AU2014264342B2 - Antiemetic extended release solid dosage forms - Google Patents

Antiemetic extended release solid dosage forms Download PDF

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Publication number
AU2014264342B2
AU2014264342B2 AU2014264342A AU2014264342A AU2014264342B2 AU 2014264342 B2 AU2014264342 B2 AU 2014264342B2 AU 2014264342 A AU2014264342 A AU 2014264342A AU 2014264342 A AU2014264342 A AU 2014264342A AU 2014264342 B2 AU2014264342 B2 AU 2014264342B2
Authority
AU
Australia
Prior art keywords
ondansetron
tablet
drug
release
test
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Active
Application number
AU2014264342A
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English (en)
Other versions
AU2014264342A1 (en
Inventor
Reza Fathi
Gilead RADAY
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Redhill Biopharma Ltd
Original Assignee
Redhill Biopharma Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=51528070&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AU2014264342(B2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Redhill Biopharma Ltd filed Critical Redhill Biopharma Ltd
Publication of AU2014264342A1 publication Critical patent/AU2014264342A1/en
Application granted granted Critical
Publication of AU2014264342B2 publication Critical patent/AU2014264342B2/en
Active legal-status Critical Current
Anticipated expiration legal-status Critical

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Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806—Coating materials
    • A61K9/2833—Organic macromolecular compounds
    • A61K9/286—Polysaccharides, e.g. gums; Cyclodextrin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4164—1,3-Diazoles
    • A61K31/4178—1,3-Diazoles not condensed 1,3-diazoles and containing further heterocyclic rings, e.g. pilocarpine, nitrofurantoin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2086—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat
    • A61K9/209—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat containing drug in at least two layers or in the core and in at least one outer layer
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806—Coating materials
    • A61K9/2833—Organic macromolecular compounds
    • A61K9/286—Polysaccharides, e.g. gums; Cyclodextrin
    • A61K9/2866—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2886—Dragees; Coated pills or tablets, e.g. with film or compression coating having two or more different drug-free coatings; Tablets of the type inert core-drug layer-inactive layer
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806—Coating materials
    • A61K9/2833—Organic macromolecular compounds
    • A61K9/284—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone
    • A61K9/2846—Poly(meth)acrylates

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Hospice & Palliative Care (AREA)
  • Otolaryngology (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
AU2014264342A 2013-03-14 2014-03-14 Antiemetic extended release solid dosage forms Active AU2014264342B2 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201361782395P 2013-03-14 2013-03-14
US61/782,395 2013-03-14
PCT/IB2014/001633 WO2014181195A2 (en) 2013-03-14 2014-03-14 Antiemetic extended release solid dosage forms

Publications (2)

Publication Number Publication Date
AU2014264342A1 AU2014264342A1 (en) 2015-10-01
AU2014264342B2 true AU2014264342B2 (en) 2017-05-18

Family

ID=51528070

Family Applications (1)

Application Number Title Priority Date Filing Date
AU2014264342A Active AU2014264342B2 (en) 2013-03-14 2014-03-14 Antiemetic extended release solid dosage forms

Country Status (19)

Country Link
US (5) US9636305B2 (enExample)
EP (1) EP2983664B1 (enExample)
JP (1) JP6282676B2 (enExample)
KR (1) KR102270521B1 (enExample)
CN (2) CN105530935A (enExample)
AU (1) AU2014264342B2 (enExample)
BR (1) BR112015022398B1 (enExample)
CA (1) CA2905553C (enExample)
CL (1) CL2015002666A1 (enExample)
ES (1) ES2946985T3 (enExample)
HK (1) HK1223012A1 (enExample)
IL (1) IL241580B (enExample)
MX (1) MX378261B (enExample)
NZ (1) NZ712159A (enExample)
PH (1) PH12015502093B1 (enExample)
RU (1) RU2679448C2 (enExample)
SG (1) SG11201507450TA (enExample)
WO (2) WO2014181195A2 (enExample)
ZA (1) ZA201506961B (enExample)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RU2679448C2 (ru) 2013-03-14 2019-02-11 Редхилл Байофарма Лтд. Твердые лекарственные формы, обладающие противорвотным действием, с замедленным высвобождением
MX373002B (es) 2014-03-11 2020-04-30 Redhill Biopharma Ltd Formas de dosificacion sólida de liberación extendida de ondansetrón para tratar bien sea síntomas de náusea, vómito o diarrea
CA2910865C (en) 2014-07-15 2016-11-29 Isa Odidi Compositions and methods for reducing overdose
KR102300335B1 (ko) * 2018-10-19 2021-09-10 주식회사 삼양홀딩스 아프레피탄트의 경구용 조성물
WO2024096892A1 (en) * 2022-11-03 2024-05-10 Lumos Pharma, Inc. Compactable oral formulations of ibutamoren

Citations (1)

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WO2003009829A2 (en) * 2001-03-19 2003-02-06 L.A.M. Pharmaceutical Corporation Antiemetic, anti-motion sustained release drug delivery system

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Also Published As

Publication number Publication date
WO2014181195A2 (en) 2014-11-13
PH12015502093B1 (en) 2018-09-26
MX2015012970A (es) 2016-04-11
BR112015022398A2 (pt) 2017-07-18
EP2983664A2 (en) 2016-02-17
HK1223012A1 (zh) 2017-07-21
ZA201506961B (en) 2017-03-29
US20140271887A1 (en) 2014-09-18
CA2905553A1 (en) 2014-11-13
AU2014264342A1 (en) 2015-10-01
CL2015002666A1 (es) 2017-02-17
WO2014181195A3 (en) 2015-12-17
BR112015022398B1 (pt) 2022-01-11
KR20150127253A (ko) 2015-11-16
WO2014184662A3 (en) 2015-04-02
ES2946985T3 (es) 2023-07-31
EP2983664A4 (en) 2017-01-04
US20200330392A1 (en) 2020-10-22
NZ712159A (en) 2019-12-20
IL241580B (en) 2020-08-31
BR112015022398A8 (pt) 2019-11-26
CN105530935A (zh) 2016-04-27
CN112274489A (zh) 2021-01-29
RU2679448C2 (ru) 2019-02-11
US9636305B2 (en) 2017-05-02
US20180028452A1 (en) 2018-02-01
US20170189340A1 (en) 2017-07-06
KR102270521B1 (ko) 2021-06-30
JP2016512493A (ja) 2016-04-28
WO2014184662A2 (en) 2014-11-20
US20140271851A1 (en) 2014-09-18
MX378261B (es) 2025-03-10
RU2015143993A (ru) 2017-04-20
CA2905553C (en) 2021-04-06
SG11201507450TA (en) 2015-10-29
PH12015502093A1 (en) 2016-01-18
RU2015143993A3 (enExample) 2018-03-21
JP6282676B2 (ja) 2018-02-21
EP2983664B1 (en) 2023-04-19

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FGA Letters patent sealed or granted (standard patent)