EA200600787A1 - Антагонисты мускариновых ацетилхолиновых рецепторов - Google Patents

Антагонисты мускариновых ацетилхолиновых рецепторов

Info

Publication number
EA200600787A1
EA200600787A1 EA200600787A EA200600787A EA200600787A1 EA 200600787 A1 EA200600787 A1 EA 200600787A1 EA 200600787 A EA200600787 A EA 200600787A EA 200600787 A EA200600787 A EA 200600787A EA 200600787 A1 EA200600787 A1 EA 200600787A1
Authority
EA
Eurasian Patent Office
Prior art keywords
antagonists
muscarine
acetyl choline
choline receptors
receptors
Prior art date
Application number
EA200600787A
Other languages
English (en)
Inventor
Майкл Р. Палович
Цзехун Вань
Чунцзе Чжу
Original Assignee
Глэксо Груп Лимитед
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Глэксо Груп Лимитед filed Critical Глэксо Груп Лимитед
Publication of EA200600787A1 publication Critical patent/EA200600787A1/ru

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D451/00—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
    • C07D451/02—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/02—Nasal agents, e.g. decongestants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/08—Bronchodilators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Abstract

Описаны антагонисты мускариновых ацетилхолиновых рецепторов и способы их использования.
EA200600787A 2003-10-17 2004-10-15 Антагонисты мускариновых ацетилхолиновых рецепторов EA200600787A1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US51216103P 2003-10-17 2003-10-17
PCT/US2004/034234 WO2005037224A2 (en) 2003-10-17 2004-10-15 Muscarinic acetylcholine receptor antagonists

Publications (1)

Publication Number Publication Date
EA200600787A1 true EA200600787A1 (ru) 2006-08-25

Family

ID=34465319

Family Applications (1)

Application Number Title Priority Date Filing Date
EA200600787A EA200600787A1 (ru) 2003-10-17 2004-10-15 Антагонисты мускариновых ацетилхолиновых рецепторов

Country Status (22)

Country Link
US (1) US7507747B2 (ru)
EP (1) EP1677796A4 (ru)
JP (1) JP2007509061A (ru)
CN (1) CN1897947A (ru)
AP (1) AP2006003575A0 (ru)
AR (1) AR046114A1 (ru)
AU (1) AU2004281167A1 (ru)
BR (1) BRPI0415281A (ru)
CA (1) CA2542636A1 (ru)
EA (1) EA200600787A1 (ru)
EC (1) ECSP066486A (ru)
IL (1) IL174846A0 (ru)
IS (1) IS8440A (ru)
MA (1) MA28109A1 (ru)
MX (1) MXPA06004242A (ru)
NO (1) NO20062071L (ru)
OA (1) OA13270A (ru)
PE (1) PE20050442A1 (ru)
TW (1) TW200528448A (ru)
UY (1) UY28567A1 (ru)
WO (1) WO2005037224A2 (ru)
ZA (1) ZA200602783B (ru)

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PE20050250A1 (es) * 2003-07-17 2005-04-08 Glaxo Group Ltd Antagonistas de los receptores muscarinicos de la acetilcolina
TW200524577A (en) * 2003-11-04 2005-08-01 Glaxo Group Ltd Muscarinic acetylcholine receptor antagonists
US20090253908A1 (en) * 2004-03-11 2009-10-08 Glaxo Group Limited Novel m3 muscarinic acetylchoine receptor antagonists
EP1725564A4 (en) * 2004-03-17 2007-09-12 Glaxo Group Ltd ANTAGONISTS OF THE M3 MUSCARIN ACETYL CHOLIN RECEPTOR
EP1725238A4 (en) * 2004-03-17 2009-04-01 Glaxo Group Ltd ACETYLCHOLINE M 3 MUSCARINIC RECEPTOR ANTAGONISTS
AR050902A1 (es) 2004-04-27 2006-12-06 Glaxo Group Ltd Compuesto de quinuclidina, composicion farmaceutica que lo comprende y su usopara preparar dicha composicion
EP1747219A4 (en) * 2004-05-13 2010-05-26 Glaxo Group Ltd Antagonists of muscarinic acetylcholine receptor
EP1957075A4 (en) * 2004-11-15 2009-11-18 Glaxo Group Ltd NOVEL ANTAGONISTS OF ACETYLCHOLINE M3 TYPE MUSCARINIC RECEPTORS
WO2007016639A2 (en) * 2005-08-02 2007-02-08 Glaxo Group Limited M3 muscarinic acetylcholine receptor antagonists
WO2007022351A2 (en) * 2005-08-18 2007-02-22 Glaxo Group Limited Muscarinic acetylcholine receptor antagonists
TW200946526A (en) 2008-02-06 2009-11-16 Glaxo Group Ltd Dual pharmacophores-PDE4-muscarinic antagonistics
UY31636A1 (es) 2008-02-06 2009-08-03 Farmacoforos duales-antagonistas muscarinicos de pde4
UY31637A1 (es) 2008-02-06 2009-08-03 Farmacoforos duales-antagonistas muscarinicos de pde4
WO2010094643A1 (en) 2009-02-17 2010-08-26 Glaxo Group Limited Quinoline derivatives and their uses for rhinitis and urticaria

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EP1725238A4 (en) 2004-03-17 2009-04-01 Glaxo Group Ltd ACETYLCHOLINE M 3 MUSCARINIC RECEPTOR ANTAGONISTS
AR050902A1 (es) 2004-04-27 2006-12-06 Glaxo Group Ltd Compuesto de quinuclidina, composicion farmaceutica que lo comprende y su usopara preparar dicha composicion
EP1747219A4 (en) 2004-05-13 2010-05-26 Glaxo Group Ltd Antagonists of muscarinic acetylcholine receptor
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Also Published As

Publication number Publication date
AU2004281167A1 (en) 2005-04-28
CN1897947A (zh) 2007-01-17
US7507747B2 (en) 2009-03-24
CA2542636A1 (en) 2005-04-28
BRPI0415281A (pt) 2006-12-19
TW200528448A (en) 2005-09-01
MA28109A1 (fr) 2006-08-01
EP1677796A2 (en) 2006-07-12
NO20062071L (no) 2006-05-08
IS8440A (is) 2006-05-05
ECSP066486A (es) 2006-10-10
WO2005037224A2 (en) 2005-04-28
UY28567A1 (es) 2005-05-31
ZA200602783B (en) 2007-11-28
JP2007509061A (ja) 2007-04-12
OA13270A (en) 2007-01-31
PE20050442A1 (es) 2005-07-09
EP1677796A4 (en) 2006-12-27
AP2006003575A0 (en) 2006-04-30
WO2005037224A3 (en) 2005-06-23
AR046114A1 (es) 2005-11-23
IL174846A0 (en) 2006-08-20
US20070135478A1 (en) 2007-06-14
MXPA06004242A (es) 2006-06-28

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