AU672675B2 - Thiazolopyrimidine derivatives - Google Patents

Thiazolopyrimidine derivatives Download PDF

Info

Publication number
AU672675B2
AU672675B2 AU59252/94A AU5925294A AU672675B2 AU 672675 B2 AU672675 B2 AU 672675B2 AU 59252/94 A AU59252/94 A AU 59252/94A AU 5925294 A AU5925294 A AU 5925294A AU 672675 B2 AU672675 B2 AU 672675B2
Authority
AU
Australia
Prior art keywords
group
carbon atoms
compounds
pyrimidine
dihydro
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
AU59252/94A
Other languages
English (en)
Other versions
AU5925294A (en
Inventor
Haruko Chatani
Michio Iwahana
Hiroo Matsumoto
Kiyoshi Nakayama
Noriko Tanaka
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Daiichi Pharmaceutical Co Ltd
Original Assignee
Daiichi Pharmaceutical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Daiichi Pharmaceutical Co Ltd filed Critical Daiichi Pharmaceutical Co Ltd
Publication of AU5925294A publication Critical patent/AU5925294A/en
Application granted granted Critical
Publication of AU672675B2 publication Critical patent/AU672675B2/en
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
AU59252/94A 1993-04-01 1994-03-31 Thiazolopyrimidine derivatives Ceased AU672675B2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP11087793 1993-04-01
JP5-110877 1993-04-01

Publications (2)

Publication Number Publication Date
AU5925294A AU5925294A (en) 1994-10-06
AU672675B2 true AU672675B2 (en) 1996-10-10

Family

ID=14546967

Family Applications (1)

Application Number Title Priority Date Filing Date
AU59252/94A Ceased AU672675B2 (en) 1993-04-01 1994-03-31 Thiazolopyrimidine derivatives

Country Status (9)

Country Link
US (1) US5599813A (OSRAM)
EP (1) EP0618208A1 (OSRAM)
CN (1) CN1100425A (OSRAM)
AU (1) AU672675B2 (OSRAM)
CA (1) CA2120395A1 (OSRAM)
FI (1) FI941487A7 (OSRAM)
NO (1) NO941135L (OSRAM)
PH (1) PH31256A (OSRAM)
TW (1) TW272193B (OSRAM)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR20000022532A (ko) * 1996-06-27 2000-04-25 오노 야꾸힝 고교 가부시키가이샤 아릴(설파이드, 설폭시드 및 설폰)유도체 및 이를 활성 성분으로 함유하는 약물
EP2311490A3 (en) 1998-07-13 2011-05-04 Board of Regents, The University of Texas System Uses of antibodies to aminophospholipids for cancer treatment
SI1107795T1 (en) 1998-09-04 2003-06-30 The Regents Of The University Of Michigan Thiomolybdate associated with at least one carbohydrate, and its use for preventing or treating diseases characterized by aberrant vascularization, such as cancer, wet type macular degeneration, rheumatoid arthritis
US6930101B1 (en) 1999-05-17 2005-08-16 The Regents Of The University Of California Thiazolopyrimidines useful as TNFα inhibitors
DE10112197A1 (de) * 2001-03-14 2002-09-19 Gruenenthal Gmbh Substituierte Pyrazolo- und Thiazolopyrimidine
EP2283868B1 (en) 2002-07-15 2016-03-30 Board of Regents, The University of Texas System Peptides binding to phosphatidylethanolamine and their use in treating viral infections and cancer
EP2371363B1 (en) 2004-01-22 2020-04-08 University of Miami Coenzyme Q10 formulations for use in the treatment of solid tumours
EP2343303A1 (de) 2004-10-07 2011-07-13 Boehringer Ingelheim International GmbH PI3-Kinase Inhibitoren
DK2219672T3 (en) 2007-11-09 2016-05-17 Peregrine Pharmaceuticals Inc The anti-VEGF antibody compositions and methods
EP2323679A4 (en) 2008-07-25 2012-08-22 Univ Colorado CLIP INHIBITORS AND METHODS FOR MODULATING IMMUNE FUNCTION
CN101899058B (zh) * 2010-05-24 2012-05-23 中国人民解放军第四军医大学 一种噻唑并嘧啶化合物及其制备方法和应用
CN103443107B (zh) * 2011-03-28 2016-04-20 弗·哈夫曼-拉罗切有限公司 噻唑并嘧啶化合物
EP3576726A1 (en) 2017-02-06 2019-12-11 Massachusetts Institute Of Technology Methods and products related to glutaminase inhibitors

Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0038731A2 (fr) * 1980-04-08 1981-10-28 Synthelabo Dérivés de thiazole, leur préparation et leur application en thérapeutique
EP0045251B1 (fr) * 1980-07-24 1983-11-30 Rhone-Poulenc Sante Nouveaux dérivés de la thiazolo (3,2-a) pyrimidine, leur préparation et les médicaments qui les contiennent
EP0404525A2 (en) * 1989-06-21 1990-12-27 Takeda Chemical Industries, Ltd. Sulfur-containing fused pyrimidine derivatives, their production and use

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1556878A (en) * 1976-01-19 1979-11-28 Diamond Shamrock Corp Imidazothiazoles
US4347248A (en) * 1981-03-23 1982-08-31 American Cyanamid Company 2,3-Disubstituted-thiazolo[3,2-a]pyrimidines

Patent Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0038731A2 (fr) * 1980-04-08 1981-10-28 Synthelabo Dérivés de thiazole, leur préparation et leur application en thérapeutique
EP0045251B1 (fr) * 1980-07-24 1983-11-30 Rhone-Poulenc Sante Nouveaux dérivés de la thiazolo (3,2-a) pyrimidine, leur préparation et les médicaments qui les contiennent
EP0404525A2 (en) * 1989-06-21 1990-12-27 Takeda Chemical Industries, Ltd. Sulfur-containing fused pyrimidine derivatives, their production and use

Also Published As

Publication number Publication date
NO941135D0 (no) 1994-03-28
CN1100425A (zh) 1995-03-22
US5599813A (en) 1997-02-04
FI941487L (fi) 1994-10-02
FI941487A0 (fi) 1994-03-30
NO941135L (no) 1994-10-03
PH31256A (en) 1998-06-18
CA2120395A1 (en) 1994-10-02
EP0618208A1 (en) 1994-10-05
TW272193B (OSRAM) 1996-03-11
FI941487A7 (fi) 1994-10-02
AU5925294A (en) 1994-10-06

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