AU2009257692A1 - Methods of treating alpha adrenergic mediated conditions - Google Patents
Methods of treating alpha adrenergic mediated conditions Download PDFInfo
- Publication number
- AU2009257692A1 AU2009257692A1 AU2009257692A AU2009257692A AU2009257692A1 AU 2009257692 A1 AU2009257692 A1 AU 2009257692A1 AU 2009257692 A AU2009257692 A AU 2009257692A AU 2009257692 A AU2009257692 A AU 2009257692A AU 2009257692 A1 AU2009257692 A1 AU 2009257692A1
- Authority
- AU
- Australia
- Prior art keywords
- amine
- dihydro
- imidazol
- benzyl
- pain
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
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| US7902247B2 (en) * | 2008-01-09 | 2011-03-08 | Allergan, Inc. | Substituted-aryl-2-phenylethyl-1H-imidazole compounds as subtype selective modulators of alpha 2B and/or alpha 2C adrenergic receptors |
| PL2605771T3 (pl) * | 2010-08-16 | 2018-10-31 | Allergan, Inc. | Sposób aktywacji limfocytów t regulacyjnych za pomocą agonistów receptorów alfa-2b-adrenergicznych |
| JP6756435B2 (ja) * | 2014-03-31 | 2020-09-16 | ザ スクリプス リサーチ インスティテュート | Ｔｒａｉｌ誘導のためのファーマコフォア |
| EP3700536A4 (en) | 2017-10-27 | 2021-11-17 | Shanghai Yao Yuan Biotechnology Co., Ltd. | COMPOSITIONS AND PROCEDURES FOR MODULATING IMMUNE REACTION BY ACTIVATING ALPHA-PROTEIN KINASE 1 |
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| US4256755A (en) | 1980-04-28 | 1981-03-17 | E. I. Du Pont De Nemours & Company | Method of using N-substituted dihydro-2-oxazolamines as analgesics |
| FR2806082B1 (fr) * | 2000-03-07 | 2002-05-17 | Adir | Nouveaux composes bicycliques antagonistes des recepteurs de la vitronectine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent |
| WO2002089794A1 (en) * | 2001-05-07 | 2002-11-14 | Universite Catholique De Louvain | Method for treating neuropathic pain and pharmaceutical preparation therefor |
| EP1333028A1 (en) * | 2002-01-31 | 2003-08-06 | Boehringer Ingelheim Pharma GmbH & Co.KG | 2'-Halo-3',5'-dialkoxyphen-1'-yl-imino-2-imidazolidine derivatives and the use thereof for the treatment of urinary incontinence |
| US7345065B2 (en) | 2002-05-21 | 2008-03-18 | Allergan, Inc. | Methods and compositions for alleviating pain |
| CN101287366A (zh) | 2005-05-19 | 2008-10-15 | 拜尔农作物科学股份公司 | 杀虫的取代的苄基氨基杂环及杂芳基衍生物 |
| WO2008123821A1 (en) * | 2007-03-01 | 2008-10-16 | Albireo Ab | 4, 5-dihydro-lh-imidazol-2-amine derivatives for use in the treatment of respiratory, cardiovascular, neurological or gastrointestinal disorders |
| CN101687812A (zh) * | 2007-07-02 | 2010-03-31 | 弗·哈夫曼-拉罗切有限公司 | 对痕量胺相关受体(taar)具有良好亲和性的2-咪唑啉化合物 |
| WO2009052075A2 (en) * | 2007-10-18 | 2009-04-23 | Allergan, Inc. | Method of treating motor disorders with alpha-2b adrenergic receptor agonists |
-
2009
- 2009-06-05 ES ES09763343.2T patent/ES2672777T3/es active Active
- 2009-06-05 WO PCT/US2009/046432 patent/WO2009152052A1/en not_active Ceased
- 2009-06-05 CN CN200980126849.0A patent/CN102099032B/zh not_active Expired - Fee Related
- 2009-06-05 AU AU2009257692A patent/AU2009257692A1/en not_active Abandoned
- 2009-06-05 SI SI200931858T patent/SI2303264T1/en unknown
- 2009-06-05 PL PL09763343T patent/PL2303264T3/pl unknown
- 2009-06-05 CA CA2959793A patent/CA2959793A1/en not_active Abandoned
- 2009-06-05 US US12/479,129 patent/US8071636B2/en active Active
- 2009-06-05 PL PL15165926T patent/PL2932968T3/pl unknown
- 2009-06-05 JP JP2011513592A patent/JP5571072B2/ja not_active Expired - Fee Related
- 2009-06-05 ES ES15165926.5T patent/ES2665293T3/es active Active
- 2009-06-05 TR TR2018/02766T patent/TR201802766T4/tr unknown
- 2009-06-05 EP EP09763343.2A patent/EP2303264B1/en active Active
- 2009-06-05 EP EP15165926.5A patent/EP2932968B1/en active Active
- 2009-06-05 DK DK15165926.5T patent/DK2932968T3/en active
- 2009-06-05 EP EP11174152A patent/EP2377534A1/en not_active Withdrawn
- 2009-06-05 HU HUE09763343A patent/HUE039357T2/hu unknown
- 2009-06-05 PT PT97633432T patent/PT2303264T/pt unknown
- 2009-06-05 PT PT151659265T patent/PT2932968T/pt unknown
- 2009-06-05 CA CA2744929A patent/CA2744929C/en active Active
- 2009-06-05 CA CA3133261A patent/CA3133261A1/en not_active Abandoned
- 2009-06-05 DK DK09763343.2T patent/DK2303264T3/en active
-
2011
- 2011-10-17 US US13/274,471 patent/US20120035235A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| PT2932968T (pt) | 2018-03-13 |
| EP2932968B1 (en) | 2018-01-17 |
| DK2303264T3 (en) | 2018-05-22 |
| EP2303264A1 (en) | 2011-04-06 |
| US8071636B2 (en) | 2011-12-06 |
| JP5571072B2 (ja) | 2014-08-13 |
| WO2009152052A8 (en) | 2010-11-11 |
| WO2009152052A1 (en) | 2009-12-17 |
| CA2744929C (en) | 2017-07-25 |
| JP2011522893A (ja) | 2011-08-04 |
| TR201802766T4 (tr) | 2018-03-21 |
| PL2303264T3 (pl) | 2018-08-31 |
| ES2665293T3 (es) | 2018-04-25 |
| EP2932968A1 (en) | 2015-10-21 |
| ES2672777T3 (es) | 2018-06-18 |
| HK1214132A1 (en) | 2016-07-22 |
| PL2932968T3 (pl) | 2018-06-29 |
| US20090306161A1 (en) | 2009-12-10 |
| CA2959793A1 (en) | 2009-12-17 |
| CA3133261A1 (en) | 2009-12-17 |
| CN102099032B (zh) | 2014-07-09 |
| EP2303264B1 (en) | 2018-04-04 |
| CN102099032A (zh) | 2011-06-15 |
| EP2377534A1 (en) | 2011-10-19 |
| SI2303264T1 (en) | 2018-08-31 |
| DK2932968T3 (en) | 2018-03-12 |
| PT2303264T (pt) | 2018-05-14 |
| HUE039357T2 (hu) | 2018-12-28 |
| CA2744929A1 (en) | 2009-12-17 |
| US20120035235A1 (en) | 2012-02-09 |
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