BG101112A - Използване на хетероциклени съединения - Google Patents

Използване на хетероциклени съединения

Info

Publication number
BG101112A
BG101112A BG101112A BG10111297A BG101112A BG 101112 A BG101112 A BG 101112A BG 101112 A BG101112 A BG 101112A BG 10111297 A BG10111297 A BG 10111297A BG 101112 A BG101112 A BG 101112A
Authority
BG
Bulgaria
Prior art keywords
heterocyclic compounds
het
heterocyclic
compounds
todiopamin
Prior art date
Application number
BG101112A
Other languages
English (en)
Other versions
BG63487B1 (bg
Inventor
Beate Hellendahl
Annegret Lansky
Beatrice Rendenbach-Mueller
Alfred Bach
Liliane Unger
Hans-Juergen Teschendorf
Carsten Wicke
Original Assignee
Abbott Gmbh & Co. Kg
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Abbott Gmbh & Co. Kg filed Critical Abbott Gmbh & Co. Kg
Publication of BG101112A publication Critical patent/BG101112A/bg
Publication of BG63487B1 publication Critical patent/BG63487B1/bg

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/26—Psychostimulants, e.g. nicotine, cocaine

Landscapes

  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Biomedical Technology (AREA)
  • Psychiatry (AREA)
  • Anesthesiology (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)

Abstract

Изобретението се отнася до използването на хетероциклени съединения с формула Het-A-Ar, в която Het, A, B и Ar имат значенията, посочени в описанието. Съединенията имат висок афинитет към допамин-D3-рецепторите и поради това се използват за лечение на заболявания, които реагират на допамин-D3-лиганди.
BG101112A 1994-07-15 1997-01-06 Използване на хетероциклени съединения BG63487B1 (bg)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE4425146A DE4425146A1 (de) 1994-07-15 1994-07-15 Verwendung heterocyclischer Verbindungen
PCT/EP1995/002782 WO1996002246A1 (de) 1994-07-15 1995-07-14 Verwendung heterocyclischer verbindungen als dopamin-d3 liganden

Publications (2)

Publication Number Publication Date
BG101112A true BG101112A (bg) 1998-04-30
BG63487B1 BG63487B1 (bg) 2002-03-29

Family

ID=6523325

Family Applications (1)

Application Number Title Priority Date Filing Date
BG101112A BG63487B1 (bg) 1994-07-15 1997-01-06 Използване на хетероциклени съединения

Country Status (22)

Country Link
US (1) US6090807A (bg)
EP (1) EP0771197B1 (bg)
JP (1) JPH10502658A (bg)
KR (2) KR100443850B1 (bg)
CN (2) CN1534023A (bg)
AT (1) ATE236629T1 (bg)
AU (1) AU704839B2 (bg)
BG (1) BG63487B1 (bg)
BR (1) BR9508296A (bg)
CA (1) CA2195242A1 (bg)
CZ (1) CZ293126B6 (bg)
DE (2) DE4425146A1 (bg)
DK (1) DK0771197T3 (bg)
ES (1) ES2196072T3 (bg)
FI (1) FI970148A0 (bg)
HU (1) HUT77608A (bg)
MX (1) MX9700430A (bg)
NO (1) NO311683B1 (bg)
NZ (1) NZ290388A (bg)
PT (1) PT771197E (bg)
SI (1) SI9520084B (bg)
WO (1) WO1996002246A1 (bg)

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DE10358004A1 (de) 2003-12-11 2005-07-14 Abbott Gmbh & Co. Kg Ketolactam-Verbindungen und ihre Verwendung
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JP4904267B2 (ja) 2004-08-09 2012-03-28 アボット ゲーエムベーハー ウント カンパニー カーゲー ドーパミンｄ３受容体の調節に応答する障害の治療に好適な４−ピペラジニル−ピリミジン化合物
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Also Published As

Publication number Publication date
NZ290388A (en) 2001-04-27
KR970704435A (ko) 1997-09-06
ATE236629T1 (de) 2003-04-15
BG63487B1 (bg) 2002-03-29
FI970148A (fi) 1997-01-14
CZ9697A3 (en) 1997-08-13
KR100443850B1 (ko) 2004-08-11
NO311683B1 (no) 2002-01-07
US6090807A (en) 2000-07-18
HUT77608A (hu) 1998-06-29
WO1996002246A1 (de) 1996-02-01
FI970148A0 (fi) 1997-01-14
AU704839B2 (en) 1999-05-06
KR20040000412A (ko) 2004-01-03
MX9700430A (es) 1998-05-31
DE4425146A1 (de) 1996-01-18
NO970163L (no) 1997-03-14
SI9520084A (en) 1997-08-31
BR9508296A (pt) 1998-05-19
CA2195242A1 (en) 1996-02-01
DK0771197T3 (da) 2003-06-23
CZ293126B6 (cs) 2004-02-18
PT771197E (pt) 2003-08-29
JPH10502658A (ja) 1998-03-10
SI9520084B (sl) 2005-02-28
CN1534023A (zh) 2004-10-06
AU3111495A (en) 1996-02-16
EP0771197A1 (de) 1997-05-07
DE59510635D1 (de) 2003-05-15
NO970163D0 (no) 1997-01-14
ES2196072T3 (es) 2003-12-16
CN1152870A (zh) 1997-06-25
EP0771197B1 (de) 2003-04-09
HU9700111D0 (en) 1997-02-28

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