BR0209877A - Derivados de piperidinacarboxamida, processo para a respectiva preparação e as composições farmacêuticas que os contêm - Google Patents
Derivados de piperidinacarboxamida, processo para a respectiva preparação e as composições farmacêuticas que os contêmInfo
- Publication number
- BR0209877A BR0209877A BR0209877-6A BR0209877A BR0209877A BR 0209877 A BR0209877 A BR 0209877A BR 0209877 A BR0209877 A BR 0209877A BR 0209877 A BR0209877 A BR 0209877A
- Authority
- BR
- Brazil
- Prior art keywords
- preparation
- pharmaceutical compositions
- compositions containing
- receptors
- piperidinecarboxamide
- Prior art date
Links
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
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- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
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- General Health & Medical Sciences (AREA)
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- Pulmonology (AREA)
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- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Hematology (AREA)
- Physical Education & Sports Medicine (AREA)
- Psychiatry (AREA)
- Urology & Nephrology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Oncology (AREA)
- Rheumatology (AREA)
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- Virology (AREA)
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- Endocrinology (AREA)
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Abstract
"DERIVADOS DE PIPERIDINACARBOXAMIDA, PROCESSO PARA A RESPECTIVA PREPARAçãO E AS COMPOSIçõES FARMACêUTICAS QUE OS CONTêM". A presente invenção refere-se aos compostos de fórmula: (1), assim como seus sais com ácidos minerais ou orgânicos, seus solvatos e/ou seus hidratos, apresentando uma afinidade muito grande ao mesmo tempo com os receptores NK~ 2~ humanos da neuroquinina A e com os receptores NK~ 3~ humanos da neuroquinina B e sendo antagonistas desses receptores. A presente invenção refere-se igualmente ao seu processo de preparação, às composições farmacêuticas que os contêm e à sua utilização para a preparação de medicamentos.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR0106691A FR2824828B1 (fr) | 2001-05-21 | 2001-05-21 | Nouveaux derives de piperidinecarboxamide, un procede pour leur preparation et les compositions pharmaceutiques les contenant |
PCT/FR2002/001663 WO2002094821A1 (fr) | 2001-05-21 | 2002-05-17 | Nouveaux derives de piperidinecarboxamide, un procede pour leur preparation et les compositions pharmaceutiques les contenant |
Publications (1)
Publication Number | Publication Date |
---|---|
BR0209877A true BR0209877A (pt) | 2004-06-08 |
Family
ID=8863515
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR0209877-6A BR0209877A (pt) | 2001-05-21 | 2002-05-17 | Derivados de piperidinacarboxamida, processo para a respectiva preparação e as composições farmacêuticas que os contêm |
Country Status (36)
Country | Link |
---|---|
US (2) | US20040180890A1 (pt) |
EP (1) | EP1395582B1 (pt) |
JP (1) | JP2004529968A (pt) |
KR (1) | KR20030097886A (pt) |
CN (1) | CN1249059C (pt) |
AR (1) | AR035247A1 (pt) |
AT (1) | ATE294798T1 (pt) |
AU (1) | AU2002313065B2 (pt) |
BG (1) | BG108341A (pt) |
BR (1) | BR0209877A (pt) |
CA (1) | CA2445631A1 (pt) |
CZ (1) | CZ20033132A3 (pt) |
DE (1) | DE60204015T2 (pt) |
DK (1) | DK1395582T3 (pt) |
EA (1) | EA006236B1 (pt) |
EE (1) | EE200300553A (pt) |
ES (1) | ES2242032T3 (pt) |
FR (1) | FR2824828B1 (pt) |
HK (1) | HK1060129A1 (pt) |
HR (1) | HRP20030923A2 (pt) |
HU (1) | HUP0401563A2 (pt) |
IL (1) | IL158660A0 (pt) |
IS (1) | IS7008A (pt) |
MA (1) | MA27022A1 (pt) |
MX (1) | MXPA03010133A (pt) |
NO (1) | NO20035163D0 (pt) |
NZ (1) | NZ529206A (pt) |
PL (1) | PL367341A1 (pt) |
PT (1) | PT1395582E (pt) |
SK (1) | SK14192003A3 (pt) |
TN (1) | TNSN03118A1 (pt) |
TW (1) | TWI258480B (pt) |
UA (1) | UA75400C2 (pt) |
WO (1) | WO2002094821A1 (pt) |
YU (1) | YU86603A (pt) |
ZA (1) | ZA200308344B (pt) |
Families Citing this family (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
ES2312856T3 (es) | 2002-12-13 | 2009-03-01 | Smithkline Beecham Corporation | Compuestos heterociclicos como antagonistas de ccr5. |
FR2873373B1 (fr) | 2004-07-23 | 2006-09-08 | Sanofi Synthelabo | Derives de 4-arylmorpholin-3-one, leur preparation et leur application en therapeutique |
US20070219214A1 (en) * | 2006-02-01 | 2007-09-20 | Solvay Pharmaceuticals Gmbh | Dual NK2/NK3-antagonists, pharmaceutical compositions comprising them, and processes for their preparation |
AU2007211475A1 (en) * | 2006-02-01 | 2007-08-09 | Solvay Pharmaceuticals Gmbh | Novel dual NK2/NK3-antagonists, pharmaceutical compositions comprising them and processes for their preparations |
FR2912058A1 (fr) * | 2007-02-07 | 2008-08-08 | Sanofi Aventis Sa | Utilisation d'un compose antagoniste des recepteurs nk2 de la neurokinine a pour la preparation de medicaments utiles pour la prevention et le traitement des dysfonctions sexuelles |
EP2244716B1 (en) * | 2008-01-11 | 2019-09-25 | United Paragon Associates Inc. | Fertilized egg isolate and use thereof |
US20110152233A1 (en) | 2009-12-18 | 2011-06-23 | Henner Knust | Pyrrolidine compounds |
TWI475015B (zh) * | 2010-03-11 | 2015-03-01 | Sumitomo Dainippon Pharma Co Ltd | N-醯基環狀胺衍生物或其醫藥上容許之鹽 |
US10314835B2 (en) | 2014-06-25 | 2019-06-11 | Emory University | Methods of managing conditioned fear with neurokinin receptor antagonists |
EP3881843A4 (en) * | 2018-11-15 | 2022-08-03 | Kyushu University, National University Corporation | PROPHYLACTIC OR THERAPEUTIC AGENT AND MEDICAL COMPOSITION FOR IL-31 MEDIATED DISEASE |
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US5689663A (en) * | 1992-06-19 | 1997-11-18 | Microsoft Corporation | Remote controller user interface and methods relating thereto |
US5780466A (en) * | 1995-01-30 | 1998-07-14 | Sanofi | Substituted heterocyclic compounds method of preparing them and pharmaceutical compositions in which they are present |
FR2729954B1 (fr) * | 1995-01-30 | 1997-08-01 | Sanofi Sa | Composes heterocycliques substitues, procede pour leur preparation et compositions pharmaceutiques les contenant |
FR2738819B1 (fr) * | 1995-09-14 | 1997-12-05 | Sanofi Sa | Nouveaux composes antagonistes selectifs du recepteur nk3 humain, procede pour leur obtention et compositions pharmaceutiques les contenant |
RU2135494C1 (ru) * | 1995-12-01 | 1999-08-27 | Санкио Компани Лимитед | Гетероциклические соединения и композиция на их основе, проявляющая антагонистическое действие в отношении рецепторов тахикинина |
JP3192631B2 (ja) * | 1997-05-28 | 2001-07-30 | 三共株式会社 | 飽和複素環化合物からなる医薬 |
BR9815348A (pt) * | 1997-12-04 | 2000-10-17 | Sankyo Co | " composto, uso deste ou de um sal farmacologicamente aceitável, éster ou outro derivado do mesmo, medicamento, agentes preventivos ou terapêuticos para asma e/ou bronquite, para rinite, para doença alérgica, e para incontinência urinária, e, processos de prevenção ou tratamento de asma e/ou bronquite, de rinite, de doença alérgica, e de incontinência urinária. " |
AU1684300A (en) * | 1998-12-10 | 2000-06-26 | Sankyo Company Limited | Cyclohexylpiperidine derivatives |
FR2791346B3 (fr) * | 1999-03-25 | 2001-04-27 | Sanofi Sa | Nouveaux derives de morpholine, procede pour leur preparation et compositions pharmaceutiques les contenant |
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