AU635739B2 - Alkyl derivates in 17/21 of 19-nor progesterone - Google Patents

Alkyl derivates in 17/21 of 19-nor progesterone Download PDF

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Publication number
AU635739B2
AU635739B2 AU55525/90A AU5552590A AU635739B2 AU 635739 B2 AU635739 B2 AU 635739B2 AU 55525/90 A AU55525/90 A AU 55525/90A AU 5552590 A AU5552590 A AU 5552590A AU 635739 B2 AU635739 B2 AU 635739B2
Authority
AU
Australia
Prior art keywords
document
formula
date
pregna
compound
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
AU55525/90A
Other languages
English (en)
Other versions
AU5552590A (en
Inventor
Nejib Mohamed Nasraoui
Claude Tchernatinsky
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Laboratoire Theramex SAM
Original Assignee
Laboratoire Theramex SAM
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Laboratoire Theramex SAM filed Critical Laboratoire Theramex SAM
Publication of AU5552590A publication Critical patent/AU5552590A/en
Application granted granted Critical
Publication of AU635739B2 publication Critical patent/AU635739B2/en
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J7/00—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of two carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J9/00—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of more than two carbon atoms, e.g. cholane, cholestane, coprostane
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J7/00—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of two carbon atoms
    • C07J7/0005—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of two carbon atoms not substituted in position 21
    • C07J7/001—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of two carbon atoms not substituted in position 21 substituted in position 20 by a keto group
    • C07J7/004—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of two carbon atoms not substituted in position 21 substituted in position 20 by a keto group substituted in position 17 alfa

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Diabetes (AREA)
  • Endocrinology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
AU55525/90A 1989-04-13 1990-04-13 Alkyl derivates in 17/21 of 19-nor progesterone Ceased AU635739B2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR8904910 1989-04-13
FR8904910A FR2645864B1 (fr) 1989-04-13 1989-04-13 Nouveaux derives alcoyles en 17/21 de la 19-nor progesterone, leurs procedes d'obtention et les compositions pharmaceutiques en renfermant

Publications (2)

Publication Number Publication Date
AU5552590A AU5552590A (en) 1990-11-05
AU635739B2 true AU635739B2 (en) 1993-04-01

Family

ID=9380699

Family Applications (1)

Application Number Title Priority Date Filing Date
AU55525/90A Ceased AU635739B2 (en) 1989-04-13 1990-04-13 Alkyl derivates in 17/21 of 19-nor progesterone

Country Status (12)

Country Link
EP (1) EP0437552A1 (ko)
JP (1) JPH04500523A (ko)
KR (1) KR920700219A (ko)
AU (1) AU635739B2 (ko)
FI (1) FI906116A0 (ko)
FR (1) FR2645864B1 (ko)
HU (1) HU208152B (ko)
NO (1) NO174393C (ko)
OA (1) OA09632A (ko)
RU (1) RU1836379C (ko)
TN (1) TNSN90053A1 (ko)
WO (1) WO1990012027A1 (ko)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2018109508A1 (en) * 2016-12-16 2018-06-21 Richter Gedeon Nyrt. Industrial process for the synthesis of nomegestrol-acetate

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2675047B1 (fr) * 1991-04-09 1995-05-12 Theramex Nouvelles compositions pharmaceutiques anti-glaucomateuses et leur procede d'obtention.
DK0593520T3 (da) * 1991-06-18 2000-04-03 Theramex Forbindelser med indhold af steroider og deres anvendelse til behandling af glaucom
FR2679236B1 (fr) * 1991-07-18 1997-01-24 Theramex Nouveaux sterouides substitues en position 6, leurs procedes d'obtention et des compositions pharmaceutiques en renfermant.

Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR1367429A (fr) * 1962-07-18 1964-07-24 American Cyanamid Co Procédé de préparation de nouveaux dérivés de la progestérone substituée en 17
AU2629588A (en) * 1987-10-27 1989-05-23 Laboratoire Theramex S.A. Derivatives of 19-norprogesterone, their preparation and their use

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2077877B1 (ko) * 1970-02-20 1974-02-01 Roussel Uclaf
FR2552766B1 (fr) * 1983-10-04 1987-06-26 Theramex Nouveau procede de preparation de derives de la serie du 17 a-hydroxy 19-nor progesterone

Patent Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR1367429A (fr) * 1962-07-18 1964-07-24 American Cyanamid Co Procédé de préparation de nouveaux dérivés de la progestérone substituée en 17
AU2629588A (en) * 1987-10-27 1989-05-23 Laboratoire Theramex S.A. Derivatives of 19-norprogesterone, their preparation and their use

Cited By (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2018109508A1 (en) * 2016-12-16 2018-06-21 Richter Gedeon Nyrt. Industrial process for the synthesis of nomegestrol-acetate
EA037842B1 (ru) * 2016-12-16 2021-05-26 Рихтер Гедеон Нирт. Промышленный способ синтеза номегэстрола ацетата
US11274119B2 (en) 2016-12-16 2022-03-15 Richter Gedeon Nyrt. Industrial process for the synthesis of nomegestrol-acetate

Also Published As

Publication number Publication date
TNSN90053A1 (fr) 1991-03-05
HU904373D0 (en) 1991-06-28
WO1990012027A1 (fr) 1990-10-18
FR2645864B1 (fr) 1991-07-12
HUT56579A (en) 1991-09-30
NO174393C (no) 1994-04-27
FI906116A0 (fi) 1990-12-12
JPH04500523A (ja) 1992-01-30
RU1836379C (ru) 1993-08-23
KR920700219A (ko) 1992-02-19
AU5552590A (en) 1990-11-05
NO905344D0 (no) 1990-12-11
NO174393B (no) 1994-01-17
OA09632A (fr) 1993-04-30
HU208152B (en) 1993-08-30
FR2645864A1 (fr) 1990-10-19
EP0437552A1 (fr) 1991-07-24
NO905344L (no) 1991-02-01

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