ES2194709T3 - Procedimiento para preparar carbamatos de tetrahidrotiopiran-o-fluorados. - Google Patents

Procedimiento para preparar carbamatos de tetrahidrotiopiran-o-fluorados.

Info

Publication number
ES2194709T3
ES2194709T3 ES00909891T ES00909891T ES2194709T3 ES 2194709 T3 ES2194709 T3 ES 2194709T3 ES 00909891 T ES00909891 T ES 00909891T ES 00909891 T ES00909891 T ES 00909891T ES 2194709 T3 ES2194709 T3 ES 2194709T3
Authority
ES
Spain
Prior art keywords
tetrahydrotiopiran
fluorated
procedure
optionally substituted
phenyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
ES00909891T
Other languages
English (en)
Inventor
James R Gage
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pharmacia and Upjohn Co
Original Assignee
Pharmacia and Upjohn Co
Upjohn Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pharmacia and Upjohn Co, Upjohn Co filed Critical Pharmacia and Upjohn Co
Application granted granted Critical
Publication of ES2194709T3 publication Critical patent/ES2194709T3/es
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/10—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D335/00—Heterocyclic compounds containing six-membered rings having one sulfur atom as the only ring hetero atom
    • C07D335/02—Heterocyclic compounds containing six-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Heterocyclic Compounds Containing Sulfur Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

Un compuesto de fórmula (IV) en la que Réster se selecciona de entre: (I) alquilo C1-C10 opcionalmente sustituido con fenilo o grupos alcoxi 1 a 3 C1-C3; (II) alquenilo C2-C5 opcionalmente sustituido con fenilo o cicloalquilo C3-C7; (III) fenilo opcionalmente sustituido con 1 a 3 C1-C3 grupos alquilo; o (IV) naftilo opcionalmente sustituido con 1 a 3 C1-C3 grupos alquilo.
ES00909891T 1999-02-01 2000-01-31 Procedimiento para preparar carbamatos de tetrahidrotiopiran-o-fluorados. Expired - Lifetime ES2194709T3 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US11815099P 1999-02-01 1999-02-01

Publications (1)

Publication Number Publication Date
ES2194709T3 true ES2194709T3 (es) 2003-12-01

Family

ID=22376779

Family Applications (2)

Application Number Title Priority Date Filing Date
ES00909891T Expired - Lifetime ES2194709T3 (es) 1999-02-01 2000-01-31 Procedimiento para preparar carbamatos de tetrahidrotiopiran-o-fluorados.
ES02009273T Expired - Lifetime ES2241920T3 (es) 1999-02-01 2000-01-31 Derivados de 2-fluoro-(oxido-tiopiran-4-il)benceno.

Family Applications After (1)

Application Number Title Priority Date Filing Date
ES02009273T Expired - Lifetime ES2241920T3 (es) 1999-02-01 2000-01-31 Derivados de 2-fluoro-(oxido-tiopiran-4-il)benceno.

Country Status (20)

Country Link
US (1) US6239283B1 (es)
EP (1) EP1149089B1 (es)
JP (1) JP2002535400A (es)
KR (1) KR20010101890A (es)
CN (2) CN1142158C (es)
AT (2) ATE293616T1 (es)
AU (1) AU767579B2 (es)
BR (1) BR0007918A (es)
CA (1) CA2359711A1 (es)
DE (2) DE60019630T2 (es)
DK (1) DK1149089T3 (es)
ES (2) ES2194709T3 (es)
HK (1) HK1042697B (es)
HU (1) HUP0200003A3 (es)
IL (1) IL144669A0 (es)
NZ (1) NZ513292A (es)
PL (1) PL349911A1 (es)
PT (1) PT1149089E (es)
WO (1) WO2000044741A2 (es)
ZA (1) ZA200105844B (es)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR100463772B1 (ko) * 1995-09-01 2005-11-09 파마시아 앤드 업존 캄파니 엘엘씨 4내지8원헤테로사이클릭환에탄소-탄소결합을갖는페닐옥사졸리디논
US6544991B2 (en) 2000-06-30 2003-04-08 Pharmacia & Upjohn Company Compositions and methods for treating bacterial infections
US7141588B2 (en) * 2002-02-25 2006-11-28 Pfizer, Inc. N-aryl-2-oxazolidinone-5-carboxamides and their derivatives
AR038536A1 (es) * 2002-02-25 2005-01-19 Upjohn Co N-aril-2-oxazolidinona-5- carboxamidas y sus derivados
BRPI0407304A (pt) * 2003-02-07 2006-01-10 Warner Lambert Co Agentes antibacterianos
CA2515311A1 (en) * 2003-02-07 2004-08-19 Warner-Lambert Company Llc Antibacterial agents
US7304050B2 (en) * 2003-09-16 2007-12-04 Pfizer Inc. Antibacterial agents
US20080262056A1 (en) * 2004-08-06 2008-10-23 Pfizer Inc Oxindole Oxazolidinones as Antibacterial Agents

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR100463772B1 (ko) * 1995-09-01 2005-11-09 파마시아 앤드 업존 캄파니 엘엘씨 4내지8원헤테로사이클릭환에탄소-탄소결합을갖는페닐옥사졸리디논
GB9702213D0 (en) 1996-02-24 1997-03-26 Zeneca Ltd Chemical compounds
CN1167701C (zh) 1996-04-11 2004-09-22 法玛西雅厄普约翰美国公司 制备噁唑烷酮胺的方法

Also Published As

Publication number Publication date
IL144669A0 (en) 2002-05-23
HK1042697A1 (en) 2002-08-23
DE60019630T2 (de) 2006-03-16
WO2000044741A3 (en) 2000-12-07
KR20010101890A (ko) 2001-11-15
ES2241920T3 (es) 2005-11-01
HK1042697B (zh) 2004-08-20
ATE235486T1 (de) 2003-04-15
DE60019630D1 (de) 2005-05-25
BR0007918A (pt) 2001-10-23
AU767579B2 (en) 2003-11-20
NZ513292A (en) 2003-08-29
DK1149089T3 (da) 2003-07-21
PL349911A1 (en) 2002-10-07
AU3207600A (en) 2000-08-18
CA2359711A1 (en) 2000-08-03
CN1495181A (zh) 2004-05-12
EP1149089A2 (en) 2001-10-31
ZA200105844B (en) 2002-07-16
CN1335842A (zh) 2002-02-13
DE60001807D1 (de) 2003-04-30
HUP0200003A3 (en) 2002-11-28
PT1149089E (pt) 2003-07-31
HUP0200003A2 (en) 2002-06-29
WO2000044741A2 (en) 2000-08-03
CN1142158C (zh) 2004-03-17
ATE293616T1 (de) 2005-05-15
DE60001807T2 (de) 2003-11-06
US6239283B1 (en) 2001-05-29
EP1149089B1 (en) 2003-03-26
JP2002535400A (ja) 2002-10-22

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