BG63632B1 - N-заместени азабициклохептанови производни, приложими като невролептици - Google Patents

N-заместени азабициклохептанови производни, приложими като невролептици Download PDF

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Publication number
BG63632B1
BG63632B1 BG101221A BG10122197A BG63632B1 BG 63632 B1 BG63632 B1 BG 63632B1 BG 101221 A BG101221 A BG 101221A BG 10122197 A BG10122197 A BG 10122197A BG 63632 B1 BG63632 B1 BG 63632B1
Authority
BG
Bulgaria
Prior art keywords
naphthyl
formula
azabicyclo
exo
compounds
Prior art date
Application number
BG101221A
Other languages
Bulgarian (bg)
English (en)
Other versions
BG101221A (en
Inventor
Gerd Steiner
Rainer Munschauer
Thomas Hoeger
Liliane Unger
Hans-Juergen Teschendorf
Original Assignee
Basf Aktiengesellschaft
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=6524943&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BG63632(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Basf Aktiengesellschaft filed Critical Basf Aktiengesellschaft
Publication of BG101221A publication Critical patent/BG101221A/xx
Publication of BG63632B1 publication Critical patent/BG63632B1/bg

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/52—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring condensed with a ring other than six-membered
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/56—Ring systems containing three or more rings
    • C07D209/80—[b, c]- or [b, d]-condensed
    • C07D209/90—Benzo [c, d] indoles; Hydrogenated benzo [c, d] indoles
    • C07D209/92—Naphthostyrils

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Psychiatry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Indole Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Luminescent Compositions (AREA)
BG101221A 1994-08-04 1997-02-12 N-заместени азабициклохептанови производни, приложими като невролептици BG63632B1 (bg)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE4427647A DE4427647A1 (de) 1994-08-04 1994-08-04 N-substituierte Azabicycloheptan-Derivate, ihre Herstellung und Verwendung
PCT/EP1995/002912 WO1996004245A1 (de) 1994-08-04 1995-07-22 N-substituierte azabicycloheptan-derivate als neuroleptika usw.

Publications (2)

Publication Number Publication Date
BG101221A BG101221A (en) 1997-08-29
BG63632B1 true BG63632B1 (bg) 2002-07-31

Family

ID=6524943

Family Applications (1)

Application Number Title Priority Date Filing Date
BG101221A BG63632B1 (bg) 1994-08-04 1997-02-12 N-заместени азабициклохептанови производни, приложими като невролептици

Country Status (29)

Country Link
US (1) US5753690A (zh)
EP (1) EP0775113B1 (zh)
JP (1) JPH10503504A (zh)
KR (1) KR970704685A (zh)
CN (1) CN1064959C (zh)
AT (1) ATE200482T1 (zh)
AU (1) AU699021B2 (zh)
BG (1) BG63632B1 (zh)
CA (1) CA2196700A1 (zh)
CZ (1) CZ289080B6 (zh)
DE (2) DE4427647A1 (zh)
DK (1) DK0775113T3 (zh)
ES (1) ES2156212T3 (zh)
FI (1) FI970449A (zh)
GR (1) GR3035744T3 (zh)
HR (1) HRP950437B1 (zh)
HU (1) HUT77768A (zh)
IL (1) IL114719A (zh)
MX (1) MX9700854A (zh)
NO (1) NO307376B1 (zh)
NZ (1) NZ290429A (zh)
PL (1) PL182810B1 (zh)
PT (1) PT775113E (zh)
RU (1) RU2160254C2 (zh)
SI (1) SI9520086B (zh)
TW (1) TW378203B (zh)
UA (1) UA44736C2 (zh)
WO (1) WO1996004245A1 (zh)
ZA (1) ZA956476B (zh)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6458821B1 (en) 1998-08-12 2002-10-01 Abbott Laboratories N-substituted azabicycloheptane derivatives, production and use thereof
DE19836406A1 (de) * 1998-08-12 2000-02-17 Basf Ag N-Substituierte Azabicycloheptan-Derivate, ihre Herstellung und Verwendung
DE19836404A1 (de) * 1998-08-12 2000-02-17 Basf Ag N-Substituierte Azabicycloheptan-Derivate, ihre Herstellung und Verwendung
DE19854147A1 (de) * 1998-11-24 2000-05-25 Basf Ag Verwendung von N-substituierten Azabicycloalkan-Derivaten zur Verwendung bei der Bekämpfung der Cocainsucht
JP4754570B2 (ja) * 2004-10-14 2011-08-24 アボット ゲーエムベーハー ウント カンパニー カーゲー ドーパミンｄ３受容体の調節に応答する障害の治療に好適なアザビシクロヘプチル化合物
EP1874801A4 (en) * 2005-03-07 2009-03-25 Univ North Carolina RECA ACTIVITY INHIBITORS TO CONTROL ANTIBIOTIC-RESISTANT BACTERIAL PATHOGENS
FR2953514B1 (fr) * 2009-12-09 2011-12-23 Servier Lab Nouveaux derives azabicyclo[3.2.0]hept-3-yl, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
WO2020239073A1 (zh) * 2019-05-30 2020-12-03 中国科学院上海药物研究所 一种并环化合物、其制备方法和用途

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE4219973A1 (de) * 1992-06-19 1993-12-23 Basf Ag N-substituierte Azabicycloheptan-Derivate, ihre Herstellung und Verwendung
DE4243287A1 (de) * 1992-06-19 1993-12-23 Basf Ag N-Substituierte Azabicycloheptan-Derivate, ihre Herstellung und Verwendung
GB9321481D0 (en) * 1993-10-18 1993-12-08 Alcan Int Ltd Tin oxide
DE4341402A1 (de) * 1993-12-04 1995-06-08 Basf Ag N-substituierte Azabicycloheptan-Derivate, ihre Herstellung und Verwendung

Also Published As

Publication number Publication date
PL318459A1 (en) 1997-06-09
HUT77768A (hu) 1998-08-28
PT775113E (pt) 2001-09-28
EP0775113B1 (de) 2001-04-11
NO970474L (no) 1997-04-01
EP0775113A1 (de) 1997-05-28
DK0775113T3 (da) 2001-05-07
HRP950437A2 (en) 1997-08-31
BG101221A (en) 1997-08-29
JPH10503504A (ja) 1998-03-31
CZ289080B6 (cs) 2001-10-17
SI9520086A (en) 1997-08-31
ATE200482T1 (de) 2001-04-15
ZA956476B (en) 1997-02-03
DE59509186D1 (de) 2001-05-17
TW378203B (en) 2000-01-01
SI9520086B (sl) 2002-02-28
WO1996004245A1 (de) 1996-02-15
US5753690A (en) 1998-05-19
NZ290429A (en) 1998-02-26
MX9700854A (es) 1997-04-30
NO307376B1 (no) 2000-03-27
CZ31197A3 (en) 1997-10-15
CN1064959C (zh) 2001-04-25
CN1156989A (zh) 1997-08-13
FI970449A (fi) 1997-04-03
RU2160254C2 (ru) 2000-12-10
PL182810B1 (pl) 2002-03-29
KR970704685A (ko) 1997-09-06
FI970449A0 (fi) 1997-02-03
AU3116595A (en) 1996-03-04
IL114719A0 (en) 1995-11-27
ES2156212T3 (es) 2001-06-16
AU699021B2 (en) 1998-11-19
DE4427647A1 (de) 1996-02-08
GR3035744T3 (en) 2001-07-31
UA44736C2 (uk) 2002-03-15
NO970474D0 (no) 1997-02-03
IL114719A (en) 2001-03-19
CA2196700A1 (en) 1996-02-15
HRP950437B1 (en) 2002-06-30

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