AU2015216957B2 - Aromatic heterocyclic compounds as antiinflammatory compounds - Google Patents

Aromatic heterocyclic compounds as antiinflammatory compounds Download PDF

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AU2015216957B2
AU2015216957B2 AU2015216957A AU2015216957A AU2015216957B2 AU 2015216957 B2 AU2015216957 B2 AU 2015216957B2 AU 2015216957 A AU2015216957 A AU 2015216957A AU 2015216957 A AU2015216957 A AU 2015216957A AU 2015216957 B2 AU2015216957 B2 AU 2015216957B2
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compound
formula
asthma
disease
treatment
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AU2015216957A1 (en
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Euan Alexander Fraser Fordyce
John King-Underwood
Alistair Ian Longshaw
Stuart Thomas Onions
Jennifer Diane Venable
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Respivert Ltd
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Respivert Ltd
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    • AHUMAN NECESSITIES
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    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/007Pulmonary tract; Aromatherapy
    • A61K9/0073Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy
    • A61K9/0075Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy for inhalation via a dry powder inhaler [DPI], e.g. comprising micronized drug mixed with lactose carrier particles
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    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
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    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
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    • A61K31/55Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
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AU2015216957A 2014-02-14 2015-02-13 Aromatic heterocyclic compounds as antiinflammatory compounds Active AU2015216957B2 (en)

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AU2019204525A AU2019204525B2 (en) 2014-02-14 2019-06-26 Aromatic heterocyclic compounds as antiinflammatory compounds

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US201461940282P 2014-02-14 2014-02-14
US61/940,282 2014-02-14
US201461941064P 2014-02-18 2014-02-18
US61/941,064 2014-02-18
PCT/EP2015/053151 WO2015121444A1 (en) 2014-02-14 2015-02-13 Aromatic heterocyclic compounds as antiinflammatory compounds

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AU2015216957B2 true AU2015216957B2 (en) 2019-04-04

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AU2015216705A Active AU2015216705B2 (en) 2014-02-14 2015-02-13 Pyrazolyl-ureas as kinase inhibitors
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US (8) US9447076B2 (https=)
EP (4) EP3357919B1 (https=)
JP (4) JP6586098B2 (https=)
KR (1) KR102413704B1 (https=)
CN (4) CN113264921B (https=)
AU (3) AU2015216957B2 (https=)
BR (1) BR112016015838B1 (https=)
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NZ601085A (en) 2010-02-01 2015-04-24 Cancer Rec Tech Ltd 1-(5-tert-butyl-2-phenyl-2h-pyrazol-3-yl)-3-[2-fluoro-4-(1-methyl-2-oxo-2,3-dihydro-1h-imidazo[4,5-b]pyridin-7-yloxy)-phenyl]-urea and related compounds and their use in therapy
EP2578582A1 (en) 2011-10-03 2013-04-10 Respivert Limited 1-Pyrazolyl-3-(4-((2-anilinopyrimidin-4-yl)oxy)napththalen-1-yl)ureas as p38 MAP kinase inhibitors
CN103917536B (zh) * 2011-10-03 2016-07-06 瑞斯比维特有限公司 1-吡唑基-3-(4-((2-(苯氨基)嘧啶-4-基)氧基)萘-1-基)脲用作p38 MAP激酶抑制剂
GB201214750D0 (en) 2012-08-17 2012-10-03 Respivert Ltd Compounds
EP2890701B1 (en) 2012-08-29 2017-03-29 Respivert Limited Kinase inhibitors
US20150210722A1 (en) 2012-08-29 2015-07-30 Respivert Limited Kinase inhibitors
US20150225373A1 (en) 2012-08-29 2015-08-13 Respivert Limited Kinase inhibitors
WO2014076484A1 (en) 2012-11-16 2014-05-22 Respivert Limited Kinase inhibitors
EP2970190A1 (en) 2013-03-14 2016-01-20 Respivert Limited Kinase inhibitors
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