BE830766A - Nouvelles cetones aromatiques douees d'activites cardiovasculaires - Google Patents

Nouvelles cetones aromatiques douees d'activites cardiovasculaires

Info

Publication number
BE830766A
BE830766A BE157788A BE157788A BE830766A BE 830766 A BE830766 A BE 830766A BE 157788 A BE157788 A BE 157788A BE 157788 A BE157788 A BE 157788A BE 830766 A BE830766 A BE 830766A
Authority
BE
Belgium
Prior art keywords
enhanced
aromatic ketones
new aromatic
cardiovascular activities
cardiovascular
Prior art date
Application number
BE157788A
Other languages
English (en)
French (fr)
Inventor
H Demarne
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Publication of BE830766A publication Critical patent/BE830766A/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D303/00Compounds containing three-membered rings having one oxygen atom as the only ring hetero atom
    • C07D303/02Compounds containing oxirane rings
    • C07D303/12Compounds containing oxirane rings with hydrocarbon radicals, substituted by singly or doubly bound oxygen atoms
    • C07D303/18Compounds containing oxirane rings with hydrocarbon radicals, substituted by singly or doubly bound oxygen atoms by etherified hydroxyl radicals
    • C07D303/20Ethers with hydroxy compounds containing no oxirane rings
    • C07D303/22Ethers with hydroxy compounds containing no oxirane rings with monohydroxy compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/02Drugs for disorders of the nervous system for peripheral neuropathies
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
BE157788A 1974-06-28 1975-06-27 Nouvelles cetones aromatiques douees d'activites cardiovasculaires BE830766A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB28925/74A GB1501632A (en) 1974-06-28 1974-06-28 Aromatic ketones having cardiovascular activity

Publications (1)

Publication Number Publication Date
BE830766A true BE830766A (fr) 1975-12-29

Family

ID=10283421

Family Applications (1)

Application Number Title Priority Date Filing Date
BE157788A BE830766A (fr) 1974-06-28 1975-06-27 Nouvelles cetones aromatiques douees d'activites cardiovasculaires

Country Status (17)

Country Link
US (2) US4252825A (cg-RX-API-DMAC10.html)
JP (2) JPS5826743B2 (cg-RX-API-DMAC10.html)
AR (1) AR205388A1 (cg-RX-API-DMAC10.html)
AT (1) AT343098B (cg-RX-API-DMAC10.html)
BE (1) BE830766A (cg-RX-API-DMAC10.html)
CA (1) CA1052820A (cg-RX-API-DMAC10.html)
CS (1) CS197248B2 (cg-RX-API-DMAC10.html)
DE (1) DE2528147A1 (cg-RX-API-DMAC10.html)
DK (1) DK143555C (cg-RX-API-DMAC10.html)
ES (1) ES438931A1 (cg-RX-API-DMAC10.html)
FR (1) FR2276032A1 (cg-RX-API-DMAC10.html)
GB (1) GB1501632A (cg-RX-API-DMAC10.html)
IE (1) IE41386B1 (cg-RX-API-DMAC10.html)
NL (1) NL7507703A (cg-RX-API-DMAC10.html)
SE (2) SE416546B (cg-RX-API-DMAC10.html)
YU (1) YU165775A (cg-RX-API-DMAC10.html)
ZA (1) ZA754141B (cg-RX-API-DMAC10.html)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1501632A (en) * 1974-06-28 1978-02-22 Cm Ind Aromatic ketones having cardiovascular activity
JPH0516363Y2 (cg-RX-API-DMAC10.html) * 1986-08-01 1993-04-28
AU2003250483A1 (en) 2002-08-19 2004-03-11 Pfizer Products Inc. Combination therapy for hyperproliferative diseases
CA2526730A1 (en) * 2003-05-30 2004-12-09 Ranbaxy Laboratories Limited Substituted pyrrole derivatives
US20050037063A1 (en) * 2003-07-21 2005-02-17 Bolton Anthony E. Combined therapies
GT200600381A (es) 2005-08-25 2007-03-28 Compuestos organicos
US7741317B2 (en) 2005-10-21 2010-06-22 Bristol-Myers Squibb Company LXR modulators
BRPI0618379A2 (pt) * 2005-11-08 2011-08-30 Ranbaxy Lab Ltd processo para preparação do hemi-sal de cálcio do ácido (3r,5r) -7-[2-(4-fluorofenil)-5-isopropil-3-fenil-4-[(4-hidroxime tilfenilamino) carbonil]-pirrol-1-il] -3, 5-diidroxi heptanóico
US7888376B2 (en) 2005-11-23 2011-02-15 Bristol-Myers Squibb Company Heterocyclic CETP inhibitors
CL2007000667A1 (es) * 2006-03-14 2008-03-14 Ranbaxi Lab Ltd Composicion farmaceutica que comprende al acido 7-[2-(4-fluorofenil)-5-isopropil-3-fenil-4-[(4-hidroximetilfenilamino)carbonil]pirrol-1-il]-3,5-dihidroxi-heptanoico o una sal y al menos un agente estabilizante; procedimiento de preparacion, util en e
JP2009543773A (ja) * 2006-07-14 2009-12-10 ランバクシー ラボラトリーズ リミテッド HMG−CoAレダクターゼ阻害剤の多形体及びその使用
ES2382009T3 (es) 2006-12-01 2012-06-04 Bristol-Myers Squibb Company Derivados de N-((3-bencil)-2,2-(bis-fenil-)-propan-1-amina como inhibidores de CETP para el tratamiento de aterosclerosis y enfermedades cardiovasculares
BR112015026513A2 (pt) 2013-04-17 2017-07-25 Pfizer derivados de n-piperidin-3-ilbenzamida para tratar as doenças cardiovasculares
WO2016055901A1 (en) 2014-10-08 2016-04-14 Pfizer Inc. Substituted amide compounds
FI3911648T3 (fi) 2019-01-18 2025-01-10 Astrazeneca Ab 6'-[[[(1s,3s)-3-[[5-(difluorometoksi)-2-pyrimidinyyli]amino]syklopentyyli]amino][1(2h),3'-bipyridin]-2-oni pcsk9:n estäjänä ja menetelmät sen käyttöön

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL301580A (cg-RX-API-DMAC10.html) * 1962-12-11
DE1493454C3 (de) * 1963-08-26 1980-04-30 C.H. Boehringer Sohn, 6507 Ingelheim 1 -Aryloxy^-hydroxy-S-isopropylaminopropane und deren Salze sowie deren Herstellung und darauf basierende Arzneimittel
US3637852A (en) * 1963-08-26 1972-01-25 Boehringer Sohn Ingelheim 1-phenoxy-2-hydroxy-3-isopropylamino-propanes and salts thereof
GB1231783A (en) * 1967-05-16 1971-05-12 May & Baker Ltd Benzene derivatives
JPS512115B2 (cg-RX-API-DMAC10.html) * 1971-09-28 1976-01-23
JPS4911847A (cg-RX-API-DMAC10.html) * 1972-05-20 1974-02-01
GB1501632A (en) * 1974-06-28 1978-02-22 Cm Ind Aromatic ketones having cardiovascular activity

Also Published As

Publication number Publication date
FR2276032B1 (cg-RX-API-DMAC10.html) 1979-08-10
IE41386L (en) 1975-12-28
SE417087B (sv) 1981-02-23
DK292475A (da) 1975-12-29
ZA754141B (en) 1976-06-30
ES438931A1 (es) 1977-05-16
FR2276032A1 (fr) 1976-01-23
SE7507359L (sv) 1975-12-29
JPS5123233A (en) 1976-02-24
JPS5929574B2 (ja) 1984-07-21
DK143555B (da) 1981-09-07
US4302601A (en) 1981-11-24
IE41386B1 (en) 1979-12-19
CS197248B2 (en) 1980-04-30
DE2528147A1 (de) 1976-01-15
AR205388A1 (es) 1976-04-30
AU8256675A (en) 1977-01-06
US4252825A (en) 1981-02-24
DK143555C (da) 1982-02-01
JPS58140050A (ja) 1983-08-19
NL7507703A (nl) 1975-12-30
CA1052820A (en) 1979-04-17
ATA497275A (de) 1977-09-15
SE416546B (sv) 1981-01-19
JPS5826743B2 (ja) 1983-06-04
SE7812646L (sv) 1978-12-08
YU165775A (en) 1982-02-28
AT343098B (de) 1978-05-10
GB1501632A (en) 1978-02-22

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Legal Events

Date Code Title Description
RE Patent lapsed

Owner name: SANOFI

Effective date: 19910630