AU2020361093B2 - Pharmaceutical drug containing heterocyclidene acetamide derivative - Google Patents
Pharmaceutical drug containing heterocyclidene acetamide derivativeInfo
- Publication number
- AU2020361093B2 AU2020361093B2 AU2020361093A AU2020361093A AU2020361093B2 AU 2020361093 B2 AU2020361093 B2 AU 2020361093B2 AU 2020361093 A AU2020361093 A AU 2020361093A AU 2020361093 A AU2020361093 A AU 2020361093A AU 2020361093 B2 AU2020361093 B2 AU 2020361093B2
- Authority
- AU
- Australia
- Prior art keywords
- dry eye
- item
- eye
- symptom
- zone
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Active
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A61K31/35—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
- A61K31/352—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom condensed with carbocyclic rings, e.g. methantheline
- A61K31/353—3,4-Dihydrobenzopyrans, e.g. chroman, catechin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/02—Inorganic compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/26—Carbohydrates, e.g. sugar alcohols, amino sugars, nucleic acids, mono-, di- or oligo-saccharides; Derivatives thereof, e.g. polysorbates, sorbitan fatty acid esters or glycyrrhizin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0048—Eye, e.g. artificial tears
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/10—Dispersions; Emulsions
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A61P27/04—Artificial tears; Irrigation solutions
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Epidemiology (AREA)
- General Chemical & Material Sciences (AREA)
- Ophthalmology & Optometry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Organic Chemistry (AREA)
- Dispersion Chemistry (AREA)
- Molecular Biology (AREA)
- Oil, Petroleum & Natural Gas (AREA)
- Inorganic Chemistry (AREA)
- Biochemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicinal Preparation (AREA)
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| AU2026202464A AU2026202464A1 (en) | 2019-10-04 | 2026-03-31 | Pharmaceutical Drug Containing Heterocyclidene Acetamide Derivative |
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2019184053 | 2019-10-04 | ||
| JP2019-184053 | 2019-10-04 | ||
| PCT/JP2020/037548 WO2021066144A1 (ja) | 2019-10-04 | 2020-10-02 | ヘテロシクリデンアセトアミド誘導体含有医薬 |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AU2026202464A Division AU2026202464A1 (en) | 2019-10-04 | 2026-03-31 | Pharmaceutical Drug Containing Heterocyclidene Acetamide Derivative |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| AU2020361093A1 AU2020361093A1 (en) | 2022-05-19 |
| AU2020361093B2 true AU2020361093B2 (en) | 2026-04-30 |
Family
ID=75338162
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AU2020361093A Active AU2020361093B2 (en) | 2019-10-04 | 2020-10-02 | Pharmaceutical drug containing heterocyclidene acetamide derivative |
| AU2026202464A Pending AU2026202464A1 (en) | 2019-10-04 | 2026-03-31 | Pharmaceutical Drug Containing Heterocyclidene Acetamide Derivative |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AU2026202464A Pending AU2026202464A1 (en) | 2019-10-04 | 2026-03-31 | Pharmaceutical Drug Containing Heterocyclidene Acetamide Derivative |
Country Status (17)
| Country | Link |
|---|---|
| US (3) | US12533337B2 (enExample) |
| EP (2) | EP4545095A3 (enExample) |
| JP (4) | JP7025094B2 (enExample) |
| KR (1) | KR20220078604A (enExample) |
| CN (1) | CN114585357A (enExample) |
| AU (2) | AU2020361093B2 (enExample) |
| BR (1) | BR112022005992A2 (enExample) |
| CA (1) | CA3156484A1 (enExample) |
| DK (1) | DK4043014T3 (enExample) |
| ES (1) | ES3031607T3 (enExample) |
| HU (1) | HUE072085T2 (enExample) |
| MX (2) | MX2022004027A (enExample) |
| MY (1) | MY207759A (enExample) |
| PH (1) | PH12022550805A1 (enExample) |
| PL (1) | PL4043014T3 (enExample) |
| PT (1) | PT4043014T (enExample) |
| WO (1) | WO2021066144A1 (enExample) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| BR112022005992A2 (pt) | 2019-10-04 | 2022-06-21 | Mochida Pharm Co Ltd | Fármaco contendo derivado de heterociclideno acetamida |
| JP7175431B1 (ja) | 2021-03-30 | 2022-11-18 | 千寿製薬株式会社 | ヘテロシクリデンアセトアミド誘導体含有懸濁液 |
| EP4595959A1 (en) * | 2022-09-29 | 2025-08-06 | Senju Pharmaceutical Co., Ltd. | Sterilized heterocyclidene-acetamide-derivative-containing suspension |
| EP4595960A1 (en) | 2022-09-29 | 2025-08-06 | Senju Pharmaceutical Co., Ltd. | Combination preparation containing heterocyclidene acetamide derivative |
Citations (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP1908753A1 (en) * | 2005-07-22 | 2008-04-09 | Mochida Pharmaceutical Co., Ltd. | Novel heterocyclidene acetamide derivative |
| WO2018221543A1 (ja) * | 2017-05-31 | 2018-12-06 | 持田製薬株式会社 | ヘテロシクリデンアセトアミド誘導体の結晶 |
Family Cites Families (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS5621566A (en) | 1979-08-01 | 1981-02-28 | Alpha- Shokuhin Kk | Preparation of bifun from homegrown rice and apparatus used for it |
| RU2451014C2 (ru) | 2005-07-22 | 2012-05-20 | Мотида Фармасьютикал Ко., Лтд. | Новое производное гетероциклиден ацетамида |
| CN101228131B (zh) | 2005-07-22 | 2013-01-09 | 持田制药株式会社 | 新的杂环亚基乙酰胺衍生物 |
| TW200927192A (en) * | 2007-11-19 | 2009-07-01 | Alcon Res Ltd | Use of TRPV1 receptor antagonists for treating dry eye and ocular pain |
| US20100210682A1 (en) * | 2009-02-19 | 2010-08-19 | Abbott Laboratories | Repeated Dosing of TRPV1 Antagonists |
| EP2377850A1 (en) | 2010-03-30 | 2011-10-19 | Pharmeste S.r.l. | TRPV1 vanilloid receptor antagonists with a bicyclic portion |
| WO2012045729A1 (en) * | 2010-10-05 | 2012-04-12 | Glaxo Group Limited | Imidazo [1, 2 -a] pyridine and pyrazolo [1, 5 -a] pyridine derivatives as trpv1 antagonists |
| GB201215857D0 (en) * | 2012-09-05 | 2012-10-24 | Sylentis Sau | siRNA and their use in methods and compositions for the treatment and/or prevention of eye conditions |
| JP7373909B2 (ja) | 2018-04-06 | 2023-11-06 | 株式会社シマノ | 変速制御装置および変速システム |
| BR112022005992A2 (pt) | 2019-10-04 | 2022-06-21 | Mochida Pharm Co Ltd | Fármaco contendo derivado de heterociclideno acetamida |
-
2020
- 2020-10-02 BR BR112022005992A patent/BR112022005992A2/pt unknown
- 2020-10-02 DK DK20872061.5T patent/DK4043014T3/da active
- 2020-10-02 CN CN202080069192.5A patent/CN114585357A/zh active Pending
- 2020-10-02 CA CA3156484A patent/CA3156484A1/en active Pending
- 2020-10-02 MX MX2022004027A patent/MX2022004027A/es unknown
- 2020-10-02 PL PL20872061.5T patent/PL4043014T3/pl unknown
- 2020-10-02 ES ES20872061T patent/ES3031607T3/es active Active
- 2020-10-02 EP EP25164201.3A patent/EP4545095A3/en active Pending
- 2020-10-02 PH PH1/2022/550805A patent/PH12022550805A1/en unknown
- 2020-10-02 AU AU2020361093A patent/AU2020361093B2/en active Active
- 2020-10-02 HU HUE20872061A patent/HUE072085T2/hu unknown
- 2020-10-02 WO PCT/JP2020/037548 patent/WO2021066144A1/ja not_active Ceased
- 2020-10-02 MY MYPI2022001736A patent/MY207759A/en unknown
- 2020-10-02 JP JP2021541679A patent/JP7025094B2/ja active Active
- 2020-10-02 EP EP20872061.5A patent/EP4043014B1/en active Active
- 2020-10-02 US US17/766,090 patent/US12533337B2/en active Active
- 2020-10-02 PT PT208720615T patent/PT4043014T/pt unknown
- 2020-10-02 KR KR1020227012080A patent/KR20220078604A/ko active Pending
-
2022
- 2022-02-07 JP JP2022017196A patent/JP7248836B2/ja active Active
- 2022-04-01 MX MX2025005474A patent/MX2025005474A/es unknown
- 2022-10-26 JP JP2022171542A patent/JP7801201B2/ja active Active
-
2025
- 2025-01-03 US US19/009,260 patent/US12502375B2/en active Active
- 2025-12-30 US US19/435,953 patent/US20260124171A1/en active Pending
-
2026
- 2026-01-05 JP JP2026000075A patent/JP2026042857A/ja active Pending
- 2026-03-31 AU AU2026202464A patent/AU2026202464A1/en active Pending
Patent Citations (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP1908753A1 (en) * | 2005-07-22 | 2008-04-09 | Mochida Pharmaceutical Co., Ltd. | Novel heterocyclidene acetamide derivative |
| WO2018221543A1 (ja) * | 2017-05-31 | 2018-12-06 | 持田製薬株式会社 | ヘテロシクリデンアセトアミド誘導体の結晶 |
Also Published As
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| US12502375B2 (en) | Pharmaceutical drug containing heterocyclidene acetamide derivative | |
| JP6861764B2 (ja) | 軸索再生および神経機能を促進するための方法および組成物 | |
| EP4275705B1 (en) | Pancreatitis treatment | |
| JP7082115B2 (ja) | 異常な新生血管形成を伴う眼疾患を処置するためにニンテダニブを使用する組成物および方法 | |
| JP2021508331A (ja) | 眼投与のためのw/o/wマイクロエマルジョン | |
| KR20160070077A (ko) | 안구내 투여를 위한 에피네프린-기반 안과용 조성물 및 이의 제조 방법 | |
| KR102902220B1 (ko) | 4-페닐부티르산을 함유하는 노시의 치료 또는 예방제 | |
| WO2016187722A1 (en) | Use of cannabinoids in the treatment of ocular inflammation and/or pain | |
| WO2013049621A1 (en) | Ophthalmic compositions comprising ppar-alpha agonists and methods of production and use thereof | |
| JP6509244B2 (ja) | 水晶体硬化抑制剤 | |
| WO2022123837A1 (ja) | 強膜菲薄化治療用点眼剤及び強膜菲薄化治療剤のスクリーニング方法 | |
| US20240156765A1 (en) | Methods of neuroprotection and uses thereof | |
| CN104324038A (zh) | 一种薯蓣皂苷元-3-位衍生物的用途 | |
| TW200918075A (en) | Compositions and methods for modulating endophthalmitis using fluoroquinolones | |
| BR122025000958A2 (pt) | Composições contendo derivado de heterociclideno acetamida e seus usos | |
| US20260048096A1 (en) | Methods and compositions for preserving the retinal outer nuclear layer (onl), photoreceptors, and retinal thickness | |
| Ribeiro et al. | Effects of meloxicam administered by different routes to control experimental uveitis in dogs | |
| JP2025531823A (ja) | Clec16aの機能不全または欠損に関連する症状を改善するための組成物および方法 | |
| WO2021261576A1 (ja) | 脂質分泌促進剤 | |
| WO2016199871A1 (ja) | 神経麻痺性角膜症の治療薬 | |
| BR122024009541A2 (pt) | Composição compreendendo nintedanib para tratar doenças oculares com neovascularização anormal | |
| HK40000009A (zh) | 使用尼达尼布来治疗具有异常新生血管形成的眼病的组合物和方法 |