BG104877A - N-заместени аминотетралини като лиганди за невропептиден y y5 рецептор, използвани при лечение на напълняване и други смущения - Google Patents

N-заместени аминотетралини като лиганди за невропептиден y y5 рецептор, използвани при лечение на напълняване и други смущения

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Publication number
BG104877A
BG104877A BG104877A BG10487700A BG104877A BG 104877 A BG104877 A BG 104877A BG 104877 A BG104877 A BG 104877A BG 10487700 A BG10487700 A BG 10487700A BG 104877 A BG104877 A BG 104877A
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Bulgaria
Prior art keywords
neuropeptide
ligands
disorders
treatment
anminotetralins
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BG104877A
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English (en)
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BG64732B1 (bg
Inventor
Scott Dax
Timothy Lovenberg
James Mcnally
Allen Reitz
Mark Youngman
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Ortho-Mcneil Pharmaceutical, Inc.
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Application filed by Ortho-Mcneil Pharmaceutical, Inc. filed Critical Ortho-Mcneil Pharmaceutical, Inc.
Publication of BG104877A publication Critical patent/BG104877A/bg
Publication of BG64732B1 publication Critical patent/BG64732B1/bg

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Abstract

Изобретението се отнася до производни на бета-аминотетралин с формула@@които са лиганди за невропептиден Y Y5 (NPY5) рецептор, до методи за получаване и фармацевтични състави, съдържащи производно набета-аминотетралин като активна съставна част. Бета-аминотетралините се използват при лечение на състояния и заболявания, свързани с NPY рецептор, подвид Y5.
BG104877A 1998-04-29 2000-10-23 N-заместени аминотетралини като лиганди за невропептиден y y5 рецептор, използвани при лечение на напълняване и други смущения BG64732B1 (bg)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US8341598P 1998-04-29 1998-04-29
US09/290,651 US6140354A (en) 1998-04-29 1999-04-12 N-substituted aminotetralins as ligands for the neuropeptide Y Y5 receptor useful in the treatment of obesity and other disorders

Publications (2)

Publication Number Publication Date
BG104877A true BG104877A (bg) 2001-06-29
BG64732B1 BG64732B1 (bg) 2006-01-31

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BG104877A BG64732B1 (bg) 1998-04-29 2000-10-23 N-заместени аминотетралини като лиганди за невропептиден y y5 рецептор, използвани при лечение на напълняване и други смущения

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US (1) US6140354A (bg)
EP (1) EP1076644B1 (bg)
JP (1) JP2004503462A (bg)
CN (1) CN1289475C (bg)
AT (1) ATE269846T1 (bg)
AU (1) AU759313B2 (bg)
BG (1) BG64732B1 (bg)
BR (1) BR9910583A (bg)
DE (1) DE69918296T2 (bg)
DK (1) DK1076644T3 (bg)
ES (1) ES2223170T3 (bg)
HU (1) HUP0102656A3 (bg)
ID (1) ID26128A (bg)
IL (1) IL139227A0 (bg)
NZ (1) NZ507763A (bg)
PL (1) PL194839B1 (bg)
PT (1) PT1076644E (bg)
RO (1) RO120542B1 (bg)
RU (1) RU2219167C2 (bg)
TR (1) TR200100137T2 (bg)
TW (1) TW530043B (bg)
WO (1) WO1999055667A1 (bg)
ZA (1) ZA992951B (bg)

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