BE871807A - 4-quinolyl-guanidines, leur preparation et leur utilisation - Google Patents

4-quinolyl-guanidines, leur preparation et leur utilisation

Info

Publication number
BE871807A
BE871807A BE191566A BE191566A BE871807A BE 871807 A BE871807 A BE 871807A BE 191566 A BE191566 A BE 191566A BE 191566 A BE191566 A BE 191566A BE 871807 A BE871807 A BE 871807A
Authority
BE
Belgium
Prior art keywords
guanidines
quinolyl
preparation
Prior art date
Application number
BE191566A
Other languages
English (en)
French (fr)
Original Assignee
Leo Pharm Prod Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Leo Pharm Prod Ltd filed Critical Leo Pharm Prod Ltd
Publication of BE871807A publication Critical patent/BE871807A/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D215/00Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/38Nitrogen atoms
    • C07D215/42Nitrogen atoms attached in position 4
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pain & Pain Management (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
BE191566A 1977-11-07 1978-11-06 4-quinolyl-guanidines, leur preparation et leur utilisation BE871807A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB4616677 1977-11-07

Publications (1)

Publication Number Publication Date
BE871807A true BE871807A (fr) 1979-05-07

Family

ID=10440127

Family Applications (1)

Application Number Title Priority Date Filing Date
BE191566A BE871807A (fr) 1977-11-07 1978-11-06 4-quinolyl-guanidines, leur preparation et leur utilisation

Country Status (24)

Country Link
US (1) US4293549A (xx)
JP (1) JPS5473784A (xx)
AT (1) AT366368B (xx)
AU (1) AU517670B2 (xx)
BE (1) BE871807A (xx)
CA (1) CA1120929A (xx)
CH (1) CH645354A5 (xx)
DE (1) DE2847792A1 (xx)
DK (1) DK153950C (xx)
ES (1) ES474900A1 (xx)
FI (1) FI69463C (xx)
FR (1) FR2407930A1 (xx)
GR (1) GR65010B (xx)
IE (1) IE47458B1 (xx)
IT (1) IT1100075B (xx)
LU (1) LU80476A1 (xx)
NL (1) NL7811035A (xx)
NZ (1) NZ188770A (xx)
PH (1) PH16296A (xx)
PT (1) PT68750A (xx)
SE (1) SE446267B (xx)
SU (1) SU828967A3 (xx)
YU (1) YU41129B (xx)
ZA (1) ZA786175B (xx)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6306846B1 (en) * 1972-05-31 2001-10-23 John R. J. Sorenson Anti-inflammatory and anti-ulcer compounds and process
IT1205640B (it) * 1983-04-06 1989-03-23 Yason Srl Nuovi composti ad attivita' antiinfiammatoria,procedimento per la loro preparazione e composizioni farmaceutiche che li contengono
US4563460A (en) * 1984-01-13 1986-01-07 William H. Rorer, Inc. Quinoline and quinazoline derivatives for treating gastrointestinal motility dysfunctions
HU195487B (en) * 1985-06-04 1988-05-30 Egyt Gyogyszervegyeszeti Gyar Process for producing quinoline derivatives
ATE66477T1 (de) * 1986-08-29 1991-09-15 Pfizer 2-guanidino-4-aryl-thiazole fuer die behandlung von peptischen geschwueren.
US6100260A (en) * 1997-04-21 2000-08-08 Sumitomo Pharmaceutical Company, Limited Isoxazole derivatives
EP0928793B1 (en) * 1998-01-02 2002-05-15 F. Hoffmann-La Roche Ag Thiazole derivatives
RU2202344C2 (ru) 1998-03-26 2003-04-20 Джапан Тобакко Инк. Антагонисты ноцицептина, производные амида, аналгетик, способ инициирования антагонистического действия к ноцицептину, способ лечения боли, фармацевтические композиции
WO2001032604A1 (en) * 1999-11-05 2001-05-10 University College London Activators of soluble guanylate cyclase
US7186725B2 (en) * 2003-01-03 2007-03-06 Genzyme Corporation Anti-inflammatory compositions and methods
WO2004064730A2 (en) * 2003-01-14 2004-08-05 Cytokinetics, Inc. Compounds, compositions and methods
GB0404434D0 (en) 2004-02-27 2004-03-31 Novartis Ag Organic compounds
EP1917244A2 (de) * 2005-08-24 2008-05-07 Abbott GmbH & Co. KG Hetaryl substituierte guanidinverbindungen und ihre verwendung als bindungspartner für 5-ht5-rezeptoren
WO2023003497A1 (ru) * 2021-07-23 2023-01-26 Общество С Ограниченной Ответственностью "Валента-Интеллект" Соединения с лизосомотропной и противовирусной активностью

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB889282A (en) * 1957-05-07 1962-02-14 Air Reduction Preparation of hexafluorodiethyl ether and medicinal compositions containing it
GB889262A (en) * 1959-07-03 1962-02-14 Ciba Ltd Quinoline compounds
US3159676A (en) * 1962-02-07 1964-12-01 Smith Kline French Lab Naphthyl containing guanidines
US3852293A (en) 1972-06-21 1974-12-03 Uniroyal Inc 4-phenyl-2-(3-pyridyl)-thiazole carboxamides
US4000279A (en) * 1974-10-29 1976-12-28 Armour Pharmaceutical Company Pharmaceutical preparations containing 5'-(8'-hydroxyquinolyl)guanidine compounds and methods of using same

Also Published As

Publication number Publication date
DK153950C (da) 1989-02-20
CA1120929A (en) 1982-03-30
IT1100075B (it) 1985-09-28
ATA773278A (de) 1981-08-15
US4293549A (en) 1981-10-06
PT68750A (en) 1978-12-01
JPS5473784A (en) 1979-06-13
IT7829514A0 (it) 1978-11-07
CH645354A5 (de) 1984-09-28
FR2407930B1 (xx) 1983-03-18
YU41129B (en) 1986-12-31
GR65010B (en) 1980-06-12
FI69463B (fi) 1985-10-31
AT366368B (de) 1982-04-13
FI69463C (fi) 1986-02-10
JPS6348873B2 (xx) 1988-09-30
YU257578A (en) 1983-01-21
SU828967A3 (ru) 1981-05-07
FR2407930A1 (fr) 1979-06-01
DE2847792C2 (xx) 1988-02-04
SE7811457L (sv) 1979-05-08
AU517670B2 (en) 1981-08-20
NZ188770A (en) 1984-07-31
FI783327A (fi) 1979-05-08
PH16296A (en) 1983-09-05
DK153950B (da) 1988-09-26
ZA786175B (en) 1979-10-31
LU80476A1 (fr) 1979-06-15
NL7811035A (nl) 1979-05-09
IE782084L (en) 1979-05-07
DE2847792A1 (de) 1979-05-10
ES474900A1 (es) 1980-04-16
IE47458B1 (en) 1984-03-21
DK493378A (da) 1979-05-08
AU4137678A (en) 1979-05-17
SE446267B (sv) 1986-08-25

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Legal Events

Date Code Title Description
RE Patent lapsed

Owner name: LEO PHARMACEUTICAL PRODUCTS LTD A/S (LOVENS KEMIS

Effective date: 19921130