AU659506B2 - Method for making steroidal peracyl glycosides - Google Patents

Method for making steroidal peracyl glycosides Download PDF

Info

Publication number
AU659506B2
AU659506B2 AU27758/92A AU2775892A AU659506B2 AU 659506 B2 AU659506 B2 AU 659506B2 AU 27758/92 A AU27758/92 A AU 27758/92A AU 2775892 A AU2775892 A AU 2775892A AU 659506 B2 AU659506 B2 AU 659506B2
Authority
AU
Australia
Prior art keywords
zinc
tigogenin
recited
cellobioside
international
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
AU27758/92A
Other languages
English (en)
Other versions
AU2775892A (en
Inventor
Douglas John M Allen
Frank Robert Busch
John Francis Lambert
Russell James Shine
Stanley Walter Walinsky
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Corp SRL
Original Assignee
Pfizer Corp Belgium
Pfizer Corp SRL
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Corp Belgium, Pfizer Corp SRL filed Critical Pfizer Corp Belgium
Publication of AU2775892A publication Critical patent/AU2775892A/en
Application granted granted Critical
Publication of AU659506B2 publication Critical patent/AU659506B2/en
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J71/00Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
    • C07J71/0005Oxygen-containing hetero ring

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Steroid Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
AU27758/92A 1991-11-25 1992-10-15 Method for making steroidal peracyl glycosides Ceased AU659506B2 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US79757491A 1991-11-25 1991-11-25
US797574 1991-11-25
PCT/US1992/008638 WO1993011150A1 (en) 1991-11-25 1992-10-15 Method for making steroidal peracyl glycosides

Publications (2)

Publication Number Publication Date
AU2775892A AU2775892A (en) 1993-06-28
AU659506B2 true AU659506B2 (en) 1995-05-18

Family

ID=25171219

Family Applications (1)

Application Number Title Priority Date Filing Date
AU27758/92A Ceased AU659506B2 (en) 1991-11-25 1992-10-15 Method for making steroidal peracyl glycosides

Country Status (13)

Country Link
EP (1) EP0619822A1 (enrdf_load_stackoverflow)
JP (1) JPH0826064B2 (enrdf_load_stackoverflow)
AU (1) AU659506B2 (enrdf_load_stackoverflow)
CA (1) CA2123684A1 (enrdf_load_stackoverflow)
FI (1) FI942394A0 (enrdf_load_stackoverflow)
HU (1) HUT67035A (enrdf_load_stackoverflow)
IL (1) IL103797A0 (enrdf_load_stackoverflow)
MX (1) MX9206761A (enrdf_load_stackoverflow)
NZ (1) NZ245244A (enrdf_load_stackoverflow)
PT (1) PT101088A (enrdf_load_stackoverflow)
TW (1) TW232699B (enrdf_load_stackoverflow)
WO (1) WO1993011150A1 (enrdf_load_stackoverflow)
ZA (1) ZA929081B (enrdf_load_stackoverflow)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2139104A1 (en) * 1992-06-26 1994-01-06 Michael P. Deninno Steroidal glycosides for treating hypercholesterolemia
NZ252006A (en) * 1992-06-26 1995-10-26 Pfizer Preparation of 1-o-steroidal peracyl-beta-glycosides
WO1994000478A1 (en) * 1992-06-26 1994-01-06 Pfizer Inc. Steroidal beta-o-cellobioside heptaalkanoate process
EP0696292A1 (en) * 1993-04-28 1996-02-14 Pfizer Inc. Spirostanyl glycosidal crystalline monohydrate
US5502038A (en) * 1993-06-21 1996-03-26 Medical Research Foundation Of Oregon Cholesterol sequestrant glycosides that inhibit intestinal cholesterol absorption
EP0737202A1 (en) * 1993-12-28 1996-10-16 Pfizer Inc. Hypocholesterolemic agents
US6150336A (en) * 1995-05-29 2000-11-21 Pfizer Inc. Steroidal glycosides
US5756470A (en) * 1996-10-29 1998-05-26 Schering Corporation Sugar-substituted 2-azetidinones useful as hypocholesterolemic agents
US6982251B2 (en) 2000-12-20 2006-01-03 Schering Corporation Substituted 2-azetidinones useful as hypocholesterolemic agents
SI1355644T1 (sl) 2001-01-26 2006-10-31 Schering Corp Uporaba substituiranih azetidinonskih spojin za zdravljenje sitosterolemije
ES2290562T3 (es) 2001-01-26 2008-02-16 Schering Corporation Combinaciones del activador del receptor activado por el proliferador de los peroxisomas (ppar) fenofibrato con el inhibidor de la absorcion de esteroles ezetimiba para indicaciones vasculares.
US7071181B2 (en) 2001-01-26 2006-07-04 Schering Corporation Methods and therapeutic combinations for the treatment of diabetes using sterol absorption inhibitors
US7056906B2 (en) 2001-09-21 2006-06-06 Schering Corporation Combinations of hormone replacement therapy composition(s) and sterol absorption inhibitor(s) and treatments for vascular conditions in post-menopausal women
US7053080B2 (en) 2001-09-21 2006-05-30 Schering Corporation Methods and therapeutic combinations for the treatment of obesity using sterol absorption inhibitors
PT1429756E (pt) 2001-09-21 2007-01-31 Schering Corp Tratamento de xantoma com derivados de azetidinona como inibidores de absorção de esteróis
MXPA05004811A (es) 2002-11-06 2005-07-22 Schering Corp Inhibidores de absorcion de colesterol para el tratamiento de trastornos autoinmunes.
ES2311806T3 (es) 2003-03-07 2009-02-16 Schering Corporation Compuesto de azetidinona sustituidos, fornulaciones y usos de los mismos para el tratamiento de hipercolesterolemia.
US7459442B2 (en) 2003-03-07 2008-12-02 Schering Corporation Substituted azetidinone compounds, processes for preparing the same, formulations and uses thereof
JP4589919B2 (ja) 2003-03-07 2010-12-01 シェーリング コーポレイション 高コレステロール血症の処置のための、置換アゼチジノン化合物、これらの処方物および使用
WO2004081004A1 (en) 2003-03-07 2004-09-23 Schering Corporation Substituted azetidinone compounds, formulations and uses thereof for the treatment of hypercholesterolemia

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4602005A (en) * 1982-05-17 1986-07-22 Medical Research Foundation Of Oregon Tigogenin cellobioside for treating hypercholesterolemia and atherosclerosis
US4602003A (en) * 1982-05-17 1986-07-22 Medical Research Foundation Of Oregon Synthetic compounds to inhibit intestinal absorption of cholesterol in the treatment of hypercholesterolemia

Also Published As

Publication number Publication date
MX9206761A (es) 1995-01-31
FI942394A7 (fi) 1994-05-24
FI942394L (fi) 1994-05-24
FI942394A0 (fi) 1994-05-24
HUT67035A (en) 1995-01-30
TW232699B (enrdf_load_stackoverflow) 1994-10-21
JPH06510794A (ja) 1994-12-01
JPH0826064B2 (ja) 1996-03-13
AU2775892A (en) 1993-06-28
IL103797A0 (en) 1993-04-04
ZA929081B (en) 1994-05-24
NZ245244A (en) 1995-04-27
HU9401374D0 (en) 1994-08-29
PT101088A (pt) 1994-02-28
EP0619822A1 (en) 1994-10-19
CA2123684A1 (en) 1993-06-10
WO1993011150A1 (en) 1993-06-10

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