BR0016534A - Benzofenona( alfa)-d-glicopiranosidas, preparo e uso terapêutico - Google Patents

Benzofenona( alfa)-d-glicopiranosidas, preparo e uso terapêutico

Info

Publication number
BR0016534A
BR0016534A BR0016534-4A BR0016534A BR0016534A BR 0016534 A BR0016534 A BR 0016534A BR 0016534 A BR0016534 A BR 0016534A BR 0016534 A BR0016534 A BR 0016534A
Authority
BR
Brazil
Prior art keywords
alpha
glycopyranosides
group
benzophenone
preparation
Prior art date
Application number
BR0016534-4A
Other languages
English (en)
Inventor
Luc Lebreton
Christiane Legendre
Soth Samreth
Original Assignee
Fournier Ind & Sante
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Fournier Ind & Sante filed Critical Fournier Ind & Sante
Publication of BR0016534A publication Critical patent/BR0016534A/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20Carbocyclic rings
    • C07H15/203Monocyclic carbocyclic rings other than cyclohexane rings; Bicyclic carbocyclic ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7028Compounds having saccharide radicals attached to non-saccharide compounds by glycosidic linkages
    • A61K31/7034Compounds having saccharide radicals attached to non-saccharide compounds by glycosidic linkages attached to a carbocyclic compound, e.g. phloridzin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H1/00Processes for the preparation of sugar derivatives

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • Genetics & Genomics (AREA)
  • Biotechnology (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Urology & Nephrology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Vascular Medicine (AREA)
  • Epidemiology (AREA)
  • Cardiology (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

"BENZOFENONA <244>-D-GLICOPIRANOSIDAS, PREPARO E USO TERAPêUTICO". A presente invenção se refere, no tocante a novos produtos industriais, a: (i) os <244.-D-glicopiranosidas [4-(4-cianobenzoil)fenil] da fórmula I: no qual o grupo R do <244>-D-glicopiranosil é um grupo do <244>-D-glicopiranosil, do <244>-D-galactopiranosil, do <244>-D-manopiranosil, do <244>-D-arabinopiranosil, do <244>-D-lixopiranosil ou do <244>-D-ribopiranosil; e (ii) seus ésters resultando da esterificação de pelo menos de uma função OH em cada grupo do glicopiranosil por um ácido alcanóico ou cicloalcanóico de C2-c4. Estes <244>-D-glicopiranosidas da novela [4-(4-cianobenzoil)fenil] são úteis em terapias para combater a chapa ateromatus.
BR0016534-4A 1999-12-23 2000-12-06 Benzofenona( alfa)-d-glicopiranosidas, preparo e uso terapêutico BR0016534A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR9916387A FR2802929B1 (fr) 1999-12-23 1999-12-23 Benzophenone alpha-d-glycopyranosides, preparation et utilisation en therapeutique
PCT/FR2000/003420 WO2001047941A2 (fr) 1999-12-23 2000-12-06 BENZOPHENONE α-D-GLYCOPYRANOSIDES, PREPARATION ET UTILISATION EN THERAPEUTIQUE

Publications (1)

Publication Number Publication Date
BR0016534A true BR0016534A (pt) 2002-09-24

Family

ID=9553754

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0016534-4A BR0016534A (pt) 1999-12-23 2000-12-06 Benzofenona( alfa)-d-glicopiranosidas, preparo e uso terapêutico

Country Status (20)

Country Link
EP (1) EP1240177B1 (pt)
JP (1) JP2003519158A (pt)
KR (1) KR20020070999A (pt)
AT (1) ATE244257T1 (pt)
AU (1) AU2523601A (pt)
BR (1) BR0016534A (pt)
CA (1) CA2395557A1 (pt)
CZ (1) CZ20022196A3 (pt)
DE (1) DE60003718T2 (pt)
DK (1) DK1240177T3 (pt)
ES (1) ES2202212T3 (pt)
FR (1) FR2802929B1 (pt)
IL (1) IL150271A0 (pt)
MX (1) MXPA02006337A (pt)
NO (1) NO20022972D0 (pt)
PL (1) PL356635A1 (pt)
PT (1) PT1240177E (pt)
RU (1) RU2002116674A (pt)
SK (1) SK9062002A3 (pt)
WO (1) WO2001047941A2 (pt)

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2492830A1 (fr) * 1980-10-29 1982-04-30 Sori Soc Rech Ind Nouveaux composes appartenant a la famille des benzoyl- et a-hydroxybenzyl-phenyl-osides, leur procede de preparation et leur application en therapeutique
FI92189C (fi) * 1986-03-17 1994-10-10 Eisai Co Ltd Menetelmä lääkeaineina käyttökelpoisen difenyylimetaanijohdannaisen valmistamiseksi
BR9911585A (pt) * 1998-06-24 2001-03-20 Fournier Ind & Sante Compostos derivados a partir de uma alfa-d-xilose, método para a preparação e uso terapêutico

Also Published As

Publication number Publication date
EP1240177B1 (fr) 2003-07-02
AU2523601A (en) 2001-07-09
NO20022972L (no) 2002-06-20
IL150271A0 (en) 2002-12-01
ATE244257T1 (de) 2003-07-15
CA2395557A1 (en) 2001-07-05
FR2802929A1 (fr) 2001-06-29
NO20022972D0 (no) 2002-06-20
WO2001047941A3 (fr) 2001-12-27
WO2001047941A2 (fr) 2001-07-05
PT1240177E (pt) 2003-11-28
MXPA02006337A (es) 2002-12-13
FR2802929B1 (fr) 2003-06-06
JP2003519158A (ja) 2003-06-17
PL356635A1 (en) 2004-06-28
EP1240177A2 (fr) 2002-09-18
CZ20022196A3 (cs) 2002-10-16
KR20020070999A (ko) 2002-09-11
RU2002116674A (ru) 2004-01-10
DE60003718T2 (de) 2004-04-15
DE60003718D1 (de) 2003-08-07
DK1240177T3 (da) 2003-10-06
ES2202212T3 (es) 2004-04-01
SK9062002A3 (en) 2002-12-03

Similar Documents

Publication Publication Date Title
HK1066010A1 (en) Optically active compounds which are useful as intermediates in the preparation of optically acitve-2-imidazoline-5-thione derivatives
AU1392199A (en) Low-ph, acid-containing personal care compositions which exhibit reduced sting
AU4327600A (en) Aryl sulfonyls as factor xa inhibitors
DE69516847D1 (de) Chlorpyrimidine als zwischenprodukte
DK1200418T3 (da) Nematodicide trifluorbutener
NZ521681A (en) Substituted benzoic acid amides and use thereof for the inhibition of angiogenesis
EE05062B1 (et) Dihdroksestrite ja nende derivaatide valmistamismeetod
ITRM930399A0 (it) Uso di esteri della l-carnitina o di acil l- carnitine con idrossiacidi per produrre composizioni farmaceutiche per il trattamento di affezioni cutanee.
TR200400228T4 (tr) Psöryazinin tedavisinde kullanılacak maddeler
UA49884C2 (uk) ПОХІДНІ &lt;font face=&#34;Symbol&#34;&gt;a&lt;/font&gt;-ГІДРОКСИКАРБОНОВОЇ КИСЛОТИ ТА ЛІКАРСЬКИЙ ЗАСІБ НА ЇХ ОСНОВІ
HUP0001693A2 (hu) Alfa-hidroxisavak és/vagy aromás o-hidroxisavak alacsony molekulatömegű oligomer észtereinek alkalmazása kozmetikai készítményekben
AU4080097A (en) Piperazino derivatives as neurokinin antagonists
CA2362698A1 (en) Resorcinol derivatives
BR0016534A (pt) Benzofenona( alfa)-d-glicopiranosidas, preparo e uso terapêutico
TR200001026T2 (tr) Nötrofil elastaz inhibitörü olarak pirolopirolon türevleri.
BRPI0013750B8 (pt) intermediários para a produção de derivados de ácido naftiridina-3-carboxílico
UY27372A1 (es) Derivados de bencimidazol 1-aril-2-n, s u o-sustituidos, su uso para la obtención de medicamentos y preparados farmacéuticos que contienen estos derivados
IT1307751B1 (it) Composizione di catalizzatore contenente fosfati per la preparazionedi poliesteri e procedimenti relativi.
HUP0001841A2 (en) Use of tranexamic acid for the preparation of a human fibrinogen composition
AR030945A1 (es) Amidas de acido fenilciclohexanocarboxilico sustituido y su uso
AU7028798A (en) Use of 2-methylthiazolidine-2,4-dicarboxylic acid as mucolytic agent
AU2300895A (en) Pharmaceutical composition comprising hyaluronic acid for the clearing of arteriosclerosis
ATE241640T1 (de) Fusidinsäure-derivate
ATE299704T1 (de) Warmgeformte feste arzneizusammensetzung zur gesteuerten wirkstoffabgabe von perindopril
AU2666600A (en) Use of phosphonous acid modified polyacrylates as sequestering agents

Legal Events

Date Code Title Description
B11A Dismissal acc. art.33 of ipl - examination not requested within 36 months of filing
B11Y Definitive dismissal - extension of time limit for request of examination expired [chapter 11.1.1 patent gazette]