AR035247A1 - Derivados de piperidinacarboxamida, un procedimiento para su preparacion y las composiciones farmaceuticas que los contienen - Google Patents

Derivados de piperidinacarboxamida, un procedimiento para su preparacion y las composiciones farmaceuticas que los contienen

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Publication number
AR035247A1
AR035247A1 ARP020101870A ARP020101870A AR035247A1 AR 035247 A1 AR035247 A1 AR 035247A1 AR P020101870 A ARP020101870 A AR P020101870A AR P020101870 A ARP020101870 A AR P020101870A AR 035247 A1 AR035247 A1 AR 035247A1
Authority
AR
Argentina
Prior art keywords
preparation
pharmaceutical compositions
compositions containing
procedure
piperidinacarboxamida
Prior art date
Application number
ARP020101870A
Other languages
English (en)
Inventor
Xavier Emonds-Alt
Vincenzo Proietto
Original Assignee
Sanofi Aventis
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi Aventis filed Critical Sanofi Aventis
Publication of AR035247A1 publication Critical patent/AR035247A1/es

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/06Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • CCHEMISTRY; METALLURGY
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    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
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Abstract

Compuestos de fórmula (1) donde R1 es hidrógeno o un radical metilo; B es una unión directa o un grupo -CH2- Z es fenilo, 2, 3-diclorofenilo o un 2,6-diclorofenilo, así como también sus sales con ácidos minerales u orgánicos, sus solvatos y/o hidratos, que presentan una afinidad muy fuerte a la vez por los receptores NK2 humanos de la neuroquinina A y por lo s receptores NK3 humanos de la neuroquinina B y son antagonistas de dichos receptores. Procedimiento de preparación, las composiciones farmacéuticas que los contienen y su utilización para la preparación de medicamentos.
ARP020101870A 2001-05-21 2002-05-21 Derivados de piperidinacarboxamida, un procedimiento para su preparacion y las composiciones farmaceuticas que los contienen AR035247A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR0106691A FR2824828B1 (fr) 2001-05-21 2001-05-21 Nouveaux derives de piperidinecarboxamide, un procede pour leur preparation et les compositions pharmaceutiques les contenant

Publications (1)

Publication Number Publication Date
AR035247A1 true AR035247A1 (es) 2004-05-05

Family

ID=8863515

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP020101870A AR035247A1 (es) 2001-05-21 2002-05-21 Derivados de piperidinacarboxamida, un procedimiento para su preparacion y las composiciones farmaceuticas que los contienen

Country Status (36)

Country Link
US (2) US20040180890A1 (es)
EP (1) EP1395582B1 (es)
JP (1) JP2004529968A (es)
KR (1) KR20030097886A (es)
CN (1) CN1249059C (es)
AR (1) AR035247A1 (es)
AT (1) ATE294798T1 (es)
AU (1) AU2002313065B2 (es)
BG (1) BG108341A (es)
BR (1) BR0209877A (es)
CA (1) CA2445631A1 (es)
CZ (1) CZ20033132A3 (es)
DE (1) DE60204015T2 (es)
DK (1) DK1395582T3 (es)
EA (1) EA006236B1 (es)
EE (1) EE200300553A (es)
ES (1) ES2242032T3 (es)
FR (1) FR2824828B1 (es)
HK (1) HK1060129A1 (es)
HR (1) HRP20030923A2 (es)
HU (1) HUP0401563A2 (es)
IL (1) IL158660A0 (es)
IS (1) IS7008A (es)
MA (1) MA27022A1 (es)
MX (1) MXPA03010133A (es)
NO (1) NO20035163D0 (es)
NZ (1) NZ529206A (es)
PL (1) PL367341A1 (es)
PT (1) PT1395582E (es)
SK (1) SK14192003A3 (es)
TN (1) TNSN03118A1 (es)
TW (1) TWI258480B (es)
UA (1) UA75400C2 (es)
WO (1) WO2002094821A1 (es)
YU (1) YU86603A (es)
ZA (1) ZA200308344B (es)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1569931B1 (en) 2002-12-13 2008-10-08 Smithkline Beecham Corporation Heterocyclic compounds as ccr5 antagonists
FR2873373B1 (fr) * 2004-07-23 2006-09-08 Sanofi Synthelabo Derives de 4-arylmorpholin-3-one, leur preparation et leur application en therapeutique
US20070219214A1 (en) * 2006-02-01 2007-09-20 Solvay Pharmaceuticals Gmbh Dual NK2/NK3-antagonists, pharmaceutical compositions comprising them, and processes for their preparation
CN101374811A (zh) * 2006-02-01 2009-02-25 索尔瓦药物有限公司 新型双重nk2/nk3-拮抗剂、含它们的药物组合物、及其制备方法
FR2912058A1 (fr) * 2007-02-07 2008-08-08 Sanofi Aventis Sa Utilisation d'un compose antagoniste des recepteurs nk2 de la neurokinine a pour la preparation de medicaments utiles pour la prevention et le traitement des dysfonctions sexuelles
CA2749333C (en) * 2008-01-11 2021-03-23 Jerald Bain Fertilized egg isolate and uses thereof
US20110152233A1 (en) 2009-12-18 2011-06-23 Henner Knust Pyrrolidine compounds
WO2011111875A1 (en) * 2010-03-11 2011-09-15 Dainippon Sumitomo Pharma Co., Ltd. N-acyl cyclic amine derivative or pharmaceutically acceptable salt thereof
EP3915560A1 (en) 2014-06-25 2021-12-01 Emory University Methods of managing conditioned fear with neurokinin receptor antagonists
WO2020101017A1 (ja) * 2018-11-15 2020-05-22 国立大学法人九州大学 Il-31介在性疾患の予防又は治療剤及び医薬組成物

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5689663A (en) * 1992-06-19 1997-11-18 Microsoft Corporation Remote controller user interface and methods relating thereto
US5780466A (en) * 1995-01-30 1998-07-14 Sanofi Substituted heterocyclic compounds method of preparing them and pharmaceutical compositions in which they are present
FR2729954B1 (fr) * 1995-01-30 1997-08-01 Sanofi Sa Composes heterocycliques substitues, procede pour leur preparation et compositions pharmaceutiques les contenant
FR2738819B1 (fr) * 1995-09-14 1997-12-05 Sanofi Sa Nouveaux composes antagonistes selectifs du recepteur nk3 humain, procede pour leur obtention et compositions pharmaceutiques les contenant
HU224225B1 (hu) * 1995-12-01 2005-06-28 Sankyo Co. Ltd. Tachikinin receptor antagonista hatású heterociklusos vegyületek, ezek előállítási eljárása és alkalmazásuk gyógyszerkészítmények előállítására
JP3192631B2 (ja) * 1997-05-28 2001-07-30 三共株式会社 飽和複素環化合物からなる医薬
ATE297906T1 (de) * 1997-12-04 2005-07-15 Sankyo Co Alicyclische acylierte heterocyclenderivate
AU1684300A (en) * 1998-12-10 2000-06-26 Sankyo Company Limited Cyclohexylpiperidine derivatives
FR2791346B3 (fr) * 1999-03-25 2001-04-27 Sanofi Sa Nouveaux derives de morpholine, procede pour leur preparation et compositions pharmaceutiques les contenant

Also Published As

Publication number Publication date
EA006236B1 (ru) 2005-10-27
HUP0401563A2 (hu) 2004-12-28
MA27022A1 (fr) 2004-12-20
IS7008A (is) 2003-10-30
PL367341A1 (en) 2005-02-21
TWI258480B (en) 2006-07-21
NO20035163D0 (no) 2003-11-20
BR0209877A (pt) 2004-06-08
WO2002094821A1 (fr) 2002-11-28
NZ529206A (en) 2005-09-30
FR2824828A1 (fr) 2002-11-22
EE200300553A (et) 2004-02-16
ES2242032T3 (es) 2005-11-01
AU2002313065B2 (en) 2007-06-28
ZA200308344B (en) 2004-10-27
ATE294798T1 (de) 2005-05-15
KR20030097886A (ko) 2003-12-31
CA2445631A1 (fr) 2002-11-28
PT1395582E (pt) 2005-08-31
TNSN03118A1 (fr) 2005-12-23
CZ20033132A3 (cs) 2004-02-18
CN1518549A (zh) 2004-08-04
HK1060129A1 (en) 2004-07-30
BG108341A (bg) 2004-12-30
US20080261976A1 (en) 2008-10-23
YU86603A (sh) 2006-05-25
DE60204015T2 (de) 2006-01-12
EA200301087A1 (ru) 2004-04-29
CN1249059C (zh) 2006-04-05
DK1395582T3 (da) 2005-08-29
HRP20030923A2 (en) 2004-02-29
UA75400C2 (en) 2006-04-17
EP1395582B1 (fr) 2005-05-04
US20040180890A1 (en) 2004-09-16
JP2004529968A (ja) 2004-09-30
SK14192003A3 (sk) 2004-06-08
IL158660A0 (en) 2004-05-12
MXPA03010133A (es) 2005-03-31
DE60204015D1 (de) 2005-06-09
FR2824828B1 (fr) 2005-05-20
EP1395582A1 (fr) 2004-03-10

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