AU2020361093B2 - Pharmaceutical drug containing heterocyclidene acetamide derivative - Google Patents

Pharmaceutical drug containing heterocyclidene acetamide derivative

Info

Publication number
AU2020361093B2
AU2020361093B2 AU2020361093A AU2020361093A AU2020361093B2 AU 2020361093 B2 AU2020361093 B2 AU 2020361093B2 AU 2020361093 A AU2020361093 A AU 2020361093A AU 2020361093 A AU2020361093 A AU 2020361093A AU 2020361093 B2 AU2020361093 B2 AU 2020361093B2
Authority
AU
Australia
Prior art keywords
dry eye
item
eye
symptom
zone
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Active
Application number
AU2020361093A
Other languages
English (en)
Other versions
AU2020361093A1 (en
Inventor
Shinya Kobayashi
Takeshi Tarui
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Senju Pharmaceutical Co Ltd
Mochida Pharmaceutical Co Ltd
Original Assignee
Senju Pharmaceutical Co Ltd
Mochida Pharmaceutical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Senju Pharmaceutical Co Ltd, Mochida Pharmaceutical Co Ltd filed Critical Senju Pharmaceutical Co Ltd
Publication of AU2020361093A1 publication Critical patent/AU2020361093A1/en
Priority to AU2026202464A priority Critical patent/AU2026202464A1/en
Application granted granted Critical
Publication of AU2020361093B2 publication Critical patent/AU2020361093B2/en
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/35—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
    • A61K31/352—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom condensed with carbocyclic rings, e.g. methantheline 
    • A61K31/353—3,4-Dihydrobenzopyrans, e.g. chroman, catechin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/02—Inorganic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/26—Carbohydrates, e.g. sugar alcohols, amino sugars, nucleic acids, mono-, di- or oligo-saccharides; Derivatives thereof, e.g. polysorbates, sorbitan fatty acid esters or glycyrrhizin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0048—Eye, e.g. artificial tears
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/10—Dispersions; Emulsions
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A61P27/04—Artificial tears; Irrigation solutions
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Ophthalmology & Optometry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Organic Chemistry (AREA)
  • Dispersion Chemistry (AREA)
  • Molecular Biology (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Inorganic Chemistry (AREA)
  • Biochemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicinal Preparation (AREA)
AU2020361093A 2019-10-04 2020-10-02 Pharmaceutical drug containing heterocyclidene acetamide derivative Active AU2020361093B2 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
AU2026202464A AU2026202464A1 (en) 2019-10-04 2026-03-31 Pharmaceutical Drug Containing Heterocyclidene Acetamide Derivative

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP2019184053 2019-10-04
JP2019-184053 2019-10-04
PCT/JP2020/037548 WO2021066144A1 (ja) 2019-10-04 2020-10-02 ヘテロシクリデンアセトアミド誘導体含有医薬

Related Child Applications (1)

Application Number Title Priority Date Filing Date
AU2026202464A Division AU2026202464A1 (en) 2019-10-04 2026-03-31 Pharmaceutical Drug Containing Heterocyclidene Acetamide Derivative

Publications (2)

Publication Number Publication Date
AU2020361093A1 AU2020361093A1 (en) 2022-05-19
AU2020361093B2 true AU2020361093B2 (en) 2026-04-30

Family

ID=75338162

Family Applications (2)

Application Number Title Priority Date Filing Date
AU2020361093A Active AU2020361093B2 (en) 2019-10-04 2020-10-02 Pharmaceutical drug containing heterocyclidene acetamide derivative
AU2026202464A Pending AU2026202464A1 (en) 2019-10-04 2026-03-31 Pharmaceutical Drug Containing Heterocyclidene Acetamide Derivative

Family Applications After (1)

Application Number Title Priority Date Filing Date
AU2026202464A Pending AU2026202464A1 (en) 2019-10-04 2026-03-31 Pharmaceutical Drug Containing Heterocyclidene Acetamide Derivative

Country Status (17)

Country Link
US (3) US12533337B2 (enExample)
EP (2) EP4545095A3 (enExample)
JP (4) JP7025094B2 (enExample)
KR (1) KR20220078604A (enExample)
CN (1) CN114585357A (enExample)
AU (2) AU2020361093B2 (enExample)
BR (1) BR112022005992A2 (enExample)
CA (1) CA3156484A1 (enExample)
DK (1) DK4043014T3 (enExample)
ES (1) ES3031607T3 (enExample)
HU (1) HUE072085T2 (enExample)
MX (2) MX2022004027A (enExample)
MY (1) MY207759A (enExample)
PH (1) PH12022550805A1 (enExample)
PL (1) PL4043014T3 (enExample)
PT (1) PT4043014T (enExample)
WO (1) WO2021066144A1 (enExample)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BR112022005992A2 (pt) 2019-10-04 2022-06-21 Mochida Pharm Co Ltd Fármaco contendo derivado de heterociclideno acetamida
JP7175431B1 (ja) 2021-03-30 2022-11-18 千寿製薬株式会社 ヘテロシクリデンアセトアミド誘導体含有懸濁液
EP4595959A1 (en) * 2022-09-29 2025-08-06 Senju Pharmaceutical Co., Ltd. Sterilized heterocyclidene-acetamide-derivative-containing suspension
EP4595960A1 (en) 2022-09-29 2025-08-06 Senju Pharmaceutical Co., Ltd. Combination preparation containing heterocyclidene acetamide derivative

Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1908753A1 (en) * 2005-07-22 2008-04-09 Mochida Pharmaceutical Co., Ltd. Novel heterocyclidene acetamide derivative
WO2018221543A1 (ja) * 2017-05-31 2018-12-06 持田製薬株式会社 ヘテロシクリデンアセトアミド誘導体の結晶

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5621566A (en) 1979-08-01 1981-02-28 Alpha- Shokuhin Kk Preparation of bifun from homegrown rice and apparatus used for it
RU2451014C2 (ru) 2005-07-22 2012-05-20 Мотида Фармасьютикал Ко., Лтд. Новое производное гетероциклиден ацетамида
CN101228131B (zh) 2005-07-22 2013-01-09 持田制药株式会社 新的杂环亚基乙酰胺衍生物
TW200927192A (en) * 2007-11-19 2009-07-01 Alcon Res Ltd Use of TRPV1 receptor antagonists for treating dry eye and ocular pain
US20100210682A1 (en) * 2009-02-19 2010-08-19 Abbott Laboratories Repeated Dosing of TRPV1 Antagonists
EP2377850A1 (en) 2010-03-30 2011-10-19 Pharmeste S.r.l. TRPV1 vanilloid receptor antagonists with a bicyclic portion
WO2012045729A1 (en) * 2010-10-05 2012-04-12 Glaxo Group Limited Imidazo [1, 2 -a] pyridine and pyrazolo [1, 5 -a] pyridine derivatives as trpv1 antagonists
GB201215857D0 (en) * 2012-09-05 2012-10-24 Sylentis Sau siRNA and their use in methods and compositions for the treatment and/or prevention of eye conditions
JP7373909B2 (ja) 2018-04-06 2023-11-06 株式会社シマノ 変速制御装置および変速システム
BR112022005992A2 (pt) 2019-10-04 2022-06-21 Mochida Pharm Co Ltd Fármaco contendo derivado de heterociclideno acetamida

Patent Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1908753A1 (en) * 2005-07-22 2008-04-09 Mochida Pharmaceutical Co., Ltd. Novel heterocyclidene acetamide derivative
WO2018221543A1 (ja) * 2017-05-31 2018-12-06 持田製薬株式会社 ヘテロシクリデンアセトアミド誘導体の結晶

Also Published As

Publication number Publication date
PT4043014T (pt) 2025-06-09
MX2025005474A (es) 2025-06-02
JP2023011735A (ja) 2023-01-24
JP7801201B2 (ja) 2026-01-16
AU2026202464A1 (en) 2026-04-16
US20260124171A1 (en) 2026-05-07
JP2022065024A (ja) 2022-04-26
JP7025094B2 (ja) 2022-02-24
KR20220078604A (ko) 2022-06-10
EP4545095A2 (en) 2025-04-30
JP2026042857A (ja) 2026-03-11
JP7248836B2 (ja) 2023-03-29
EP4043014A1 (en) 2022-08-17
EP4545095A3 (en) 2025-07-02
JPWO2021066144A1 (ja) 2021-12-02
PL4043014T3 (pl) 2025-08-11
CN114585357A (zh) 2022-06-03
US20250134854A1 (en) 2025-05-01
EP4043014B1 (en) 2025-03-19
US20220370404A1 (en) 2022-11-24
PH12022550805A1 (en) 2023-10-02
WO2021066144A1 (ja) 2021-04-08
US12502375B2 (en) 2025-12-23
MX2022004027A (es) 2022-07-19
HUE072085T2 (hu) 2025-10-28
MY207759A (en) 2025-03-17
DK4043014T3 (da) 2025-06-23
US12533337B2 (en) 2026-01-27
BR112022005992A2 (pt) 2022-06-21
CA3156484A1 (en) 2021-04-08
EP4043014A4 (en) 2023-10-11
ES3031607T3 (en) 2025-07-09
AU2020361093A1 (en) 2022-05-19

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