BE1001271A5 - Nouvelles prostacyclines. - Google Patents
Nouvelles prostacyclines. Download PDFInfo
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- BE1001271A5 BE1001271A5 BE8701358A BE8701358A BE1001271A5 BE 1001271 A5 BE1001271 A5 BE 1001271A5 BE 8701358 A BE8701358 A BE 8701358A BE 8701358 A BE8701358 A BE 8701358A BE 1001271 A5 BE1001271 A5 BE 1001271A5
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- 239000008158 vegetable oil Substances 0.000 description 1
- 210000003462 vein Anatomy 0.000 description 1
- 239000000080 wetting agent Substances 0.000 description 1
- BPICBUSOMSTKRF-UHFFFAOYSA-N xylazine Chemical compound CC1=CC=CC(C)=C1NC1=NCCCS1 BPICBUSOMSTKRF-UHFFFAOYSA-N 0.000 description 1
- 229960001600 xylazine Drugs 0.000 description 1
- QUEDXNHFTDJVIY-UHFFFAOYSA-N γ-tocopherol Chemical class OC1=C(C)C(C)=C2OC(CCCC(C)CCCC(C)CCCC(C)C)(C)CCC2=C1 QUEDXNHFTDJVIY-UHFFFAOYSA-N 0.000 description 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D307/93—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems condensed with a ring other than six-membered
- C07D307/935—Not further condensed cyclopenta [b] furans or hydrogenated cyclopenta [b] furans
- C07D307/937—Not further condensed cyclopenta [b] furans or hydrogenated cyclopenta [b] furans with hydrocarbon or substituted hydrocarbon radicals directly attached in position 2, e.g. prostacyclins
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/08—Vasodilators for multiple indications
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Furan Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US93652286A | 1986-12-01 | 1986-12-01 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BE1001271A5 true BE1001271A5 (fr) | 1989-09-12 |
Family
ID=25468757
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BE8701358A BE1001271A5 (fr) | 1986-12-01 | 1987-11-30 | Nouvelles prostacyclines. |
Country Status (14)
Citations (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB2088856A (en) * | 1980-10-27 | 1982-06-16 | Chinoin Gyogyszer Es Vegyeszet | 7-substituted pg12-derivatives their preparation and pharmaceutical compositions containing them |
| EP0054795A2 (en) * | 1980-12-09 | 1982-06-30 | Teijin Limited | Novel halogenated prostacyclins, process for the production thereof, and pharmaceutical use thereof |
| JPS5867682A (ja) * | 1981-10-16 | 1983-04-22 | Teijin Ltd | フルオロｐｇｉ↓２類の製法 |
| JPS58150583A (ja) * | 1982-03-04 | 1983-09-07 | Teijin Ltd | 新規なハロゲン化プロスタサイクリン類、それらの製造法およびそれらを活性成分とする薬学的組成物 |
| EP0148953A1 (en) * | 1983-06-10 | 1985-07-24 | Asahi Glass Company Ltd. | 7-fluoroprostaglandins and process for their preparation |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4558142A (en) * | 1981-03-11 | 1985-12-10 | Hoffmann-La Roche Inc. | 7-Fluoro-prostacyclin analogs |
| CH648556A5 (de) * | 1981-03-11 | 1985-03-29 | Hoffmann La Roche | Fluorprostacycline. |
| US4634782A (en) * | 1985-06-24 | 1987-01-06 | Hoffmann-La Roche Inc. | 7-fluoro-dihydro PGI compounds |
-
1987
- 1987-11-06 CH CH4345/87A patent/CH674363A5/de not_active IP Right Cessation
- 1987-11-27 FR FR8716485A patent/FR2607501A1/fr active Pending
- 1987-11-27 JP JP62297860A patent/JPS63145275A/ja active Pending
- 1987-11-27 ZA ZA878947A patent/ZA878947B/xx unknown
- 1987-11-27 NL NL8702855A patent/NL8702855A/nl not_active Application Discontinuation
- 1987-11-27 NZ NZ222723A patent/NZ222723A/en unknown
- 1987-11-30 DK DK627787A patent/DK627787A/da not_active Application Discontinuation
- 1987-11-30 GB GB8727991A patent/GB2198130B/en not_active Expired - Lifetime
- 1987-11-30 SE SE8704770A patent/SE8704770L/xx not_active Application Discontinuation
- 1987-11-30 AU AU81907/87A patent/AU597128B2/en not_active Ceased
- 1987-11-30 IT IT22814/87A patent/IT1223390B/it active
- 1987-11-30 DE DE19873740595 patent/DE3740595A1/de not_active Withdrawn
- 1987-11-30 BE BE8701358A patent/BE1001271A5/fr not_active IP Right Cessation
- 1987-11-30 AT AT0313887A patent/AT391697B/de not_active IP Right Cessation
Patent Citations (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB2088856A (en) * | 1980-10-27 | 1982-06-16 | Chinoin Gyogyszer Es Vegyeszet | 7-substituted pg12-derivatives their preparation and pharmaceutical compositions containing them |
| EP0054795A2 (en) * | 1980-12-09 | 1982-06-30 | Teijin Limited | Novel halogenated prostacyclins, process for the production thereof, and pharmaceutical use thereof |
| JPS5867682A (ja) * | 1981-10-16 | 1983-04-22 | Teijin Ltd | フルオロｐｇｉ↓２類の製法 |
| JPS58150583A (ja) * | 1982-03-04 | 1983-09-07 | Teijin Ltd | 新規なハロゲン化プロスタサイクリン類、それらの製造法およびそれらを活性成分とする薬学的組成物 |
| EP0148953A1 (en) * | 1983-06-10 | 1985-07-24 | Asahi Glass Company Ltd. | 7-fluoroprostaglandins and process for their preparation |
Non-Patent Citations (3)
| Title |
|---|
| CHEMICAL ABSTRACTS, vol. 100, no. 11, 12 mars 1984, page 525, résumé no. 85494v, Columbus, Ohio, US; & JP-A-58 150 583 (TEIJIN LTD) 07-09-1983 * |
| CHEMICAL ABSTRACTS, vol. 99, no. 11, 12 septembre 1983, page 543, résumé no. 87908t, Columbus, Ohio, US; & JP-A-58 67 682 (TEIJIN LTD) 22-04-1983 * |
| TETRAHEDRON, vol. 39, no. 22, 1983, pages 3807-3819, Pergamon Press Ltd, Oxford, GB; K. BANNAI et al.: "Synthesis of chemically stable prostacyclin analogs" * |
Also Published As
| Publication number | Publication date |
|---|---|
| GB2198130A (en) | 1988-06-08 |
| FR2607501A1 (fr) | 1988-06-03 |
| DK627787A (da) | 1988-06-02 |
| GB2198130B (en) | 1990-08-08 |
| GB8727991D0 (en) | 1988-01-06 |
| AU8190787A (en) | 1988-06-02 |
| DE3740595A1 (de) | 1988-06-16 |
| AT391697B (de) | 1990-11-12 |
| SE8704770L (sv) | 1988-06-02 |
| NL8702855A (nl) | 1988-07-01 |
| DK627787D0 (da) | 1987-11-30 |
| AU597128B2 (en) | 1990-05-24 |
| CH674363A5 (enrdf_load_stackoverflow) | 1990-05-31 |
| IT8722814A0 (it) | 1987-11-30 |
| ZA878947B (en) | 1988-06-01 |
| IT1223390B (it) | 1990-09-19 |
| ATA313887A (de) | 1990-05-15 |
| NZ222723A (en) | 1990-11-27 |
| SE8704770D0 (sv) | 1987-11-30 |
| JPS63145275A (ja) | 1988-06-17 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| RE | Patent lapsed |
Owner name: F. HOFFMANN-LA ROCHE A.G. Effective date: 19911130 |