BR0008712A - Complexos equinocandina/carboidrato - Google Patents

Complexos equinocandina/carboidrato

Info

Publication number
BR0008712A
BR0008712A BR0008712-2A BR0008712A BR0008712A BR 0008712 A BR0008712 A BR 0008712A BR 0008712 A BR0008712 A BR 0008712A BR 0008712 A BR0008712 A BR 0008712A
Authority
BR
Brazil
Prior art keywords
echinocandin
complex
carbohydrate
carbohydrate complexes
treatments
Prior art date
Application number
BR0008712-2A
Other languages
English (en)
Inventor
Larry Arnold Larew
Nathaniel Milton
James Lawrence Sabatowski
Enneth Philip Moder
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of BR0008712A publication Critical patent/BR0008712A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K9/00—Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof
    • C07K9/006—Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof the peptide sequence being part of a ring structure
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/50—Cyclic peptides containing at least one abnormal peptide link
    • C07K7/54—Cyclic peptides containing at least one abnormal peptide link with at least one abnormal peptide link in the ring
    • C07K7/56—Cyclic peptides containing at least one abnormal peptide link with at least one abnormal peptide link in the ring the cyclisation not occurring through 2,4-diamino-butanoic acid
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • General Chemical & Material Sciences (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Communicable Diseases (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicinal Preparation (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Peptides Or Proteins (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Solid-Sorbent Or Filter-Aiding Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)

Abstract

Patente de Invenção: "COMPLEXOSEQUINOCANDINA/CARBOIDRATO". Um complexo de umcomposto equinocandina com um carboidrato é descrito tendomelhorada estabilidade térmica e solubilidade em água. Umprocesso para fazer o complexo equinocandina/carboidrato étambém descrito, assim como o uso do complexo em formulaçõesfarmacêuticas e tratamentos de infecções fúngicas.
BR0008712-2A 1999-03-03 2000-03-02 Complexos equinocandina/carboidrato BR0008712A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US12269299P 1999-03-03 1999-03-03
PCT/US2000/005508 WO2000052037A1 (en) 1999-03-03 2000-03-02 Echinocandin/carbohydrate complexes

Publications (1)

Publication Number Publication Date
BR0008712A true BR0008712A (pt) 2001-12-26

Family

ID=22404173

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0008712-2A BR0008712A (pt) 1999-03-03 2000-03-02 Complexos equinocandina/carboidrato

Country Status (18)

Country Link
US (3) US7041637B2 (pt)
EP (1) EP1157030B1 (pt)
JP (1) JP4272359B2 (pt)
KR (1) KR20020003864A (pt)
CN (1) CN1345333A (pt)
AT (1) ATE248187T1 (pt)
AU (1) AU772633B2 (pt)
BR (1) BR0008712A (pt)
CA (1) CA2362016A1 (pt)
DE (1) DE60004793T2 (pt)
DK (1) DK1157030T3 (pt)
ES (1) ES2204548T3 (pt)
HK (1) HK1040088B (pt)
IL (1) IL145187A0 (pt)
PT (1) PT1157030E (pt)
RU (1) RU2001126723A (pt)
WO (1) WO2000052037A1 (pt)
ZA (1) ZA200108004B (pt)

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AU771727B2 (en) 1999-03-03 2004-04-01 Eli Lilly And Company Processes for making pharmaceutical oral ECB formulations and compositions
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ATE338060T1 (de) 1999-03-03 2006-09-15 Lilly Co Eli Bildung und anionenaustausch von inneren kristallinen ammoniumsalzen des echinocandins b
WO2000051564A1 (en) 1999-03-03 2000-09-08 Eli Lilly And Company Echinocandin pharmaceutical formulations containing micelle-forming surfactants
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JP2005053782A (ja) * 2001-08-31 2005-03-03 Fujisawa Pharmaceut Co Ltd 環状リポペプチド化合物の新規結晶
US6991800B2 (en) * 2002-06-13 2006-01-31 Vicuron Pharmaceuticals Inc. Antifungal parenteral products
RU2284832C2 (ru) * 2004-08-30 2006-10-10 Николай Александрович Киселев Антимикробная композиция для перорального введения
KR101163160B1 (ko) * 2006-03-07 2012-07-17 드리테 파텐트포트폴리오 베타일리궁스게젤샤프트 엠베하 운트 코. 카게 보존제의 가용화물 및 이들의 제조 방법
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CN102614491B (zh) 2011-01-31 2014-04-16 上海天伟生物制药有限公司 一种含有棘白菌素类抗真菌剂米卡芬净的药用组合物及其制备方法和用途
CN102614492B (zh) * 2011-01-31 2013-12-11 上海天伟生物制药有限公司 一种含有棘白菌素类抗真菌剂米卡芬净的液体药用组合物
CN102627689B (zh) * 2012-03-30 2014-08-06 上海天伟生物制药有限公司 一种环肽类化合物的水合物及其制备方法和用途
PL3058958T3 (pl) 2015-02-23 2019-02-28 Selectchemie Ag Kompozycja anidulafunginy
CN110339341A (zh) * 2018-04-03 2019-10-18 江苏恒瑞医药股份有限公司 一种达托霉素或其盐的组合物
KR20210076040A (ko) * 2018-10-11 2021-06-23 임브리아 파마슈티칼스, 인크. Tca 회로 중간체 및 그의 사용 방법
CN109574811B (zh) * 2018-11-22 2021-12-24 中山大学 一种阿尼芬净侧链中间体对戊氧基三联苯甲酸的制备方法
CN116903706B (zh) * 2023-06-13 2024-05-17 深圳市祥根生物有限公司 一种棘白菌素类药物及其制备方法和用途

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Also Published As

Publication number Publication date
CA2362016A1 (en) 2000-09-08
DK1157030T3 (da) 2003-12-22
AU3863500A (en) 2000-09-21
EP1157030A1 (en) 2001-11-28
US20020160942A1 (en) 2002-10-31
IL145187A0 (en) 2002-06-30
ES2204548T3 (es) 2004-05-01
JP4272359B2 (ja) 2009-06-03
US20060111277A1 (en) 2006-05-25
ATE248187T1 (de) 2003-09-15
AU772633B2 (en) 2004-05-06
KR20020003864A (ko) 2002-01-15
HK1040088B (zh) 2004-04-16
RU2001126723A (ru) 2003-09-27
HK1040088A1 (en) 2002-05-24
PT1157030E (pt) 2004-01-30
EP1157030B1 (en) 2003-08-27
DE60004793T2 (de) 2004-07-01
ZA200108004B (en) 2003-06-25
US20090258820A1 (en) 2009-10-15
US8022033B2 (en) 2011-09-20
DE60004793D1 (de) 2003-10-02
WO2000052037A8 (en) 2001-03-22
US7550428B2 (en) 2009-06-23
JP2002539090A (ja) 2002-11-19
CN1345333A (zh) 2002-04-17
WO2000052037A1 (en) 2000-09-08
US7041637B2 (en) 2006-05-09

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Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE A 6A, 7A E 8A ANUIDADES.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: REFERENTE AO DESPACHO PUBLICADO NA RPI 1962 DE 12/08/2008.

B15K Others concerning applications: alteration of classification

Ipc: C07K 9/00 (2006.01), C07K 7/56 (2006.01), A61K 38/