BG61841B1 - Алкилови производни на тразодона - Google Patents
Алкилови производни на тразодона Download PDFInfo
- Publication number
- BG61841B1 BG61841B1 BG98896A BG9889694A BG61841B1 BG 61841 B1 BG61841 B1 BG 61841B1 BG 98896 A BG98896 A BG 98896A BG 9889694 A BG9889694 A BG 9889694A BG 61841 B1 BG61841 B1 BG 61841B1
- Authority
- BG
- Bulgaria
- Prior art keywords
- formula
- compound
- alkyl
- hydrogen
- alk
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
- C07D295/06—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by halogen atoms or nitro radicals
- C07D295/073—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by halogen atoms or nitro radicals with the ring nitrogen atoms and the substituents separated by carbocyclic rings or by carbon chains interrupted by carbocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/26—Psychostimulants, e.g. nicotine, cocaine
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C229/00—Compounds containing amino and carboxyl groups bound to the same carbon skeleton
- C07C229/02—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton
- C07C229/04—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated
- C07C229/06—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated having only one amino and one carboxyl group bound to the carbon skeleton
- C07C229/10—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated having only one amino and one carboxyl group bound to the carbon skeleton the nitrogen atom of the amino group being further bound to acyclic carbon atoms or to carbon atoms of rings other than six-membered aromatic rings
- C07C229/16—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated having only one amino and one carboxyl group bound to the carbon skeleton the nitrogen atom of the amino group being further bound to acyclic carbon atoms or to carbon atoms of rings other than six-membered aromatic rings to carbon atoms of hydrocarbon radicals substituted by amino or carboxyl groups, e.g. ethylenediamine-tetra-acetic acid, iminodiacetic acids
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
- C07D295/06—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by halogen atoms or nitro radicals
- C07D295/067—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by halogen atoms or nitro radicals with the ring nitrogen atoms and the substituents attached to the same carbon chain, which is not interrupted by carbocyclic rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Psychiatry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Pain & Pain Management (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ITMI920084A IT1258790B (it) | 1992-01-17 | 1992-01-17 | Alchil derivati del trazodone |
| PCT/EP1993/000080 WO1993014091A1 (en) | 1992-01-17 | 1993-01-14 | Alkyl derivatives of trazodone with cns activity |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| BG98896A BG98896A (bg) | 1995-03-31 |
| BG61841B1 true BG61841B1 (bg) | 1998-07-31 |
Family
ID=11361589
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BG98896A BG61841B1 (bg) | 1992-01-17 | 1994-07-08 | Алкилови производни на тразодона |
Country Status (25)
| Country | Link |
|---|---|
| EP (1) | EP0623131B1 (cs) |
| JP (1) | JP2856912B2 (cs) |
| KR (1) | KR100254690B1 (cs) |
| AT (1) | ATE136307T1 (cs) |
| AU (1) | AU671973B2 (cs) |
| BG (1) | BG61841B1 (cs) |
| BR (1) | BR9305752A (cs) |
| CA (1) | CA2128202C (cs) |
| CZ (1) | CZ282910B6 (cs) |
| DE (1) | DE69302087T2 (cs) |
| DK (1) | DK0623131T3 (cs) |
| ES (1) | ES2088270T3 (cs) |
| FI (2) | FI110186B (cs) |
| GE (1) | GEP20001939B (cs) |
| GR (1) | GR3020420T3 (cs) |
| HU (5) | HU217968B (cs) |
| IT (1) | IT1258790B (cs) |
| NO (2) | NO302365B1 (cs) |
| NZ (1) | NZ246598A (cs) |
| PL (1) | PL170913B1 (cs) |
| RO (1) | RO113465B1 (cs) |
| RU (1) | RU2126801C1 (cs) |
| SK (1) | SK280561B6 (cs) |
| WO (1) | WO1993014091A1 (cs) |
| ZA (1) | ZA93292B (cs) |
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU718075B2 (en) * | 1993-07-01 | 2000-04-06 | Angelini Ricerche S.P.A. Societa Consortile | Intermediates for the preparation of pharmacologically active enantiomers of triazolone compounds |
| IT1268414B1 (it) | 1993-07-01 | 1997-02-27 | Angelini Francesco Ist Ricerca | Enantiomeri farmacologicamente attivi |
| DE19637237A1 (de) * | 1996-09-13 | 1998-03-19 | Merck Patent Gmbh | Piperazin-Derivate |
| US6514989B1 (en) * | 2001-07-20 | 2003-02-04 | Hoffmann-La Roche Inc. | Aromatic and heteroaromatic substituted 1,2,4-triazolo pyridine derivatives |
| MY139563A (en) * | 2002-09-04 | 2009-10-30 | Bristol Myers Squibb Co | Heterocyclic aromatic compounds useful as growth hormone secretagogues |
| TW200726765A (en) * | 2005-06-17 | 2007-07-16 | Bristol Myers Squibb Co | Triazolopyridine cannabinoid receptor 1 antagonists |
| ITMI20051193A1 (it) * | 2005-06-24 | 2006-12-25 | Acraf | Uso farmaceutico di una 1-3-clorofenil-3-alchilpiperazina |
| WO2012072665A1 (en) | 2010-11-30 | 2012-06-07 | Pharmaneuroboost N.V. | Compositions comprising pipamperone and serotonin antagonist reuptake inhibitors |
| RU2706700C1 (ru) | 2019-09-24 | 2019-11-20 | Общество с ограниченной ответственностью "Научно-производственная компания "СКиФФ" | Фармацевтическая композиция для коррекции поведения кошек и собак в стрессовых ситуациях |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US100505A (en) * | 1870-03-08 | Improvement in sash-bolt | ||
| IT1066857B (it) * | 1965-12-15 | 1985-03-12 | Acraf | Derivati della s ipiazolo 4.3 a piridina e processi per la loro preparazione |
| DE2641378A1 (de) * | 1975-09-24 | 1977-04-07 | Sandoz Ag | Neue organische verbindungen, ihre verwendung und herstellung |
| CH624682A5 (cs) * | 1976-11-10 | 1981-08-14 | Sandoz Ag | |
| US4390695A (en) * | 1980-06-23 | 1983-06-28 | E. R. Squibb & Sons, Inc. | Imido, amido and amino derivatives of mercaptoacyl prolines and pipecolic acids |
-
1992
- 1992-01-17 GE GEAP19922648A patent/GEP20001939B/en unknown
- 1992-01-17 IT ITMI920084A patent/IT1258790B/it active IP Right Grant
-
1993
- 1993-01-14 ES ES93902204T patent/ES2088270T3/es not_active Expired - Lifetime
- 1993-01-14 JP JP5512150A patent/JP2856912B2/ja not_active Expired - Fee Related
- 1993-01-14 EP EP93902204A patent/EP0623131B1/en not_active Expired - Lifetime
- 1993-01-14 RO RO94-01203A patent/RO113465B1/ro unknown
- 1993-01-14 BR BR9305752A patent/BR9305752A/pt not_active Application Discontinuation
- 1993-01-14 NZ NZ246598A patent/NZ246598A/xx not_active IP Right Cessation
- 1993-01-14 CZ CZ941732A patent/CZ282910B6/cs not_active IP Right Cessation
- 1993-01-14 AU AU33504/93A patent/AU671973B2/en not_active Ceased
- 1993-01-14 WO PCT/EP1993/000080 patent/WO1993014091A1/en active IP Right Grant
- 1993-01-14 HU HU9502179A patent/HU217968B/hu not_active IP Right Cessation
- 1993-01-14 PL PL93304665A patent/PL170913B1/pl not_active IP Right Cessation
- 1993-01-14 DK DK93902204.2T patent/DK0623131T3/da active
- 1993-01-14 AT AT93902204T patent/ATE136307T1/de not_active IP Right Cessation
- 1993-01-14 RU RU94036769A patent/RU2126801C1/ru not_active IP Right Cessation
- 1993-01-14 SK SK846-94A patent/SK280561B6/sk not_active IP Right Cessation
- 1993-01-14 KR KR1019940702475A patent/KR100254690B1/ko not_active Expired - Fee Related
- 1993-01-14 CA CA002128202A patent/CA2128202C/en not_active Expired - Fee Related
- 1993-01-14 DE DE69302087T patent/DE69302087T2/de not_active Expired - Fee Related
- 1993-01-14 HU HU9402119A patent/HU218678B/hu not_active IP Right Cessation
- 1993-01-15 ZA ZA93292A patent/ZA93292B/xx unknown
-
1994
- 1994-07-08 BG BG98896A patent/BG61841B1/bg unknown
- 1994-07-15 NO NO942668A patent/NO302365B1/no not_active IP Right Cessation
- 1994-07-15 FI FI943386A patent/FI110186B/fi active
-
1995
- 1995-07-19 HU HU9502178A patent/HU217981B/hu not_active IP Right Cessation
- 1995-07-19 HU HU9502177A patent/HU219493B/hu not_active IP Right Cessation
- 1995-07-19 HU HU9502180A patent/HU217982B/hu not_active IP Right Cessation
-
1996
- 1996-07-02 GR GR960401793T patent/GR3020420T3/el unknown
-
1997
- 1997-09-26 NO NO974462A patent/NO303686B1/no not_active IP Right Cessation
-
2002
- 2002-09-16 FI FI20021652A patent/FI113266B/fi active
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