BG62934B1 - НОВИ ПИРИМИДО(1,2-а)ИНДОЛИ - Google Patents

НОВИ ПИРИМИДО(1,2-а)ИНДОЛИ Download PDF

Info

Publication number
BG62934B1
BG62934B1 BG101379A BG10137997A BG62934B1 BG 62934 B1 BG62934 B1 BG 62934B1 BG 101379 A BG101379 A BG 101379A BG 10137997 A BG10137997 A BG 10137997A BG 62934 B1 BG62934 B1 BG 62934B1
Authority
BG
Bulgaria
Prior art keywords
carbon atoms
branched
branched chain
alkyl
optionally substituted
Prior art date
Application number
BG101379A
Other languages
Bulgarian (bg)
English (en)
Other versions
BG101379A (en
Inventor
Ulrich Mueller
Peter Eckenberg
Rudi Gruetzmann
Hilmar Bischoff
Dirk Denzer
Stefan Wohlfeil
Stefan Lohmer
Ulrich Nielsch
Peter Kolkhof
Original Assignee
Bayer Aktiengesellschaft
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Aktiengesellschaft filed Critical Bayer Aktiengesellschaft
Publication of BG101379A publication Critical patent/BG101379A/xx
Publication of BG62934B1 publication Critical patent/BG62934B1/bg

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Cardiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Indole Compounds (AREA)
BG101379A 1996-04-04 1997-04-02 НОВИ ПИРИМИДО(1,2-а)ИНДОЛИ BG62934B1 (bg)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19613550A DE19613550A1 (de) 1996-04-04 1996-04-04 Neue Pyrimido[1,2-a]indole

Publications (2)

Publication Number Publication Date
BG101379A BG101379A (en) 1997-11-28
BG62934B1 true BG62934B1 (bg) 2000-11-30

Family

ID=7790502

Family Applications (1)

Application Number Title Priority Date Filing Date
BG101379A BG62934B1 (bg) 1996-04-04 1997-04-02 НОВИ ПИРИМИДО(1,2-а)ИНДОЛИ

Country Status (33)

Country Link
US (1) US6114341A (fr)
EP (1) EP0799828A3 (fr)
JP (1) JPH1059972A (fr)
KR (1) KR970070008A (fr)
CN (2) CN1067393C (fr)
AR (1) AR006497A1 (fr)
AU (1) AU725786B2 (fr)
BG (1) BG62934B1 (fr)
BR (1) BR9701675A (fr)
CA (1) CA2201434A1 (fr)
CO (1) CO4520306A1 (fr)
CZ (1) CZ102297A3 (fr)
DE (1) DE19613550A1 (fr)
DZ (1) DZ2201A1 (fr)
EE (1) EE9700078A (fr)
HN (1) HN1997000045A (fr)
HR (1) HRP970154A2 (fr)
HU (1) HUP9700708A3 (fr)
ID (1) ID16520A (fr)
IL (3) IL120590A (fr)
MA (1) MA24131A1 (fr)
MY (1) MY126362A (fr)
NO (1) NO309092B1 (fr)
NZ (1) NZ314497A (fr)
PE (1) PE42398A1 (fr)
PL (1) PL319249A1 (fr)
SG (1) SG63698A1 (fr)
SK (1) SK42797A3 (fr)
SV (1) SV1997000025A (fr)
TN (1) TNSN97061A1 (fr)
TR (1) TR199700261A2 (fr)
YU (1) YU12397A (fr)
ZA (1) ZA972829B (fr)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE19826469A1 (de) * 1998-06-13 2000-05-25 Bayer Ag Verfahren zur Herstellung von 2,4-Dimethylcarbolin und 2,4-Dimethylpyrimido[1,2-a]indol
WO2001074817A1 (fr) * 2000-03-30 2001-10-11 Yamanouchi Pharmaceutical Co., Ltd. Derives d'hydrazide
DE10030375A1 (de) * 2000-06-21 2002-01-03 Bayer Ag Verwendung von MTP-Inhibitoren zur Senkung von ppTRL
JP4254093B2 (ja) * 2001-10-17 2009-04-15 宇部興産株式会社 ５−ハロゲノインドールの製法
DE10349175A1 (de) * 2003-10-22 2005-05-19 Bayer Healthcare Ag Mittel zur Gewichtsreduktion
SI1725234T1 (sl) 2004-03-05 2013-04-30 The Trustees Of The University Of Pennsylvania Postopki zdravljenja nepravilnosti ali bolezni povezanih s hiperlipidemijo in hiperholesterolemijo z minimiziranjem stranskih uäśinkov
AU2005230397B2 (en) * 2004-04-09 2010-04-08 Elanco Animal Health Ireland Limited Intermittent dosing regimen for the treatment of overweight with MTP-inhibitors
MX2007013932A (es) 2005-05-12 2008-01-28 Bard Inc C R Filtro de coagulo de sangre removible.
JP2008542255A (ja) * 2005-05-27 2008-11-27 ファイザー・プロダクツ・インク 肥満症の治療または体重減量の維持のためのカンナビノイド−１受容体アンタゴニストおよびミクロソームトリグリセリド輸送タンパク質阻害物質の併用
CA2616818C (fr) 2005-08-09 2014-08-05 C.R. Bard, Inc. Filtre pour caillots de sang generateurs d'embolie et systeme de mise en place
AU2006304689A1 (en) * 2005-10-18 2007-04-26 Aegerion Pharmaceuticals Compositions for lowering serum cholesterol and/or triglycerides
US10188496B2 (en) 2006-05-02 2019-01-29 C. R. Bard, Inc. Vena cava filter formed from a sheet
US20080161279A1 (en) * 2006-12-21 2008-07-03 Wisler Gerald L Methods of Treating Obesity

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2200584A1 (de) * 1971-01-11 1972-07-27 Wyeth John & Brother Ltd Heterocyclische Verbindungen,Verfahren zu ihrer Herstellung und ihre Verwendung in pharmazeutischen Zubereitungen
ZA718536B (en) * 1971-01-11 1972-09-27 Wyeth John & Brother Ltd Heterocyclic compounds
GB8614246D0 (en) * 1986-06-11 1986-07-16 Wyeth John & Brother Ltd Substituted pyrimidoindoles
DE4112533A1 (de) * 1991-04-17 1992-10-22 Bayer Ag Verfahren zur herstellung von enantiomerenreinen substituierten (chinolin-2-yl-methoxy)phenyl-essigsaeuren
DE4200954A1 (de) * 1991-04-26 1992-10-29 Bayer Ag Heterocyclisch substituierte phenylessigsaeurederivate
DE4208051A1 (de) * 1992-03-13 1993-09-16 Bayer Ag Substituierte phenylessigsaeureamide
DE4208052A1 (de) * 1992-03-13 1993-09-16 Bayer Ag Imidazolyl substituierte phenylessigsaeureamide
DE4309968A1 (de) * 1993-03-26 1994-09-29 Bayer Ag Phenylglycinamide von heterocyclisch substituierten Phenylessigsäurederivaten
US5576342A (en) * 1992-03-13 1996-11-19 Bayer Aktiengesellschaft Phenylglycinamides of heterocyclically substitued phenylacetic acid derivatives
KR950704328A (ko) * 1992-11-05 1995-11-17 데이비드 로버츠 5-HT₄ 수용체 길항제로서의 피페리딘 유도체(Piperidine Derivatives as 5-HT₄ Receptor Antagonists)
DE4302956A1 (de) * 1993-02-03 1994-08-04 Bayer Ag Substituierte Imidazo(4,5-b)pyridine und Benzimidazole

Also Published As

Publication number Publication date
SK42797A3 (en) 1997-11-05
PE42398A1 (es) 1998-10-12
ZA972829B (en) 1997-10-31
ID16520A (id) 1997-10-09
HUP9700708A2 (hu) 1998-10-28
IL131645A (en) 2000-12-06
AR006497A1 (es) 1999-08-25
NO971512L (no) 1997-10-06
SV1997000025A (es) 1997-10-23
CN1176965A (zh) 1998-03-25
TR199700261A2 (xx) 1997-10-21
EE9700078A (et) 1997-10-15
KR970070008A (ko) 1997-11-07
IL120590A (en) 2000-02-17
NO971512D0 (no) 1997-04-03
CA2201434A1 (fr) 1997-10-04
US6114341A (en) 2000-09-05
EP0799828A3 (fr) 1998-04-08
HU9700708D0 (en) 1997-05-28
IL131645A0 (en) 2001-01-28
CZ102297A3 (en) 1997-10-15
MA24131A1 (fr) 1997-10-01
HRP970154A2 (en) 1998-04-30
YU12397A (en) 1999-11-22
CN1067393C (zh) 2001-06-20
EP0799828A2 (fr) 1997-10-08
MY126362A (en) 2006-09-29
BG101379A (en) 1997-11-28
DE19613550A1 (de) 1997-10-09
AU725786B2 (en) 2000-10-19
TNSN97061A1 (fr) 2005-03-15
HUP9700708A3 (en) 2000-01-28
DZ2201A1 (fr) 2002-12-03
NZ314497A (en) 1999-10-28
CN1312246A (zh) 2001-09-12
AU1660397A (en) 1997-10-09
CO4520306A1 (es) 1997-10-15
NO309092B1 (no) 2000-12-11
PL319249A1 (en) 1997-10-13
BR9701675A (pt) 1998-11-03
IL120590A0 (en) 1997-08-14
MX9702445A (es) 1997-10-31
JPH1059972A (ja) 1998-03-03
HN1997000045A (es) 1997-06-26
SG63698A1 (en) 1999-03-30

Similar Documents

Publication Publication Date Title
US6245775B1 (en) Cycloalkano-indole and -azaindole derivatives
US5356911A (en) Substituted biphenylpyridones
BG62934B1 (bg) НОВИ ПИРИМИДО(1,2-а)ИНДОЛИ
HUT55367A (en) Process for producing biphenylmethane derivatives including condensed carbo or heterocyclic imidazole unit, as well as pharmaceutical compositions comprising such compounds
CA2186086A1 (fr) Derives de substitution de xanthines
US6034115A (en) Indolyl-substituted phenylacetic acid derivatives
US6194424B1 (en) Arylacetamides and their use as medicaments
CA2202703A1 (fr) Nouveaux pyridazino-, pyrimido-, pyrazino- et triazino-indoles
US5830902A (en) Quinuclidine derivative having tricyclic hetero condensed ring
US6255330B1 (en) Heterocyclically substituted phenylglycinolamides
MXPA97002445A (en) New pyrimid [1,2-] indo
JPH02200685A (ja) 新規なインドール誘導体
CZ20003952A3 (cs) Sloučenina pyrrolo[l,2-b]pyridazinu, farmaceutické prostředky a způsoby inhibice uvolňování mastných kyselin