BE777689A - Nouveaux derives de l'imidazoline, compositions therapeutiques les contenant ainsi que le procede de preparation de ces derives et de ces compositions - Google Patents
Nouveaux derives de l'imidazoline, compositions therapeutiques les contenant ainsi que le procede de preparation de ces derives et de ces compositionsInfo
- Publication number
- BE777689A BE777689A BE777689A BE777689A BE777689A BE 777689 A BE777689 A BE 777689A BE 777689 A BE777689 A BE 777689A BE 777689 A BE777689 A BE 777689A BE 777689 A BE777689 A BE 777689A
- Authority
- BE
- Belgium
- Prior art keywords
- derivatives
- imidazoline
- preparation
- compositions
- compositions containing
- Prior art date
Links
- 239000000203 mixture Substances 0.000 title 2
- 150000002462 imidazolines Chemical class 0.000 title 1
- 230000001225 therapeutic effect Effects 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D307/78—Benzo [b] furans; Hydrogenated benzo [b] furans
- C07D307/79—Benzo [b] furans; Hydrogenated benzo [b] furans with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/06—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB332771 | 1971-01-27 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BE777689A true BE777689A (fr) | 1972-07-05 |
Family
ID=9756227
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BE777689A BE777689A (fr) | 1971-01-27 | 1972-01-05 | Nouveaux derives de l'imidazoline, compositions therapeutiques les contenant ainsi que le procede de preparation de ces derives et de ces compositions |
Country Status (17)
| Country | Link |
|---|---|
| US (1) | US3818035A (pm) |
| JP (1) | JPS4938273B1 (pm) |
| AT (1) | AT311336B (pm) |
| BE (1) | BE777689A (pm) |
| CA (1) | CA962273A (pm) |
| CH (1) | CH535254A (pm) |
| DE (1) | DE2203373C3 (pm) |
| DK (1) | DK138496B (pm) |
| FI (1) | FI55841C (pm) |
| GB (1) | GB1333471A (pm) |
| HU (1) | HU162823B (pm) |
| NL (1) | NL150454B (pm) |
| NO (1) | NO134115C (pm) |
| SE (1) | SE378426B (pm) |
| SU (1) | SU474145A3 (pm) |
| YU (1) | YU34694B (pm) |
| ZA (1) | ZA72286B (pm) |
Families Citing this family (28)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3927023A (en) * | 1974-05-24 | 1975-12-16 | Warner Lambert Co | Imidazolyl benzofurans |
| DE3049542A1 (de) * | 1980-12-31 | 1982-07-29 | Basf Ag, 6700 Ludwigshafen | Azolylalkyl-2,3-dihydrobenzofurane, diese enthaltende fungizide und verfahren zu ihrer herstellung |
| ZA825413B (en) * | 1981-08-26 | 1983-06-29 | Pfizer | Thromboxane synthetase inhibitors, processes for their production, and pharmaceutical compositions comprising them |
| US4851554A (en) * | 1987-04-06 | 1989-07-25 | University Of Tennessee Research Corporation | Certain 3-substituted 2-alkyl benzofuran derivatives |
| US4806663A (en) * | 1987-04-06 | 1989-02-21 | The University Of Tennessee Research Corporation | Certain 3-substituted 2-alkyl benzofuran derivatives |
| US4831156A (en) * | 1987-09-30 | 1989-05-16 | The University Of Tennessee Research Corp. | 3-substituted 2-alkyl indole derivatives |
| EP0924209B1 (en) * | 1997-12-19 | 2003-05-02 | Eli Lilly And Company | Hypoglycemic imidazoline compounds |
| US7777035B2 (en) * | 2005-06-22 | 2010-08-17 | Chemocentryx, Inc. | Azaindazole compounds and methods of use |
| RU2008130455A (ru) * | 2006-01-27 | 2010-03-10 | Ф.Хоффманн-Ля Рош Аг (Ch) | Применение замещенных производных 2-имидазола или имидазолинов |
| RU2009112496A (ru) * | 2006-10-19 | 2010-11-27 | Ф. Хоффманн-Ля Рош Аг (Ch) | Аминометил-4-имидазолы |
| RU2009112495A (ru) * | 2006-10-19 | 2010-11-27 | Ф. Хоффманн-Ля Рош Аг (Ch) | Аминометил-2-имидазолы со сродством к рецепторам, ассоциированным со следовыми аминами |
| CN101535292A (zh) * | 2006-11-02 | 2009-09-16 | 弗·哈夫曼-拉罗切有限公司 | 作为痕量胺相关受体的调节剂的取代的2-咪唑类化合物 |
| JP2010510184A (ja) * | 2006-11-16 | 2010-04-02 | エフ．ホフマン−ラ ロシュ アーゲー | 置換４−イミダゾール類 |
| AU2007332641A1 (en) * | 2006-12-13 | 2008-06-19 | F. Hoffmann-La Roche Ag | Novel 2 -imidazoles as ligands for trace amine associated receptors (TAAR) |
| US20080146523A1 (en) | 2006-12-18 | 2008-06-19 | Guido Galley | Imidazole derivatives |
| RU2473545C2 (ru) * | 2007-02-02 | 2013-01-27 | Ф.Хоффманн-Ля Рош Аг | Новые 2-аминооксазолины в качестве лигандов taar1 для заболеваний цнс |
| JP5130305B2 (ja) * | 2007-02-15 | 2013-01-30 | エフ．ホフマン−ラ ロシュ アーゲー | Ｔａａｒ１リガンドとしての２−アミノオキサゾリン |
| KR101150561B1 (ko) | 2007-07-02 | 2012-06-08 | 에프. 호프만-라 로슈 아게 | 미량 아민 결합 수용체(ｔａａｒ)에 대한 양호한 친화도를 갖는 2-이미다졸린 |
| MX2009013745A (es) * | 2007-07-03 | 2010-01-26 | Hoffmann La Roche | 4-imidazolinas y su uso como antidepresivos. |
| RU2010104632A (ru) * | 2007-07-27 | 2011-09-20 | Ф.Хоффманн-Ля Рош Аг (Ch) | 2-азетидинметанамины и 2-пирролидинметанамины в качестве лигандов taar |
| JP2010535172A (ja) * | 2007-08-02 | 2010-11-18 | エフ．ホフマン−ラ ロシュ アーゲー | Ｃｎｓ障害の処置のためのベンズアミド誘導体の使用 |
| CA2695331A1 (en) * | 2007-08-03 | 2009-02-12 | F. Hoffmann-La Roche Ag | Pyridinecarboxamide and benzamide derivatives as taar1 ligands |
| US8242153B2 (en) * | 2008-07-24 | 2012-08-14 | Hoffmann-La Roche Inc. | 4,5-dihydro-oxazol-2YL derivatives |
| CA2728480A1 (en) * | 2008-07-24 | 2010-01-28 | F. Hoffmann-La Roche Ag | 4,5-dihydro-oxazol-2-yl derivatives |
| US20100311798A1 (en) * | 2009-06-05 | 2010-12-09 | Decoret Guillaume | 2-aminooxazolines as taar1 ligands |
| US8354441B2 (en) * | 2009-11-11 | 2013-01-15 | Hoffmann-La Roche Inc. | Oxazoline derivatives |
| US9452980B2 (en) | 2009-12-22 | 2016-09-27 | Hoffmann-La Roche Inc. | Substituted benzamides |
| MY195528A (en) | 2016-03-17 | 2023-01-30 | Hoffmann La Roche | 5-Ethyl-4-Methyl-Pyrazole-3-Carboxamide Derivative Having Activity as Agonist of Taar |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE1121054B (de) * | 1960-11-23 | 1962-01-04 | Merck Ag E | Verfahren zur Herstellung eines neuen Imidazolinderivates und dessen Saeureadditionssalzen |
-
1971
- 1971-01-27 GB GB332771A patent/GB1333471A/en not_active Expired
-
1972
- 1972-01-05 BE BE777689A patent/BE777689A/xx not_active IP Right Cessation
- 1972-01-06 CH CH17272A patent/CH535254A/fr not_active IP Right Cessation
- 1972-01-10 US US00216795A patent/US3818035A/en not_active Expired - Lifetime
- 1972-01-17 ZA ZA720286A patent/ZA72286B/xx unknown
- 1972-01-25 DE DE2203373A patent/DE2203373C3/de not_active Expired
- 1972-01-26 DK DK34572AA patent/DK138496B/da unknown
- 1972-01-26 YU YU181/72A patent/YU34694B/xx unknown
- 1972-01-26 NO NO192/72A patent/NO134115C/no unknown
- 1972-01-26 HU HULA791A patent/HU162823B/hu not_active IP Right Cessation
- 1972-01-26 SE SE7200867A patent/SE378426B/xx unknown
- 1972-01-27 CA CA133,337A patent/CA962273A/en not_active Expired
- 1972-01-27 SU SU1742351A patent/SU474145A3/ru active
- 1972-01-27 NL NL727201121A patent/NL150454B/xx not_active IP Right Cessation
- 1972-01-27 FI FI219/72A patent/FI55841C/fi active
- 1972-01-27 JP JP47010207A patent/JPS4938273B1/ja active Pending
- 1972-01-27 AT AT64772A patent/AT311336B/de not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| NO134115B (pm) | 1976-05-10 |
| AU3817772A (en) | 1973-07-26 |
| DE2203373A1 (de) | 1972-08-17 |
| NO134115C (pm) | 1976-08-18 |
| NL7201121A (pm) | 1972-07-31 |
| DK138496B (da) | 1978-09-18 |
| SE378426B (pm) | 1975-09-01 |
| HU162823B (pm) | 1973-04-28 |
| GB1333471A (en) | 1973-10-10 |
| YU18172A (en) | 1979-07-10 |
| US3818035A (en) | 1974-06-18 |
| JPS4938273B1 (pm) | 1974-10-16 |
| FI55841B (fi) | 1979-06-29 |
| ZA72286B (en) | 1972-09-27 |
| FI55841C (fi) | 1979-10-10 |
| DE2203373C3 (de) | 1978-04-13 |
| DE2203373B2 (de) | 1977-08-11 |
| YU34694B (en) | 1979-12-31 |
| CH535254A (fr) | 1973-03-31 |
| NL150454B (nl) | 1976-08-16 |
| SU474145A3 (ru) | 1975-06-14 |
| CA962273A (en) | 1975-02-04 |
| AT311336B (de) | 1973-11-12 |
| DK138496C (pm) | 1979-02-26 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| RE | Patent lapsed |
Owner name: SANOFI Effective date: 19900131 |