KR20220078604A - 헤테로시클리덴아세트아미드 유도체 함유 의약 - Google Patents

헤테로시클리덴아세트아미드 유도체 함유 의약 Download PDF

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Publication number
KR20220078604A
KR20220078604A KR1020227012080A KR20227012080A KR20220078604A KR 20220078604 A KR20220078604 A KR 20220078604A KR 1020227012080 A KR1020227012080 A KR 1020227012080A KR 20227012080 A KR20227012080 A KR 20227012080A KR 20220078604 A KR20220078604 A KR 20220078604A
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South Korea
Prior art keywords
eye
dry eye
item
composition
ylidene
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KR1020227012080A
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English (en)
Korean (ko)
Inventor
다케시 다루이
신야 고바야시
Original Assignee
센주 세이야꾸 가부시키가이샤
모찌다 세이야쿠 가부시끼가이샤
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Publication of KR20220078604A publication Critical patent/KR20220078604A/ko
Pending legal-status Critical Current

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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/35—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
    • A61K31/352—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom condensed with carbocyclic rings, e.g. methantheline 
    • A61K31/353—3,4-Dihydrobenzopyrans, e.g. chroman, catechin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/02—Inorganic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/26—Carbohydrates, e.g. sugar alcohols, amino sugars, nucleic acids, mono-, di- or oligo-saccharides; Derivatives thereof, e.g. polysorbates, sorbitan fatty acid esters or glycyrrhizin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0048—Eye, e.g. artificial tears
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/10—Dispersions; Emulsions
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A61P27/04—Artificial tears; Irrigation solutions
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Ophthalmology & Optometry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Organic Chemistry (AREA)
  • Dispersion Chemistry (AREA)
  • Molecular Biology (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Inorganic Chemistry (AREA)
  • Biochemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicinal Preparation (AREA)
KR1020227012080A 2019-10-04 2020-10-02 헤테로시클리덴아세트아미드 유도체 함유 의약 Pending KR20220078604A (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP2019184053 2019-10-04
JPJP-P-2019-184053 2019-10-04
PCT/JP2020/037548 WO2021066144A1 (ja) 2019-10-04 2020-10-02 ヘテロシクリデンアセトアミド誘導体含有医薬

Publications (1)

Publication Number Publication Date
KR20220078604A true KR20220078604A (ko) 2022-06-10

Family

ID=75338162

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1020227012080A Pending KR20220078604A (ko) 2019-10-04 2020-10-02 헤테로시클리덴아세트아미드 유도체 함유 의약

Country Status (17)

Country Link
US (3) US12533337B2 (enExample)
EP (2) EP4545095A3 (enExample)
JP (4) JP7025094B2 (enExample)
KR (1) KR20220078604A (enExample)
CN (1) CN114585357A (enExample)
AU (2) AU2020361093B2 (enExample)
BR (1) BR112022005992A2 (enExample)
CA (1) CA3156484A1 (enExample)
DK (1) DK4043014T3 (enExample)
ES (1) ES3031607T3 (enExample)
HU (1) HUE072085T2 (enExample)
MX (2) MX2022004027A (enExample)
MY (1) MY207759A (enExample)
PH (1) PH12022550805A1 (enExample)
PL (1) PL4043014T3 (enExample)
PT (1) PT4043014T (enExample)
WO (1) WO2021066144A1 (enExample)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BR112022005992A2 (pt) 2019-10-04 2022-06-21 Mochida Pharm Co Ltd Fármaco contendo derivado de heterociclideno acetamida
JP7175431B1 (ja) 2021-03-30 2022-11-18 千寿製薬株式会社 ヘテロシクリデンアセトアミド誘導体含有懸濁液
EP4595959A1 (en) * 2022-09-29 2025-08-06 Senju Pharmaceutical Co., Ltd. Sterilized heterocyclidene-acetamide-derivative-containing suspension
EP4595960A1 (en) 2022-09-29 2025-08-06 Senju Pharmaceutical Co., Ltd. Combination preparation containing heterocyclidene acetamide derivative

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5621566A (en) 1979-08-01 1981-02-28 Alpha- Shokuhin Kk Preparation of bifun from homegrown rice and apparatus used for it
RU2451014C2 (ru) 2005-07-22 2012-05-20 Мотида Фармасьютикал Ко., Лтд. Новое производное гетероциклиден ацетамида
JP4754566B2 (ja) 2005-07-22 2011-08-24 持田製薬株式会社 新規なヘテロシクリデンアセトアミド誘導体
CN101228131B (zh) 2005-07-22 2013-01-09 持田制药株式会社 新的杂环亚基乙酰胺衍生物
TW200927192A (en) * 2007-11-19 2009-07-01 Alcon Res Ltd Use of TRPV1 receptor antagonists for treating dry eye and ocular pain
US20100210682A1 (en) * 2009-02-19 2010-08-19 Abbott Laboratories Repeated Dosing of TRPV1 Antagonists
EP2377850A1 (en) 2010-03-30 2011-10-19 Pharmeste S.r.l. TRPV1 vanilloid receptor antagonists with a bicyclic portion
WO2012045729A1 (en) * 2010-10-05 2012-04-12 Glaxo Group Limited Imidazo [1, 2 -a] pyridine and pyrazolo [1, 5 -a] pyridine derivatives as trpv1 antagonists
GB201215857D0 (en) * 2012-09-05 2012-10-24 Sylentis Sau siRNA and their use in methods and compositions for the treatment and/or prevention of eye conditions
JP6230743B1 (ja) 2017-05-31 2017-11-15 持田製薬株式会社 ヘテロシクリデンアセトアミド誘導体の結晶
JP7373909B2 (ja) 2018-04-06 2023-11-06 株式会社シマノ 変速制御装置および変速システム
BR112022005992A2 (pt) 2019-10-04 2022-06-21 Mochida Pharm Co Ltd Fármaco contendo derivado de heterociclideno acetamida

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
파마시아 Vol.50 No.3 2014:201 내지 206

Also Published As

Publication number Publication date
PT4043014T (pt) 2025-06-09
MX2025005474A (es) 2025-06-02
AU2020361093B2 (en) 2026-04-30
JP2023011735A (ja) 2023-01-24
JP7801201B2 (ja) 2026-01-16
AU2026202464A1 (en) 2026-04-16
US20260124171A1 (en) 2026-05-07
JP2022065024A (ja) 2022-04-26
JP7025094B2 (ja) 2022-02-24
EP4545095A2 (en) 2025-04-30
JP2026042857A (ja) 2026-03-11
JP7248836B2 (ja) 2023-03-29
EP4043014A1 (en) 2022-08-17
EP4545095A3 (en) 2025-07-02
JPWO2021066144A1 (ja) 2021-12-02
PL4043014T3 (pl) 2025-08-11
CN114585357A (zh) 2022-06-03
US20250134854A1 (en) 2025-05-01
EP4043014B1 (en) 2025-03-19
US20220370404A1 (en) 2022-11-24
PH12022550805A1 (en) 2023-10-02
WO2021066144A1 (ja) 2021-04-08
US12502375B2 (en) 2025-12-23
MX2022004027A (es) 2022-07-19
HUE072085T2 (hu) 2025-10-28
MY207759A (en) 2025-03-17
DK4043014T3 (da) 2025-06-23
US12533337B2 (en) 2026-01-27
BR112022005992A2 (pt) 2022-06-21
CA3156484A1 (en) 2021-04-08
EP4043014A4 (en) 2023-10-11
ES3031607T3 (en) 2025-07-09
AU2020361093A1 (en) 2022-05-19

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