BR0007918A - Processo para preparar oxazolidinonas cìclicas contendo flúor e enxofre - Google Patents

Processo para preparar oxazolidinonas cìclicas contendo flúor e enxofre

Info

Publication number
BR0007918A
BR0007918A BR0007918-9A BR0007918A BR0007918A BR 0007918 A BR0007918 A BR 0007918A BR 0007918 A BR0007918 A BR 0007918A BR 0007918 A BR0007918 A BR 0007918A
Authority
BR
Brazil
Prior art keywords
sulfur
containing fluorine
preparing cyclic
oxazolidinones
oxazolidinones containing
Prior art date
Application number
BR0007918-9A
Other languages
English (en)
Inventor
James R Gage
Original Assignee
Upjohn Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Upjohn Co filed Critical Upjohn Co
Publication of BR0007918A publication Critical patent/BR0007918A/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/10Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D335/00Heterocyclic compounds containing six-membered rings having one sulfur atom as the only ring hetero atom
    • C07D335/02Heterocyclic compounds containing six-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Heterocyclic Compounds Containing Sulfur Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

"PROCESSO PARA PREPARAR OXAZOLIDINONAS CìCLICAS CONTENDO FLúOR E ENXOFRE". A invenção é um processo para preparação de agentes antibacterianos de oxazolidinona cíclica contendo flúor e enxofre que utiliza o carbamato de tetrahidrotiopiran-o fluorado importante da fórmula (IV).
BR0007918-9A 1999-02-01 2000-01-31 Processo para preparar oxazolidinonas cìclicas contendo flúor e enxofre BR0007918A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US11815099P 1999-02-01 1999-02-01
PCT/US2000/000506 WO2000044741A2 (en) 1999-02-01 2000-01-31 Process to prepare cyclic-sulfur fluorine containing oxazolidinones

Publications (1)

Publication Number Publication Date
BR0007918A true BR0007918A (pt) 2001-10-23

Family

ID=22376779

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0007918-9A BR0007918A (pt) 1999-02-01 2000-01-31 Processo para preparar oxazolidinonas cìclicas contendo flúor e enxofre

Country Status (20)

Country Link
US (1) US6239283B1 (pt)
EP (1) EP1149089B1 (pt)
JP (1) JP2002535400A (pt)
KR (1) KR20010101890A (pt)
CN (2) CN1495181A (pt)
AT (2) ATE293616T1 (pt)
AU (1) AU767579B2 (pt)
BR (1) BR0007918A (pt)
CA (1) CA2359711A1 (pt)
DE (2) DE60001807T2 (pt)
DK (1) DK1149089T3 (pt)
ES (2) ES2194709T3 (pt)
HK (1) HK1042697B (pt)
HU (1) HUP0200003A3 (pt)
IL (1) IL144669A0 (pt)
NZ (1) NZ513292A (pt)
PL (1) PL349911A1 (pt)
PT (1) PT1149089E (pt)
WO (1) WO2000044741A2 (pt)
ZA (1) ZA200105844B (pt)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
UA52620C2 (uk) * 1995-09-01 2003-01-15 Фармація Енд Апджон Компані Фенілоксазолідинони, що мають с-с-зв'язок з 4-8-членними гетероциклічними кільцями
ATE301474T1 (de) 2000-06-30 2005-08-15 Pharmacia & Upjohn Co Llc Zusammensetzungen zur behandlung baktrieller infektionen, welche ein oxazolidinonderivat, sulbactam und ampicillin enthalten
US7141588B2 (en) 2002-02-25 2006-11-28 Pfizer, Inc. N-aryl-2-oxazolidinone-5-carboxamides and their derivatives
AR038536A1 (es) 2002-02-25 2005-01-19 Upjohn Co N-aril-2-oxazolidinona-5- carboxamidas y sus derivados
WO2004069832A2 (en) * 2003-02-07 2004-08-19 Warner-Lambert Company Llc Antibacterial agents
JP2006516989A (ja) * 2003-02-07 2006-07-13 ワーナー−ランバート・カンパニー、リミテッド、ライアビリティ、カンパニー 抗菌剤として使用するための二環式環によりn−置換されたオキサゾリジノン誘導体
US7304050B2 (en) 2003-09-16 2007-12-04 Pfizer Inc. Antibacterial agents
CA2576041A1 (en) * 2004-08-06 2006-02-16 Pharmacia & Upjohn Company Llc Oxazolidinones containing oxindoles as antibacterial agents

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
UA52620C2 (uk) * 1995-09-01 2003-01-15 Фармація Енд Апджон Компані Фенілоксазолідинони, що мають с-с-зв'язок з 4-8-членними гетероциклічними кільцями
GB9702213D0 (en) 1996-02-24 1997-03-26 Zeneca Ltd Chemical compounds
EP1114819B1 (en) 1996-04-11 2008-01-09 Pharmacia & Upjohn Company LLC Process to prepare oxazolidinones

Also Published As

Publication number Publication date
AU3207600A (en) 2000-08-18
HUP0200003A3 (en) 2002-11-28
DE60019630D1 (de) 2005-05-25
ZA200105844B (en) 2002-07-16
CN1495181A (zh) 2004-05-12
HUP0200003A2 (en) 2002-06-29
ATE235486T1 (de) 2003-04-15
KR20010101890A (ko) 2001-11-15
JP2002535400A (ja) 2002-10-22
CN1335842A (zh) 2002-02-13
CN1142158C (zh) 2004-03-17
PT1149089E (pt) 2003-07-31
HK1042697A1 (en) 2002-08-23
ATE293616T1 (de) 2005-05-15
US6239283B1 (en) 2001-05-29
CA2359711A1 (en) 2000-08-03
IL144669A0 (en) 2002-05-23
EP1149089B1 (en) 2003-03-26
WO2000044741A3 (en) 2000-12-07
EP1149089A2 (en) 2001-10-31
DE60019630T2 (de) 2006-03-16
DK1149089T3 (da) 2003-07-21
DE60001807D1 (de) 2003-04-30
PL349911A1 (en) 2002-10-07
WO2000044741A2 (en) 2000-08-03
ES2241920T3 (es) 2005-11-01
DE60001807T2 (de) 2003-11-06
NZ513292A (en) 2003-08-29
AU767579B2 (en) 2003-11-20
HK1042697B (zh) 2004-08-20
ES2194709T3 (es) 2003-12-01

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Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE A 7A, 8A E 9A ANUIDADES

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: REFERENTE AO DESPACHO 8.6 NA RPI2003 DE 26/05/2009.