BG60066A3 - Method for the preparation of 4--/3-/4-oxothiazolydine// butynylamine - Google Patents

Method for the preparation of 4--/3-/4-oxothiazolydine// butynylamine

Info

Publication number
BG60066A3
BG60066A3 BG94208A BG9420891A BG60066A3 BG 60066 A3 BG60066 A3 BG 60066A3 BG 94208 A BG94208 A BG 94208A BG 9420891 A BG9420891 A BG 9420891A BG 60066 A3 BG60066 A3 BG 60066A3
Authority
BG
Bulgaria
Prior art keywords
oxothiazolydine
butynylamine
preparation
Prior art date
Application number
BG94208A
Other languages
English (en)
Inventor
Nicholas J Hrib
Original Assignee
Us Hoechst Roussel Pharmaceuti
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Us Hoechst Roussel Pharmaceuti filed Critical Us Hoechst Roussel Pharmaceuti
Publication of BG60066A3 publication Critical patent/BG60066A3/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D277/00Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/60Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425Thiazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A61P29/02Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID] without antiinflammatory effect
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D277/00Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/08Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D277/12Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D277/14Oxygen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/06Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/10Spiro-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Pain & Pain Management (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurology (AREA)
  • Cardiology (AREA)
  • Biomedical Technology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Neurosurgery (AREA)
  • Rheumatology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
BG94208A 1990-04-16 1991-04-09 Method for the preparation of 4--/3-/4-oxothiazolydine// butynylamine BG60066A3 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US07/509,280 US5034392A (en) 1990-04-16 1990-04-16 4-(3-(4-oxothiazolidinyl)butynylamines

Publications (1)

Publication Number Publication Date
BG60066A3 true BG60066A3 (en) 1993-09-15

Family

ID=24025983

Family Applications (1)

Application Number Title Priority Date Filing Date
BG94208A BG60066A3 (en) 1990-04-16 1991-04-09 Method for the preparation of 4--/3-/4-oxothiazolydine// butynylamine

Country Status (26)

Country Link
US (1) US5034392A (ru)
EP (1) EP0452850B1 (ru)
JP (1) JPH07119223B2 (ru)
KR (1) KR0163598B1 (ru)
AR (1) AR248402A1 (ru)
AT (1) ATE163010T1 (ru)
AU (1) AU636972B2 (ru)
BG (1) BG60066A3 (ru)
CA (1) CA2040489C (ru)
CZ (1) CZ284447B6 (ru)
DE (1) DE69128845T2 (ru)
DK (1) DK0452850T3 (ru)
ES (1) ES2112844T3 (ru)
FI (1) FI94755C (ru)
GR (1) GR3026319T3 (ru)
HU (1) HUT61017A (ru)
IE (1) IE911257A1 (ru)
IL (1) IL97852A (ru)
MX (1) MX25359A (ru)
NO (1) NO300134B1 (ru)
NZ (1) NZ237811A (ru)
PL (1) PL165488B1 (ru)
PT (1) PT97371B (ru)
RO (1) RO108683B1 (ru)
RU (1) RU2001914C1 (ru)
ZA (1) ZA912783B (ru)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5273977A (en) * 1990-11-05 1993-12-28 Warner-Lambert Company Substituted tetrahydropyridines and hydroxypiperidines as central nervous system agents
US5147881A (en) * 1990-11-14 1992-09-15 Pfizer Inc 4-(1,2-benzisoxazolyl)piperidine antipsychotic agents
US5194436A (en) * 1991-01-10 1993-03-16 Hoechst-Roussel Pharmaceuticals Inc. 1-piperazinyl-2-butenes and -2-butynes
US5130315A (en) * 1991-01-10 1992-07-14 Raymond R. Wittekind 1-piperazinyl-2-butenes and -2-butynes

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3354178A (en) * 1965-04-09 1967-11-21 Sterling Drug Inc Nu-(4-amino-2-butynyl)-nu-alkylcarboxamides
ES2052675T3 (es) * 1987-11-20 1994-07-16 Hoechst Roussel Pharma 3-(4-piperazinil-sustituido en 1)butil)-4-tiazolidinonas, un procedimiento para su preparacion y su uso como medicamentos.

Also Published As

Publication number Publication date
FI94755C (fi) 1995-10-25
NO300134B1 (no) 1997-04-14
GR3026319T3 (en) 1998-06-30
EP0452850A1 (en) 1991-10-23
CZ284447B6 (cs) 1998-11-11
AR248402A1 (es) 1995-08-18
CS9101065A2 (en) 1991-11-12
IE911257A1 (en) 1991-10-23
NO911465D0 (no) 1991-04-15
HU911239D0 (en) 1991-10-28
JPH07119223B2 (ja) 1995-12-20
AU7502891A (en) 1991-10-17
FI911783A (fi) 1991-10-17
AU636972B2 (en) 1993-05-13
MX25359A (es) 1994-05-31
CA2040489A1 (en) 1991-10-17
RU2001914C1 (ru) 1993-10-30
JPH04234879A (ja) 1992-08-24
HUT61017A (en) 1992-11-30
FI94755B (fi) 1995-07-14
NO911465L (no) 1991-10-17
KR910018367A (ko) 1991-11-30
DK0452850T3 (da) 1998-09-23
ATE163010T1 (de) 1998-02-15
FI911783A0 (fi) 1991-04-12
DE69128845T2 (de) 1998-07-09
EP0452850B1 (en) 1998-02-04
CA2040489C (en) 2003-06-10
KR0163598B1 (ko) 1998-12-01
PL165488B1 (pl) 1994-12-30
IL97852A0 (en) 1992-06-21
US5034392A (en) 1991-07-23
ES2112844T3 (es) 1998-04-16
IL97852A (en) 1994-11-28
NZ237811A (en) 1993-12-23
ZA912783B (en) 1991-12-24
DE69128845D1 (de) 1998-03-12
RO108683B1 (ro) 1994-07-29
PT97371B (pt) 1998-08-31
PT97371A (pt) 1992-01-31
PL289892A1 (en) 1992-07-27

Similar Documents

Publication Publication Date Title
EP0311983A3 (en) Method for the preparation of titanium-silicalites
EP0439829A3 (en) Process for the preparation of copolyestercarbonates
BG50834A3 (en) Method for the preparation of 3- acyl- 2- oxindole- 1- carboxamides
EP0439745A3 (en) Process for the preparation of 2-chloro-5-methyl-pyridine
ZA915396B (en) Process for the preparation of 1-hydroxymethylpyrazoles
BG60066A3 (en) Method for the preparation of 4--/3-/4-oxothiazolydine// butynylamine
EP0595228A3 (en) Process for the preparation of ketals
EP0444460A3 (en) Process for the preparation of acrolin
EP0449778A3 (en) Process for the preparation of hydroxyphenylepropionates
IL97512A0 (en) Process for the preparation of 1-hydroxyalkyl-5-nitro-imidazoles
EP0474016A3 (en) Method for the preparation of 2,3-dihydro-benzofuranes
IL98877A0 (en) Process for the preparation of n-alkylsulfonylamino-sulfonylureas
IL96282A0 (en) Method for the preparation of 5-chlorcarbonyl-5h-dibenz-/b,f/-azepin
ZA887372B (en) Method for the preparation of anilinofumarate
EP0297447A3 (en) Method for the preparation of 2-cyclopentenones
GR3020992T3 (en) Method for the preparation of aminotriazin derivatives
EP0459242A3 (en) Process for the preparation of phenolethers
IL98876A0 (en) Process for the preparation of n-alkylsulfonyl aminosulfonylureas
BG90875A (en) Method for the preparation of potassium dl-asparate and magnesium-bis-dl-aspartate
EP0467308A3 (en) Process for the preparation of 2-hydroxy-3-halogen-5-nitropyridines
PL276494A1 (en) Method for the tionaphthene preparation
GB9111703D0 (en) Method of transsilylation
HUT65995A (en) New method for the preparation of 6-methylene-steroids
GB9205920D0 (en) Process for the preparation of pyrethroide derivatives
PL276633A1 (en) Method for preparation of the 3-chlorpropyltrichlorsilane