AU594972B2 - N-substituted-arylalkyl and arylalkylene aminoheterocyclics as cardiovascular antihistaminic and antisecretory agents - Google Patents
N-substituted-arylalkyl and arylalkylene aminoheterocyclics as cardiovascular antihistaminic and antisecretory agents Download PDFInfo
- Publication number
- AU594972B2 AU594972B2 AU62473/86A AU6247386A AU594972B2 AU 594972 B2 AU594972 B2 AU 594972B2 AU 62473/86 A AU62473/86 A AU 62473/86A AU 6247386 A AU6247386 A AU 6247386A AU 594972 B2 AU594972 B2 AU 594972B2
- Authority
- AU
- Australia
- Prior art keywords
- acceptable salt
- pharmaceutically acceptable
- bis
- fluorophenyl
- mole
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Ceased
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D223/00—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom
- C07D223/02—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom not condensed with other rings
- C07D223/04—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom not condensed with other rings with only hydrogen atoms, halogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
- C07D211/10—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with radicals containing only carbon and hydrogen atoms attached to ring carbon atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pyridine Compounds (AREA)
- Pyrane Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pyrrole Compounds (AREA)
- Quinoline Compounds (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US81970186A | 1986-01-17 | 1986-01-17 | |
US819701 | 1986-01-17 |
Publications (2)
Publication Number | Publication Date |
---|---|
AU6247386A AU6247386A (en) | 1987-07-23 |
AU594972B2 true AU594972B2 (en) | 1990-03-22 |
Family
ID=25228814
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AU62473/86A Ceased AU594972B2 (en) | 1986-01-17 | 1986-09-09 | N-substituted-arylalkyl and arylalkylene aminoheterocyclics as cardiovascular antihistaminic and antisecretory agents |
Country Status (11)
Country | Link |
---|---|
JP (1) | JPH0772171B2 (pt) |
KR (1) | KR900005368B1 (pt) |
AU (1) | AU594972B2 (pt) |
DK (1) | DK347986A (pt) |
GR (1) | GR862024B (pt) |
IL (1) | IL78939A (pt) |
IN (1) | IN163948B (pt) |
NZ (1) | NZ217408A (pt) |
PH (3) | PH23843A (pt) |
PT (1) | PT84128B (pt) |
ZA (1) | ZA864522B (pt) |
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AU629534B2 (en) * | 1988-02-24 | 1992-10-08 | A.H. Robins Company, Incorporated | New methods and related compounds |
Families Citing this family (17)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
PH23283A (en) * | 1986-02-26 | 1989-06-30 | Eisai Co Ltd | Piperidine derivative, pharmaceutical composition containing the same and method of use thereof |
AU629535B2 (en) * | 1988-02-10 | 1992-10-08 | A.H. Robins Company, Incorporated | N-substituted-arylalkyl and arylalkylene aminoheterocyclics as cardiovascular antihistaminic and antisecretory agents |
GB8825505D0 (en) * | 1988-11-01 | 1988-12-07 | Pfizer Ltd | Therapeutic agents |
GB8906166D0 (en) * | 1989-03-17 | 1989-05-04 | Pfizer Ltd | Therapeutic agents |
GB8928042D0 (en) * | 1989-12-12 | 1990-02-14 | Pfizer Ltd | Muscarinic receptor antagonists |
US6004980A (en) * | 1990-06-01 | 1999-12-21 | Merrell Pharmaceuticals, Inc. | (+)-α-(2,3-dimethoxyphenyl)-1-[2-(4-fluorophenyl)ethyl]-4-piperidinemethanol |
CA2093798C (en) * | 1990-10-10 | 2000-02-01 | John J. Piwinski | Pyridine and pyridine n-oxide derivatives of diaryl methyl piperidines or piperazines, and compositions and methods of use thereof |
DE4111861A1 (de) * | 1991-04-11 | 1992-10-15 | Schwabe Willmar Gmbh & Co | Benzopyranone, verfahren zu ihrer herstellung und verwendung |
WO1993011108A1 (en) * | 1991-11-29 | 1993-06-10 | Zeria Pharmaceutical Co., Ltd. | Piperidine derivative and medicine containing the same |
US5807858A (en) * | 1996-06-05 | 1998-09-15 | Delta Pharmaceutical, Inc. | Compositions and methods for reducing respiratory depression |
US5681830A (en) * | 1992-02-03 | 1997-10-28 | Delta Pharmaceuticals, Inc. | Opioid compounds |
EP0635012B1 (en) * | 1992-03-27 | 1996-07-10 | Schering Corporation | Unbridged bis-aryl carbinol derivatives, compositions and methods of use |
HUT71132A (en) * | 1992-03-27 | 1995-11-28 | Schering Corp | Bis-aryl-carbinol derivatives, pharmaceutical compositions containing them and process for producing |
HU221726B1 (hu) | 1993-07-30 | 2002-12-28 | Ardent Pharmaceuticals Inc. | Piperazinszármazékok, e vegyületeket tartalmazó gyógyászati készítmények és eljárás a vegyületek előállítására |
JP4057088B2 (ja) * | 1996-04-22 | 2008-03-05 | 株式会社カネカ | ピロリジン誘導体の製造方法 |
US6028083A (en) * | 1997-07-25 | 2000-02-22 | Hoechst Marion Roussel, Inc. | Esters of (+)-α-(2,3-dimethoxyphenyl)-1-[2-(4-fluorophenyl) ethyl]-4-piperidinemethanol |
TW200510298A (en) * | 2003-06-13 | 2005-03-16 | Theravance Inc | Substituted pyrrolidine and related compounds |
Citations (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AU506432B2 (en) * | 1976-08-13 | 1980-01-03 | G. D. Searle & Co | 4 ((4 Diphenylmethyl) l-piperidinyl)methyl) benzenamines |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4632925A (en) * | 1985-10-07 | 1986-12-30 | Hoffmann-La Roche Inc. | N-substituted diphenylpiperidines and antiobesity use thereof |
US4810713A (en) * | 1985-12-20 | 1989-03-07 | A. H. Robins Company, Incorporated | Arylalkyl-heterocyclic amines, n-substituted by aryloxyalkyl groups used in a method for allergy treatment |
-
1986
- 1986-05-27 IN IN407/MAS/86A patent/IN163948B/en unknown
- 1986-05-27 IL IL78939A patent/IL78939A/xx not_active IP Right Cessation
- 1986-06-17 ZA ZA864522A patent/ZA864522B/xx unknown
- 1986-07-18 JP JP61169673A patent/JPH0772171B2/ja not_active Expired - Lifetime
- 1986-07-22 DK DK347986A patent/DK347986A/da not_active Application Discontinuation
- 1986-07-30 PH PH34083A patent/PH23843A/en unknown
- 1986-07-30 GR GR862024A patent/GR862024B/el unknown
- 1986-08-29 NZ NZ217408A patent/NZ217408A/xx unknown
- 1986-09-09 AU AU62473/86A patent/AU594972B2/en not_active Ceased
-
1987
- 1987-01-15 KR KR1019870000264A patent/KR900005368B1/ko not_active IP Right Cessation
- 1987-01-16 PT PT84128A patent/PT84128B/pt not_active IP Right Cessation
-
1988
- 1988-07-14 PH PH37224A patent/PH24983A/en unknown
- 1988-07-14 PH PH37223A patent/PH24904A/en unknown
Patent Citations (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AU506432B2 (en) * | 1976-08-13 | 1980-01-03 | G. D. Searle & Co | 4 ((4 Diphenylmethyl) l-piperidinyl)methyl) benzenamines |
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AU629534B2 (en) * | 1988-02-24 | 1992-10-08 | A.H. Robins Company, Incorporated | New methods and related compounds |
Also Published As
Publication number | Publication date |
---|---|
KR870007131A (ko) | 1987-08-17 |
NZ217408A (en) | 1990-03-27 |
IN163948B (pt) | 1988-12-10 |
PT84128B (pt) | 1989-05-31 |
PH24983A (en) | 1990-12-26 |
JPH0772171B2 (ja) | 1995-08-02 |
ZA864522B (en) | 1987-02-25 |
DK347986D0 (da) | 1986-07-22 |
PH24904A (en) | 1990-12-26 |
JPS62169763A (ja) | 1987-07-25 |
PH23843A (en) | 1989-11-23 |
DK347986A (da) | 1987-07-18 |
PT84128A (en) | 1987-02-01 |
AU6247386A (en) | 1987-07-23 |
KR900005368B1 (ko) | 1990-07-28 |
IL78939A0 (en) | 1986-09-30 |
GR862024B (en) | 1986-12-24 |
IL78939A (en) | 1990-04-29 |
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