BG106846A - Novel heteroaryl derivatives, their preparation and use - Google Patents

Novel heteroaryl derivatives, their preparation and use

Info

Publication number
BG106846A
BG106846A BG106846A BG10684602A BG106846A BG 106846 A BG106846 A BG 106846A BG 106846 A BG106846 A BG 106846A BG 10684602 A BG10684602 A BG 10684602A BG 106846 A BG106846 A BG 106846A
Authority
BG
Bulgaria
Prior art keywords
cr6r7
heteroaryl derivatives
preparation
disorders
compulsive
Prior art date
Application number
BG106846A
Other languages
Bulgarian (bg)
English (en)
Inventor
Thomas Ruhland
- JENSEN Christian KROG
Ivan Mikkelsen
Mario Rottlaender
Gitte Mikkelsen
Ejner Moltzen
Kim Andersen
Original Assignee
H. Lundbeck A/S
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by H. Lundbeck A/S filed Critical H. Lundbeck A/S
Publication of BG106846A publication Critical patent/BG106846A/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/78—Benzo [b] furans; Hydrogenated benzo [b] furans
    • C07D307/79—Benzo [b] furans; Hydrogenated benzo [b] furans with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D319/00—Heterocyclic compounds containing six-membered rings having two oxygen atoms as the only ring hetero atoms
    • C07D319/10—1,4-Dioxanes; Hydrogenated 1,4-dioxanes
    • C07D319/14—1,4-Dioxanes; Hydrogenated 1,4-dioxanes condensed with carbocyclic rings or ring systems
    • C07D319/16—1,4-Dioxanes; Hydrogenated 1,4-dioxanes condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • C07D319/18—Ethylenedioxybenzenes, not substituted on the hetero ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D333/52—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
    • C07D333/54—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Psychiatry (AREA)
  • Hospice & Palliative Care (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Compounds That Contain Two Or More Ring Oxygen Atoms (AREA)
BG106846A 1999-12-30 2002-06-19 Novel heteroaryl derivatives, their preparation and use BG106846A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DKPA199901884 1999-12-30
PCT/DK2000/000741 WO2001049683A1 (en) 1999-12-30 2000-12-29 Novel heteroaryl derivatives, their preparation and use

Publications (1)

Publication Number Publication Date
BG106846A true BG106846A (en) 2003-02-28

Family

ID=8108797

Family Applications (1)

Application Number Title Priority Date Filing Date
BG106846A BG106846A (en) 1999-12-30 2002-06-19 Novel heteroaryl derivatives, their preparation and use

Country Status (22)

Country Link
US (1) US20030050306A1 (is)
EP (1) EP1246820A1 (is)
JP (1) JP2003519229A (is)
KR (1) KR20020063286A (is)
CN (1) CN1414963A (is)
AR (1) AR027133A1 (is)
AU (1) AU2352001A (is)
BG (1) BG106846A (is)
BR (1) BR0016954A (is)
CA (1) CA2395984A1 (is)
CZ (1) CZ20022280A3 (is)
EA (1) EA200200733A1 (is)
HU (1) HUP0204084A3 (is)
IL (1) IL149993A0 (is)
IS (1) IS6403A (is)
NO (1) NO20023188L (is)
NZ (1) NZ519478A (is)
PL (1) PL355610A1 (is)
SK (1) SK9432002A3 (is)
TR (1) TR200201679T2 (is)
WO (1) WO2001049683A1 (is)
ZA (1) ZA200204464B (is)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP5080716B2 (ja) 2001-07-20 2012-11-21 サイコジェニックス・インコーポレーテッド 注意欠陥・多動性障害の治療
TWI320783B (en) 2005-04-14 2010-02-21 Otsuka Pharma Co Ltd Heterocyclic compound
AR055203A1 (es) * 2005-08-31 2007-08-08 Otsuka Pharma Co Ltd Derivados de benzotiofeno con propiedades antipsicoticas
WO2008024724A1 (en) 2006-08-21 2008-02-28 Genentech, Inc. Aza-benzothiophenyl compounds and methods of use
JP4785881B2 (ja) * 2007-02-27 2011-10-05 大塚製薬株式会社 医薬

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK148392D0 (da) * 1992-12-09 1992-12-09 Lundbeck & Co As H Heterocykliske forbindelser
IT1266582B1 (it) * 1993-07-30 1997-01-09 Recordati Chem Pharm Derivati (di)azacicloesanici e diazacicloeptanici
AR022303A1 (es) * 1999-01-22 2002-09-04 Lundbeck & Co As H Derivados de piperidina, tetrahidropiridina y piperazina, su preparacion y utilizacion

Also Published As

Publication number Publication date
AU2352001A (en) 2001-07-16
AR027133A1 (es) 2003-03-12
KR20020063286A (ko) 2002-08-01
EP1246820A1 (en) 2002-10-09
CZ20022280A3 (cs) 2002-10-16
TR200201679T2 (tr) 2002-10-21
NO20023188D0 (no) 2002-07-01
ZA200204464B (en) 2003-09-04
PL355610A1 (en) 2004-05-04
CN1414963A (zh) 2003-04-30
JP2003519229A (ja) 2003-06-17
HUP0204084A2 (hu) 2003-03-28
US20030050306A1 (en) 2003-03-13
IS6403A (is) 2002-05-31
SK9432002A3 (en) 2002-11-06
HUP0204084A3 (en) 2005-02-28
IL149993A0 (en) 2002-12-01
NO20023188L (no) 2002-07-01
WO2001049683A1 (en) 2001-07-12
CA2395984A1 (en) 2001-07-12
EA200200733A1 (ru) 2002-12-26
BR0016954A (pt) 2003-04-29
NZ519478A (en) 2004-02-27

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