BR0209267A - Pirimidinas fundidas como antagonistas do fator de liberação de corticotropina (crf) - Google Patents

Pirimidinas fundidas como antagonistas do fator de liberação de corticotropina (crf)

Info

Publication number
BR0209267A
BR0209267A BR0209267-0A BR0209267A BR0209267A BR 0209267 A BR0209267 A BR 0209267A BR 0209267 A BR0209267 A BR 0209267A BR 0209267 A BR0209267 A BR 0209267A
Authority
BR
Brazil
Prior art keywords
crf
antagonists
releasing factor
corticotropin releasing
fused pyrimidines
Prior art date
Application number
BR0209267-0A
Other languages
English (en)
Portuguese (pt)
Inventor
Anna Maria Capelli
Romano Di Fabio
Chiara Marchionni
Fabrizio Micheli
Alessandra Pasquarello
Benedetta Perini
Yves St-Denis
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB0110567A external-priority patent/GB0110567D0/en
Priority claimed from GB0110569A external-priority patent/GB0110569D0/en
Priority claimed from GB0110570A external-priority patent/GB0110570D0/en
Priority claimed from GB0117420A external-priority patent/GB0117420D0/en
Priority claimed from GB0117399A external-priority patent/GB0117399D0/en
Priority claimed from GB0117401A external-priority patent/GB0117401D0/en
Priority claimed from GB0203201A external-priority patent/GB0203201D0/en
Priority claimed from GB0206834A external-priority patent/GB0206834D0/en
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Publication of BR0209267A publication Critical patent/BR0209267A/pt

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
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    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
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    • A61K51/02—Preparations containing radioactive substances for use in therapy or testing in vivo characterised by the carrier, i.e. characterised by the agent or material covalently linked or complexing the radioactive nucleus
    • A61K51/04—Organic compounds
    • A61K51/041—Heterocyclic compounds
    • A61K51/044—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins
    • A61K51/0459—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins having six-membered rings with two nitrogen atoms as the only ring hetero atoms, e.g. piperazine
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    • A61K51/0463—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
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    • A61K51/0465—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
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    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
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  • Optics & Photonics (AREA)
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  • Epidemiology (AREA)
  • Physics & Mathematics (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Diabetes (AREA)
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  • Pulmonology (AREA)
  • Pain & Pain Management (AREA)
  • Dermatology (AREA)
  • Endocrinology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Urology & Nephrology (AREA)
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BR0209267-0A 2001-04-30 2002-04-30 Pirimidinas fundidas como antagonistas do fator de liberação de corticotropina (crf) BR0209267A (pt)

Applications Claiming Priority (9)

Application Number Priority Date Filing Date Title
GB0110567A GB0110567D0 (en) 2001-04-30 2001-04-30 Chemical compounds
GB0110569A GB0110569D0 (en) 2001-04-30 2001-04-30 Chemical compounds
GB0110570A GB0110570D0 (en) 2001-04-30 2001-04-30 Chemical compounds
GB0117420A GB0117420D0 (en) 2001-07-17 2001-07-17 Chemical compounds
GB0117399A GB0117399D0 (en) 2001-07-17 2001-07-17 Chemical compounds
GB0117401A GB0117401D0 (en) 2001-07-17 2001-07-17 Chemical compounds
GB0203201A GB0203201D0 (en) 2002-02-11 2002-02-11 Chemical compounds
GB0206834A GB0206834D0 (en) 2002-03-22 2002-03-22 Chemical compounds
PCT/GB2002/002029 WO2002088095A1 (en) 2001-04-30 2002-04-30 Fused pyrimidines as antagonists of the corticotropin releasing factor (crf)

Publications (1)

Publication Number Publication Date
BR0209267A true BR0209267A (pt) 2004-06-15

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ID=27571152

Family Applications (1)

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BR0209267-0A BR0209267A (pt) 2001-04-30 2002-04-30 Pirimidinas fundidas como antagonistas do fator de liberação de corticotropina (crf)

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US (1) US7279474B2 (enExample)
EP (1) EP1383747B1 (enExample)
JP (1) JP2004528349A (enExample)
KR (1) KR20040015206A (enExample)
CN (1) CN1649848A (enExample)
AR (1) AR033295A1 (enExample)
AT (1) ATE386727T1 (enExample)
AU (1) AU2002253357B2 (enExample)
BR (1) BR0209267A (enExample)
CA (1) CA2446514A1 (enExample)
CZ (1) CZ20032946A3 (enExample)
DE (1) DE60225127T2 (enExample)
ES (1) ES2301633T3 (enExample)
HU (1) HUP0304054A2 (enExample)
IL (1) IL158062A0 (enExample)
MX (1) MXPA03009938A (enExample)
NO (1) NO20034836L (enExample)
PL (1) PL366934A1 (enExample)
WO (1) WO2002088095A1 (enExample)

Families Citing this family (66)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ATE397609T1 (de) * 2001-06-12 2008-06-15 Glaxo Group Ltd Corticotropinfreisetzungsfaktor antagonisten
GB0117396D0 (en) * 2001-07-17 2001-09-05 Glaxo Group Ltd Chemical compounds
EP1583531B1 (en) * 2003-01-16 2007-04-18 SB Pharmco Puerto Rico Inc Heteroaryl-substituted pyrrolo[2, 3- b]pyridine derivatives as crf receptor antagonists
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