BR0004901A - Processo para a preparação de éteres cìclicos de compostos com piperidinilaminometila e trifluorometila - Google Patents
Processo para a preparação de éteres cìclicos de compostos com piperidinilaminometila e trifluorometilaInfo
- Publication number
- BR0004901A BR0004901A BR0004901-8A BR0004901A BR0004901A BR 0004901 A BR0004901 A BR 0004901A BR 0004901 A BR0004901 A BR 0004901A BR 0004901 A BR0004901 A BR 0004901A
- Authority
- BR
- Brazil
- Prior art keywords
- preparation
- compounds
- piperidinylaminomethyl
- trifluoromethyl
- cyclic ethers
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 title abstract 6
- 238000002360 preparation method Methods 0.000 title abstract 5
- 238000000034 method Methods 0.000 title abstract 4
- 150000004292 cyclic ethers Chemical class 0.000 title abstract 3
- -1 piperidinylaminomethyl Chemical group 0.000 title abstract 3
- 125000002023 trifluoromethyl group Chemical group FC(F)(F)* 0.000 title abstract 2
- 239000000203 mixture Substances 0.000 abstract 2
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 2
- WZKSXHQDXQKIQJ-UHFFFAOYSA-N F[C](F)F Chemical class F[C](F)F WZKSXHQDXQKIQJ-UHFFFAOYSA-N 0.000 abstract 1
- 125000000217 alkyl group Chemical group 0.000 abstract 1
- 125000001188 haloalkyl group Chemical group 0.000 abstract 1
- 125000001475 halogen functional group Chemical group 0.000 abstract 1
- 229910052739 hydrogen Inorganic materials 0.000 abstract 1
- 239000001257 hydrogen Substances 0.000 abstract 1
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 1
- 238000000746 purification Methods 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C69/00—Esters of carboxylic acids; Esters of carbonic or haloformic acids
- C07C69/96—Esters of carbonic or haloformic acids
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D311/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
- C07D311/02—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D311/76—Benzo[c]pyrans
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Neurosurgery (AREA)
- General Health & Medical Sciences (AREA)
- Biomedical Technology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Neurology (AREA)
- Public Health (AREA)
- Psychiatry (AREA)
- Pain & Pain Management (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Pyrane Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US16022699P | 1999-10-18 | 1999-10-18 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BR0004901A true BR0004901A (pt) | 2001-05-29 |
Family
ID=22576040
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BR0004901-8A BR0004901A (pt) | 1999-10-18 | 2000-10-18 | Processo para a preparação de éteres cìclicos de compostos com piperidinilaminometila e trifluorometila |
Country Status (24)
| Country | Link |
|---|---|
| US (2) | US6486325B1 (Direct) |
| EP (1) | EP1095939B1 (Direct) |
| JP (1) | JP3564685B2 (Direct) |
| KR (1) | KR100459952B1 (Direct) |
| CN (1) | CN1293193A (Direct) |
| AR (1) | AR026053A1 (Direct) |
| AT (1) | ATE257477T1 (Direct) |
| AU (1) | AU784275B2 (Direct) |
| BR (1) | BR0004901A (Direct) |
| CA (1) | CA2323315C (Direct) |
| CZ (1) | CZ299029B6 (Direct) |
| DE (1) | DE60007599T2 (Direct) |
| DK (1) | DK1095939T3 (Direct) |
| ES (1) | ES2211455T3 (Direct) |
| HU (1) | HUP0004061A2 (Direct) |
| ID (1) | ID27627A (Direct) |
| IL (1) | IL139012A (Direct) |
| IN (1) | IN190078B (Direct) |
| PL (1) | PL343290A1 (Direct) |
| PT (1) | PT1095939E (Direct) |
| RU (1) | RU2184116C1 (Direct) |
| TR (1) | TR200003002A2 (Direct) |
| YU (1) | YU60600A (Direct) |
| ZA (1) | ZA200005695B (Direct) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TW426667B (en) * | 1997-11-19 | 2001-03-21 | Pfizer | Piperidinylaminomethyl trifluoromethyl cyclic ether compounds as substance P antagonists |
| KR20040064687A (ko) * | 2001-12-21 | 2004-07-19 | 도오레 화인케미칼 가부시키가이샤 | 광학 활성 시스 피페리딘 유도체의 제조법 |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5374637A (en) * | 1989-03-22 | 1994-12-20 | Janssen Pharmaceutica N.V. | N-(3-hydroxy-4-piperidinyl)(dihydrobenzofuran, dihydro-2H-benzopyran or dihydrobenzodioxin)carboxamide derivatives |
| CA2106200C (en) * | 1991-03-26 | 1996-11-19 | Terry J. Rosen | Stereoselective preparation of substituted piperidines |
| US5294744A (en) * | 1993-04-20 | 1994-03-15 | Pfizer Inc. | Formylation process for aromatic aldehydes |
| US5886011A (en) * | 1995-03-27 | 1999-03-23 | Hisamitsu Pharmaceutical Co., Inc. | Piperidine derivatives as substance P antagonists |
| EP0840732B1 (en) * | 1995-07-07 | 2001-03-07 | Pfizer Inc. | Substituted benzolactam compounds as substance p antagonists |
| TW340842B (en) * | 1995-08-24 | 1998-09-21 | Pfizer | Substituted benzylaminopiperidine compounds |
| TW426667B (en) * | 1997-11-19 | 2001-03-21 | Pfizer | Piperidinylaminomethyl trifluoromethyl cyclic ether compounds as substance P antagonists |
| BR0011284A (pt) * | 1999-05-21 | 2002-03-05 | Pfizer Prod Inc | Derivados de 1-trifluorometil-4-hidroxi-7-piperidinilaminometilcr omano |
-
2000
- 2000-10-02 AT AT00308640T patent/ATE257477T1/de not_active IP Right Cessation
- 2000-10-02 DK DK00308640T patent/DK1095939T3/da active
- 2000-10-02 PT PT00308640T patent/PT1095939E/pt unknown
- 2000-10-02 EP EP00308640A patent/EP1095939B1/en not_active Expired - Lifetime
- 2000-10-02 ES ES00308640T patent/ES2211455T3/es not_active Expired - Lifetime
- 2000-10-02 DE DE60007599T patent/DE60007599T2/de not_active Expired - Fee Related
- 2000-10-05 JP JP2000305667A patent/JP3564685B2/ja not_active Expired - Fee Related
- 2000-10-05 YU YU60600A patent/YU60600A/sh unknown
- 2000-10-12 AU AU65474/00A patent/AU784275B2/en not_active Ceased
- 2000-10-12 IL IL139012A patent/IL139012A/en not_active IP Right Cessation
- 2000-10-13 AR ARP000105423A patent/AR026053A1/es unknown
- 2000-10-13 IN IN924MU2000 patent/IN190078B/en unknown
- 2000-10-16 CA CA002323315A patent/CA2323315C/en not_active Expired - Fee Related
- 2000-10-16 ID IDP20000892D patent/ID27627A/id unknown
- 2000-10-16 ZA ZA200005695A patent/ZA200005695B/xx unknown
- 2000-10-16 TR TR2000/03002A patent/TR200003002A2/xx unknown
- 2000-10-17 CN CN00125993A patent/CN1293193A/zh active Pending
- 2000-10-17 US US09/690,346 patent/US6486325B1/en not_active Expired - Fee Related
- 2000-10-17 RU RU2000126151/04A patent/RU2184116C1/ru not_active IP Right Cessation
- 2000-10-17 HU HU0004061A patent/HUP0004061A2/hu unknown
- 2000-10-17 CZ CZ20003840A patent/CZ299029B6/cs not_active IP Right Cessation
- 2000-10-17 KR KR10-2000-0060966A patent/KR100459952B1/ko not_active Expired - Fee Related
- 2000-10-18 PL PL00343290A patent/PL343290A1/xx not_active Application Discontinuation
- 2000-10-18 BR BR0004901-8A patent/BR0004901A/pt not_active Application Discontinuation
-
2002
- 2002-11-13 US US10/065,725 patent/US20030236268A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| PL343290A1 (en) | 2001-04-23 |
| KR20010051069A (ko) | 2001-06-25 |
| DE60007599D1 (de) | 2004-02-12 |
| AR026053A1 (es) | 2002-12-26 |
| IL139012A0 (en) | 2001-11-25 |
| ATE257477T1 (de) | 2004-01-15 |
| PT1095939E (pt) | 2004-04-30 |
| EP1095939A2 (en) | 2001-05-02 |
| KR100459952B1 (ko) | 2004-12-04 |
| DK1095939T3 (da) | 2004-04-13 |
| ES2211455T3 (es) | 2004-07-16 |
| JP3564685B2 (ja) | 2004-09-15 |
| US20030236268A1 (en) | 2003-12-25 |
| ZA200005695B (en) | 2002-04-16 |
| CN1293193A (zh) | 2001-05-02 |
| HU0004061D0 (en) | 2000-12-28 |
| TR200003002A2 (tr) | 2001-05-21 |
| AU6547400A (en) | 2001-04-26 |
| YU60600A (sh) | 2002-12-10 |
| US6486325B1 (en) | 2002-11-26 |
| EP1095939B1 (en) | 2004-01-07 |
| EP1095939A3 (en) | 2001-05-23 |
| RU2184116C1 (ru) | 2002-06-27 |
| DE60007599T2 (de) | 2004-11-11 |
| CA2323315A1 (en) | 2001-04-18 |
| IN190078B (Direct) | 2003-06-07 |
| CZ20003840A3 (cs) | 2002-02-13 |
| HUP0004061A2 (hu) | 2002-05-29 |
| CZ299029B6 (cs) | 2008-04-09 |
| CA2323315C (en) | 2008-07-29 |
| AU784275B2 (en) | 2006-03-02 |
| IL139012A (en) | 2007-06-17 |
| JP2001151773A (ja) | 2001-06-05 |
| ID27627A (id) | 2001-04-19 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B07A | Application suspended after technical examination (opinion) [chapter 7.1 patent gazette] | ||
| B09B | Patent application refused [chapter 9.2 patent gazette] |
Free format text: INDEFIRO O PEDIDO DE ACORDO COM O(S) ARTIGO(S) 8O, 11 E 13 DA LPI. |
|
| B09B | Patent application refused [chapter 9.2 patent gazette] |
Free format text: MANTIDO O INDEFERIMENTO UMA VEZ QUE NAO FOI APRESENTADO RECURSO DENTRO DO PRAZO LEGAL. |