BG108683A - Quinuclidine derivatives, processes for preparing them and their uses as m2 and/or m3 muscarinic receptor inhibitors - Google Patents

Quinuclidine derivatives, processes for preparing them and their uses as m2 and/or m3 muscarinic receptor inhibitors

Info

Publication number
BG108683A
BG108683A BG108683A BG10868304A BG108683A BG 108683 A BG108683 A BG 108683A BG 108683 A BG108683 A BG 108683A BG 10868304 A BG10868304 A BG 10868304A BG 108683 A BG108683 A BG 108683A
Authority
BG
Bulgaria
Prior art keywords
preparing
processes
muscarinic receptor
receptor inhibitors
quinuclidine derivatives
Prior art date
Application number
BG108683A
Other languages
Bulgarian (bg)
English (en)
Inventor
Michel Guyaux
Chimmanamada Dinesh
Charles Mioskowski
Luc Quere
Jean-Philippe Starck
Patrice Talaga
Alain Wagner
Matteo ZANDA
Original Assignee
Ucb S.A.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ucb S.A. filed Critical Ucb S.A.
Publication of BG108683A publication Critical patent/BG108683A/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D453/00—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
    • C07D453/02—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Anesthesiology (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Urology & Nephrology (AREA)
  • Pulmonology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
BG108683A 2001-10-17 2004-04-15 Quinuclidine derivatives, processes for preparing them and their uses as m2 and/or m3 muscarinic receptor inhibitors BG108683A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP01124727 2001-10-17

Publications (1)

Publication Number Publication Date
BG108683A true BG108683A (en) 2005-04-30

Family

ID=8178984

Family Applications (1)

Application Number Title Priority Date Filing Date
BG108683A BG108683A (en) 2001-10-17 2004-04-15 Quinuclidine derivatives, processes for preparing them and their uses as m2 and/or m3 muscarinic receptor inhibitors

Country Status (19)

Country Link
US (1) US7361668B2 (hu)
EP (1) EP1438309A1 (hu)
JP (1) JP2005512974A (hu)
KR (1) KR20050030169A (hu)
CN (1) CN1571787A (hu)
BG (1) BG108683A (hu)
BR (1) BR0212983A (hu)
CA (1) CA2462980A1 (hu)
CZ (1) CZ2004501A3 (hu)
HU (1) HUP0401849A3 (hu)
IL (1) IL160896A0 (hu)
IS (1) IS7186A (hu)
MX (1) MXPA04002983A (hu)
NO (1) NO20042023L (hu)
NZ (1) NZ532283A (hu)
PL (1) PL370087A1 (hu)
RU (1) RU2004110717A (hu)
WO (1) WO2003033495A1 (hu)
ZA (1) ZA200402060B (hu)

Families Citing this family (76)

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US8883819B2 (en) 2011-09-01 2014-11-11 Irm Llc Bicyclic heterocycle derivatives for the treatment of pulmonary arterial hypertension
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WO2013038390A1 (en) 2011-09-16 2013-03-21 Novartis Ag N-substituted heterocyclyl carboxamides
ES2558457T3 (es) 2011-09-16 2016-02-04 Novartis Ag Compuestos heterocíclicos para el tratamiento de fibrosis quística
WO2013038378A1 (en) 2011-09-16 2013-03-21 Novartis Ag Pyridine amide derivatives
US9174994B2 (en) 2011-11-23 2015-11-03 Intellikine, Llc Enhanced treatment regimens using mTor inhibitors
US8809340B2 (en) 2012-03-19 2014-08-19 Novartis Ag Crystalline form
CN104245701A (zh) 2012-04-03 2014-12-24 诺华有限公司 有酪氨酸激酶抑制剂的组合产品和其应用
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Also Published As

Publication number Publication date
KR20050030169A (ko) 2005-03-29
IL160896A0 (en) 2004-08-31
JP2005512974A (ja) 2005-05-12
US20050020660A1 (en) 2005-01-27
HUP0401849A2 (hu) 2004-12-28
US7361668B2 (en) 2008-04-22
BR0212983A (pt) 2004-10-13
IS7186A (is) 2004-03-18
NO20042023L (no) 2004-05-14
EP1438309A1 (en) 2004-07-21
CA2462980A1 (en) 2003-04-24
PL370087A1 (en) 2005-05-16
ZA200402060B (en) 2005-03-15
CZ2004501A3 (cs) 2004-09-15
WO2003033495A1 (en) 2003-04-24
MXPA04002983A (es) 2004-07-15
NZ532283A (en) 2005-06-24
HUP0401849A3 (en) 2007-05-02
CN1571787A (zh) 2005-01-26
RU2004110717A (ru) 2005-10-20

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