DK2932968T3 - CONNECTION TO TREATMENT OF ALFA-ADRENERG MEDIED CONDITIONS - Google Patents
CONNECTION TO TREATMENT OF ALFA-ADRENERG MEDIED CONDITIONS Download PDFInfo
- Publication number
- DK2932968T3 DK2932968T3 DK15165926.5T DK15165926T DK2932968T3 DK 2932968 T3 DK2932968 T3 DK 2932968T3 DK 15165926 T DK15165926 T DK 15165926T DK 2932968 T3 DK2932968 T3 DK 2932968T3
- Authority
- DK
- Denmark
- Prior art keywords
- pain
- amine
- dihydro
- tautomer
- pharmaceutically acceptable
- Prior art date
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Landscapes
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
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- Engineering & Computer Science (AREA)
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- General Health & Medical Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
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- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Organic Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
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- Biomedical Technology (AREA)
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- Diabetes (AREA)
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- Heart & Thoracic Surgery (AREA)
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- Child & Adolescent Psychology (AREA)
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Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US5983708P | 2008-06-09 | 2008-06-09 | |
| EP09763343.2A EP2303264B1 (en) | 2008-06-09 | 2009-06-05 | Methods of treating alpha adrenergic mediated conditions using imidazoline derivatives |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DK2932968T3 true DK2932968T3 (en) | 2018-03-12 |
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| DK15165926.5T DK2932968T3 (en) | 2008-06-09 | 2009-06-05 | CONNECTION TO TREATMENT OF ALFA-ADRENERG MEDIED CONDITIONS |
| DK09763343.2T DK2303264T3 (en) | 2008-06-09 | 2009-06-05 | METHODS FOR TREATING ALPHA-ADRENERG-MEDIATED CONDITIONS USING IMIDAZOLINE DERIVATIVES |
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| Application Number | Title | Priority Date | Filing Date |
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| DK09763343.2T DK2303264T3 (en) | 2008-06-09 | 2009-06-05 | METHODS FOR TREATING ALPHA-ADRENERG-MEDIATED CONDITIONS USING IMIDAZOLINE DERIVATIVES |
Country Status (14)
| Country | Link |
|---|---|
| US (2) | US8071636B2 (https=) |
| EP (3) | EP2303264B1 (https=) |
| JP (1) | JP5571072B2 (https=) |
| CN (1) | CN102099032B (https=) |
| AU (1) | AU2009257692A1 (https=) |
| CA (3) | CA2959793A1 (https=) |
| DK (2) | DK2932968T3 (https=) |
| ES (2) | ES2672777T3 (https=) |
| HU (1) | HUE039357T2 (https=) |
| PL (2) | PL2303264T3 (https=) |
| PT (2) | PT2303264T (https=) |
| SI (1) | SI2303264T1 (https=) |
| TR (1) | TR201802766T4 (https=) |
| WO (1) | WO2009152052A1 (https=) |
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| US20120083508A1 (en) * | 2006-12-22 | 2012-04-05 | Allergan, Inc. | Alpha-2b receptor agonist and anticonvulsant compositions for treating chronic pain |
| US7902247B2 (en) * | 2008-01-09 | 2011-03-08 | Allergan, Inc. | Substituted-aryl-2-phenylethyl-1H-imidazole compounds as subtype selective modulators of alpha 2B and/or alpha 2C adrenergic receptors |
| PL2605771T3 (pl) * | 2010-08-16 | 2018-10-31 | Allergan, Inc. | Sposób aktywacji limfocytów t regulacyjnych za pomocą agonistów receptorów alfa-2b-adrenergicznych |
| JP6756435B2 (ja) * | 2014-03-31 | 2020-09-16 | ザ スクリプス リサーチ インスティテュート | Ｔｒａｉｌ誘導のためのファーマコフォア |
| EP3700536A4 (en) | 2017-10-27 | 2021-11-17 | Shanghai Yao Yuan Biotechnology Co., Ltd. | COMPOSITIONS AND PROCEDURES FOR MODULATING IMMUNE REACTION BY ACTIVATING ALPHA-PROTEIN KINASE 1 |
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| NL6708160A (https=) * | 1966-06-30 | 1968-01-02 | ||
| DE2259160A1 (de) * | 1972-12-02 | 1974-06-06 | Boehringer Sohn Ingelheim | Neue substituierte 2-phenylaminoimidazoline, deren saeureadditionssalze und verfahren zur herstellung derselben sowie ihre verwendung als arzneimittel |
| US4256755A (en) | 1980-04-28 | 1981-03-17 | E. I. Du Pont De Nemours & Company | Method of using N-substituted dihydro-2-oxazolamines as analgesics |
| FR2806082B1 (fr) * | 2000-03-07 | 2002-05-17 | Adir | Nouveaux composes bicycliques antagonistes des recepteurs de la vitronectine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent |
| WO2002089794A1 (en) * | 2001-05-07 | 2002-11-14 | Universite Catholique De Louvain | Method for treating neuropathic pain and pharmaceutical preparation therefor |
| EP1333028A1 (en) * | 2002-01-31 | 2003-08-06 | Boehringer Ingelheim Pharma GmbH & Co.KG | 2'-Halo-3',5'-dialkoxyphen-1'-yl-imino-2-imidazolidine derivatives and the use thereof for the treatment of urinary incontinence |
| US7345065B2 (en) | 2002-05-21 | 2008-03-18 | Allergan, Inc. | Methods and compositions for alleviating pain |
| CN101287366A (zh) | 2005-05-19 | 2008-10-15 | 拜尔农作物科学股份公司 | 杀虫的取代的苄基氨基杂环及杂芳基衍生物 |
| WO2008123821A1 (en) * | 2007-03-01 | 2008-10-16 | Albireo Ab | 4, 5-dihydro-lh-imidazol-2-amine derivatives for use in the treatment of respiratory, cardiovascular, neurological or gastrointestinal disorders |
| CN101687812A (zh) * | 2007-07-02 | 2010-03-31 | 弗·哈夫曼-拉罗切有限公司 | 对痕量胺相关受体(taar)具有良好亲和性的2-咪唑啉化合物 |
| WO2009052075A2 (en) * | 2007-10-18 | 2009-04-23 | Allergan, Inc. | Method of treating motor disorders with alpha-2b adrenergic receptor agonists |
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Also Published As
| Publication number | Publication date |
|---|---|
| PT2932968T (pt) | 2018-03-13 |
| EP2932968B1 (en) | 2018-01-17 |
| AU2009257692A1 (en) | 2009-12-17 |
| DK2303264T3 (en) | 2018-05-22 |
| EP2303264A1 (en) | 2011-04-06 |
| US8071636B2 (en) | 2011-12-06 |
| JP5571072B2 (ja) | 2014-08-13 |
| WO2009152052A8 (en) | 2010-11-11 |
| WO2009152052A1 (en) | 2009-12-17 |
| CA2744929C (en) | 2017-07-25 |
| JP2011522893A (ja) | 2011-08-04 |
| TR201802766T4 (tr) | 2018-03-21 |
| PL2303264T3 (pl) | 2018-08-31 |
| ES2665293T3 (es) | 2018-04-25 |
| EP2932968A1 (en) | 2015-10-21 |
| ES2672777T3 (es) | 2018-06-18 |
| HK1214132A1 (en) | 2016-07-22 |
| PL2932968T3 (pl) | 2018-06-29 |
| US20090306161A1 (en) | 2009-12-10 |
| CA2959793A1 (en) | 2009-12-17 |
| CA3133261A1 (en) | 2009-12-17 |
| CN102099032B (zh) | 2014-07-09 |
| EP2303264B1 (en) | 2018-04-04 |
| CN102099032A (zh) | 2011-06-15 |
| EP2377534A1 (en) | 2011-10-19 |
| SI2303264T1 (en) | 2018-08-31 |
| PT2303264T (pt) | 2018-05-14 |
| HUE039357T2 (hu) | 2018-12-28 |
| CA2744929A1 (en) | 2009-12-17 |
| US20120035235A1 (en) | 2012-02-09 |
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