BG107653A - Спиро-пиримидин - 2,4,6-трионови инхибитори на металопротеиназa - Google Patents
Спиро-пиримидин - 2,4,6-трионови инхибитори на металопротеиназa Download PDFInfo
- Publication number
- BG107653A BG107653A BG107653A BG10765303A BG107653A BG 107653 A BG107653 A BG 107653A BG 107653 A BG107653 A BG 107653A BG 10765303 A BG10765303 A BG 10765303A BG 107653 A BG107653 A BG 107653A
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- Prior art keywords
- alkyl
- pyridin
- group
- compound
- formula
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/10—Spiro-condensed systems
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- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/10—Spiro-condensed systems
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- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
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- Public Health (AREA)
- Engineering & Computer Science (AREA)
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- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Immunology (AREA)
- Physical Education & Sports Medicine (AREA)
- Endocrinology (AREA)
- Reproductive Health (AREA)
- Oncology (AREA)
- Rheumatology (AREA)
- Communicable Diseases (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Dermatology (AREA)
- Pain & Pain Management (AREA)
- Pulmonology (AREA)
- Gynecology & Obstetrics (AREA)
- Diabetes (AREA)
- Heart & Thoracic Surgery (AREA)
- Ophthalmology & Optometry (AREA)
- Tropical Medicine & Parasitology (AREA)
- Cardiology (AREA)
- Pregnancy & Childbirth (AREA)
- Hematology (AREA)
- Virology (AREA)
- Obesity (AREA)
- Psychology (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US24338900P | 2000-10-26 | 2000-10-26 | |
| PCT/IB2001/001986 WO2002034753A2 (en) | 2000-10-26 | 2001-10-23 | Spiro-pyrimidine-2,4,6-trione metalloproteinase inhibitors |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BG107653A true BG107653A (bg) | 2003-12-31 |
Family
ID=22918584
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BG107653A BG107653A (bg) | 2000-10-26 | 2003-03-20 | Спиро-пиримидин - 2,4,6-трионови инхибитори на металопротеиназa |
Country Status (32)
| Country | Link |
|---|---|
| EP (1) | EP1332146A2 (sk) |
| JP (1) | JP2004518635A (sk) |
| KR (1) | KR20040004412A (sk) |
| CN (1) | CN1501937A (sk) |
| AP (1) | AP2001002318A0 (sk) |
| AR (1) | AR035069A1 (sk) |
| AU (1) | AU2002210813A1 (sk) |
| BG (1) | BG107653A (sk) |
| BR (1) | BR0114913A (sk) |
| CA (1) | CA2425283A1 (sk) |
| CZ (1) | CZ20031083A3 (sk) |
| EA (1) | EA005762B1 (sk) |
| EC (1) | ECSP034567A (sk) |
| EE (1) | EE200300196A (sk) |
| GT (1) | GT200100213A (sk) |
| HN (1) | HN2001000244A (sk) |
| HR (1) | HRP20030332A2 (sk) |
| HU (1) | HUP0301577A3 (sk) |
| IL (1) | IL154948A0 (sk) |
| IS (1) | IS6762A (sk) |
| MA (1) | MA26957A1 (sk) |
| MX (1) | MXPA03003735A (sk) |
| NO (1) | NO20031853L (sk) |
| OA (1) | OA12529A (sk) |
| PA (1) | PA8531401A1 (sk) |
| PE (1) | PE20020589A1 (sk) |
| PL (1) | PL366201A1 (sk) |
| SK (1) | SK4972003A3 (sk) |
| SV (1) | SV2003000705A (sk) |
| TN (1) | TNSN01149A1 (sk) |
| WO (1) | WO2002034753A2 (sk) |
| ZA (1) | ZA200302190B (sk) |
Families Citing this family (36)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DOP2002000332A (es) | 2001-02-14 | 2002-08-30 | Warner Lambert Co | Inhibidores de piridina de metaloproteinasas de la matriz |
| DOP2002000333A (es) | 2001-02-14 | 2002-09-30 | Warner Lambert Co | Derivados de acido isoftalico como inhibidores de metaloproteinasas de la matriz |
| EP1368323B1 (en) | 2001-02-14 | 2010-06-30 | Warner-Lambert Company LLC | Pyrimidine matrix metalloproteinase inhibitors |
| PA8539501A1 (es) | 2001-02-14 | 2002-09-30 | Warner Lambert Co | Compuestos triazolo como inhibidores de mmp |
| ES2231708T3 (es) | 2001-02-14 | 2005-05-16 | Warner-Lambert Company Llc | Benzotiadicinas inhibidoras de metaloproteinasa de matriz. |
| US6924276B2 (en) | 2001-09-10 | 2005-08-02 | Warner-Lambert Company | Diacid-substituted heteroaryl derivatives as matrix metalloproteinase inhibitors |
| WO2003032999A1 (en) | 2001-10-12 | 2003-04-24 | Warner-Lambert Company Llc | Alkyne matrix metalloproteinase inhibitors |
| US6962922B2 (en) | 2001-10-12 | 2005-11-08 | Warner-Lambert Company Llc | Alkynylated quinazoline compounds |
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2001
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- 2001-10-23 IL IL15494801A patent/IL154948A0/xx unknown
- 2001-10-23 WO PCT/IB2001/001986 patent/WO2002034753A2/en not_active Application Discontinuation
- 2001-10-23 EA EA200300306A patent/EA005762B1/ru not_active IP Right Cessation
- 2001-10-23 HU HU0301577A patent/HUP0301577A3/hu unknown
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- 2001-10-23 BR BR0114913-0A patent/BR0114913A/pt not_active IP Right Cessation
- 2001-10-23 JP JP2002537743A patent/JP2004518635A/ja not_active Withdrawn
- 2001-10-23 CN CNA018179231A patent/CN1501937A/zh active Pending
- 2001-10-23 EP EP01978721A patent/EP1332146A2/en not_active Withdrawn
- 2001-10-23 AU AU2002210813A patent/AU2002210813A1/en not_active Abandoned
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- 2001-10-23 KR KR10-2003-7005753A patent/KR20040004412A/ko not_active Application Discontinuation
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- 2001-10-25 TN TNTNSN01149A patent/TNSN01149A1/fr unknown
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