida |
Country Status (17)
| Country | Link |
|---|---|
| US (2) | US7351836B2 (pt) |
| EP (1) | EP1424329B1 (pt) |
| JP (1) | JP4309262B2 (pt) |
| KR (1) | KR100888905B1 (pt) |
| AR (2) | AR037231A1 (pt) |
| AT (1) | ATE396976T1 (pt) |
| BR (1) | BRPI0211749B8 (pt) |
| CA (1) | CA2456531C (pt) |
| CY (1) | CY1108861T1 (pt) |
| DE (1) | DE60226879D1 (pt) |
| DK (1) | DK1424329T3 (pt) |
| ES (2) | ES2184633B1 (pt) |
| HK (1) | HK1066214A1 (pt) |
| MX (1) | MXPA04001147A (pt) |
| NO (1) | NO326162B1 (pt) |
| PT (1) | PT1424329E (pt) |
| WO (1) | WO2003016285A1 (pt) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| BR112015000507A2 (pt) | 2012-07-12 | 2017-06-27 | Chiesi Farm Spa | inibição de enzimas |
| WO2022269384A1 (en) * | 2021-06-24 | 2022-12-29 | Ami Organics Ltd. | A process for the direct synthesis of fedratinib intermediate |
| KR102703324B1 (ko) * | 2022-11-08 | 2024-09-06 | 국민대학교산학협력단 | 아미노벤즈이미다졸 유도체 및 이의 제조방법 |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TNSN99111A1 (fr) * | 1998-06-11 | 2005-11-10 | Pfizer | Derives de sulfonylbenzene nouveaux, procede pour leur preparation et compositions pharmaceutiques les contenant. |
| JP4216475B2 (ja) * | 1998-07-02 | 2009-01-28 | クリプターグラフィー リサーチ インコーポレイテッド | 漏洩抵抗力を有する暗号索引付き鍵の更新方法及びデバイス |
| AR024222A1 (es) * | 1998-10-16 | 2002-09-25 | Palau Pharma Sa | Imidazoles con actividad antiinflamatoria un procedimiento para su preparacion y composiciones farmaceuticas que lo contienen |
| ES2159489B1 (es) * | 2000-03-23 | 2002-04-16 | Uriach & Cia Sa J | Nuevos derivados de imidazol con actividad antiinflamatoria. |
-
2001
- 2001-08-07 ES ES200101853A patent/ES2184633B1/es not_active Expired - Fee Related
-
2002
- 2002-08-01 DE DE60226879T patent/DE60226879D1/de not_active Expired - Lifetime
- 2002-08-01 CA CA2456531A patent/CA2456531C/en not_active Expired - Lifetime
- 2002-08-01 BR BRPI0211749A patent/BRPI0211749B8/pt not_active IP Right Cessation
- 2002-08-01 MX MXPA04001147A patent/MXPA04001147A/es active IP Right Grant
- 2002-08-01 PT PT02794802T patent/PT1424329E/pt unknown
- 2002-08-01 JP JP2003521211A patent/JP4309262B2/ja not_active Expired - Fee Related
- 2002-08-01 EP EP02794802A patent/EP1424329B1/en not_active Expired - Lifetime
- 2002-08-01 AT AT02794802T patent/ATE396976T1/de active
- 2002-08-01 ES ES02794802T patent/ES2307817T3/es not_active Expired - Lifetime
- 2002-08-01 WO PCT/ES2002/000385 patent/WO2003016285A1/es active IP Right Grant
- 2002-08-01 US US10/485,950 patent/US7351836B2/en not_active Expired - Fee Related
- 2002-08-01 KR KR1020047001749A patent/KR100888905B1/ko not_active IP Right Cessation
- 2002-08-01 DK DK02794802T patent/DK1424329T3/da active
- 2002-08-06 AR ARP020102972A patent/AR037231A1/es not_active Application Discontinuation
-
2004
- 2004-03-05 NO NO20040981A patent/NO326162B1/no not_active IP Right Cessation
- 2004-11-17 HK HK04109044A patent/HK1066214A1/xx not_active IP Right Cessation
-
2008
- 2008-04-01 US US12/060,574 patent/US8476456B2/en not_active Expired - Fee Related
- 2008-08-21 CY CY20081100892T patent/CY1108861T1/el unknown
-
2012
- 2012-04-25 AR ARP120101436A patent/AR086065A2/es unknown
Also Published As
| Publication number | Publication date |
|---|---|
| JP2005502659A (ja) | 2005-01-27 |
| CA2456531A1 (en) | 2003-02-27 |
| ES2184633B1 (es) | 2004-08-01 |
| BRPI0211749B8 (pt) | 2021-05-25 |
| MXPA04001147A (es) | 2004-07-08 |
| WO2003016285A8 (es) | 2003-08-28 |
| JP4309262B2 (ja) | 2009-08-05 |
| EP1424329A1 (en) | 2004-06-02 |
| AR086065A2 (es) | 2013-11-13 |
| CY1108861T1 (el) | 2014-08-13 |
| ES2307817T3 (es) | 2008-12-01 |
| DK1424329T3 (da) | 2008-09-29 |
| BR0211749A (pt) | 2004-10-13 |
| DE60226879D1 (de) | 2008-07-10 |
| KR100888905B1 (ko) | 2009-03-16 |
| EP1424329B1 (en) | 2008-05-28 |
| US7351836B2 (en) | 2008-04-01 |
| US8476456B2 (en) | 2013-07-02 |
| CA2456531C (en) | 2010-12-14 |
| PT1424329E (pt) | 2008-08-06 |
| US20040242872A1 (en) | 2004-12-02 |
| NO20040981L (no) | 2004-03-05 |
| NO326162B1 (no) | 2008-10-13 |
| AR037231A1 (es) | 2004-11-03 |
| US20090012307A1 (en) | 2009-01-08 |
| KR20040020079A (ko) | 2004-03-06 |
| ES2184633A1 (es) | 2003-04-01 |
| HK1066214A1 (en) | 2005-03-18 |
| ATE396976T1 (de) | 2008-06-15 |
| WO2003016285A1 (es) | 2003-02-27 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B25A | Requested transfer of rights approved |
Owner name: PALAU PHARMA, S.A. (ES) Free format text: TRANSFERIDO DE: J. URIACH AND CIA. S.A. |
|
| B06F | Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette] | ||
| B15K | Others concerning applications: alteration of classification |
Free format text: ALTERADA DA INT.CL: C07D 233/68, C07D 233/64, C07C 311/16 Ipc: C07D 233/68 (2011.01), C07D 233/64 (2011.01), C07C |
|
| B07D | Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette] | ||
| B07E | Notification of approval relating to section 229 industrial property law [chapter 7.5 patent gazette] |
Free format text: NOTIFICACAO DE ANUENCIA RELACIONADA COM O ART 229 DA LPI |
|
| B09A | Decision: intention to grant [chapter 9.1 patent gazette] | ||
| B16A | Patent or certificate of addition of invention granted [chapter 16.1 patent gazette] |
Free format text: PRAZO DE VALIDADE: 10 (DEZ) ANOS CONTADOS A PARTIR DE 10/09/2013, OBSERVADAS AS CONDICOES LEGAIS. |
|
| B16C | Correction of notification of the grant [chapter 16.3 patent gazette] |
Free format text: PRAZO DE VALIDADE: 20 (VINTE) ANOS CONTADOS A PARTIR DE 01/08/2002 OBSERVADAS AS CONDICOES LEGAIS. PATENTE CONCEDIDA CONFORME ADI 5.529/DF |
|
| B21A | Patent or certificate of addition expired [chapter 21.1 patent gazette] |
Free format text: PATENTE EXTINTA EM 01/08/2022 |