AU2009220244B2 - Contrast agents for applications including perfusion imaging - Google Patents

Contrast agents for applications including perfusion imaging Download PDF

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Publication number
AU2009220244B2
AU2009220244B2 AU2009220244A AU2009220244A AU2009220244B2 AU 2009220244 B2 AU2009220244 B2 AU 2009220244B2 AU 2009220244 A AU2009220244 A AU 2009220244A AU 2009220244 A AU2009220244 A AU 2009220244A AU 2009220244 B2 AU2009220244 B2 AU 2009220244B2
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imaging
imaging moiety
alkyl
alkoxyalkyl
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AU2009220244A1 (en
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David S. Casebier
Mikhail Kagan
Joel Lazewatsky
Simon P. Robinson
Ming Yu
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Lantheus Medical Imaging Inc
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Lantheus Medical Imaging Inc
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K51/00—Preparations containing radioactive substances for use in therapy or testing in vivo
    • A61K51/02—Preparations containing radioactive substances for use in therapy or testing in vivo characterised by the carrier, i.e. characterised by the agent or material covalently linked or complexing the radioactive nucleus
    • A61K51/04—Organic compounds
    • A61K51/041—Heterocyclic compounds
    • A61K51/044—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins
    • A61K51/0459—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins having six-membered rings with two nitrogen atoms as the only ring hetero atoms, e.g. piperazine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents

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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Optics & Photonics (AREA)
  • Physics & Mathematics (AREA)
  • Epidemiology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Organic Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
AU2009220244A 2008-02-29 2009-02-27 Contrast agents for applications including perfusion imaging Active AU2009220244B2 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
AU2015200027A AU2015200027B2 (en) 2008-02-29 2015-01-06 Contrast agents for applications including perfusion imaging

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US6759308P 2008-02-29 2008-02-29
US61/067,593 2008-02-29
PCT/US2009/001247 WO2009110984A2 (en) 2008-02-29 2009-02-27 Contrast agents for applications including perfusion imaging

Related Child Applications (1)

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AU2015200027A Division AU2015200027B2 (en) 2008-02-29 2015-01-06 Contrast agents for applications including perfusion imaging

Publications (2)

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AU2009220244A1 AU2009220244A1 (en) 2009-09-11
AU2009220244B2 true AU2009220244B2 (en) 2014-10-09

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US (2) US9408927B2 (enExample)
EP (1) EP2257315B1 (enExample)
JP (3) JP5946992B2 (enExample)
KR (1) KR101616139B1 (enExample)
CN (1) CN102014969B (enExample)
AU (1) AU2009220244B2 (enExample)
CA (2) CA2716354C (enExample)
DK (1) DK2257315T3 (enExample)
ES (1) ES2767973T3 (enExample)
IL (1) IL207853A (enExample)
PT (1) PT2257315T (enExample)
WO (2) WO2009110984A2 (enExample)

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WO2009110984A2 (en) 2008-02-29 2009-09-11 Lantheus Medical Imaging, Inc. Contrast agents for applications including perfusion imaging
US20100241001A1 (en) * 2009-03-20 2010-09-23 Palmeri Mark L Ultrasound Methods, Systems and Computer Program Products for Imaging Fluids
ES2770364T3 (es) * 2009-04-15 2020-07-01 Lantheus Medical Imaging Inc Estabilización de composiciones radiofarmacéuticas utilizando ácido ascórbico
RU2631500C2 (ru) * 2010-02-08 2017-09-25 Лантеус Медикал Имаджинг, Инк. Способы и устройство для синтезирования радиофармацевтических препаратов и их промежуточных продуктов
US9550000B2 (en) 2011-09-09 2017-01-24 Lantheus Medical Imaging, Inc. Compositions, methods, and systems for the synthesis and use of imaging agents
WO2013058774A1 (en) * 2011-10-21 2013-04-25 Lantheus Medical Imaging, Inc. Compositions comprising ascorbic acid and an imaging agent and related methods
CN103254140B (zh) * 2012-02-17 2016-02-17 北京师范大学 新型18f标记取代喹唑啉类化合物及其制备方法和肿瘤pet显像应用
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GB201915206D0 (en) 2019-10-21 2019-12-04 Ge Healthcare Ltd Use of cyclodextrins as a radiostabilizer
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US20070036716A1 (en) * 2005-08-10 2007-02-15 Casebier David S Methods of making radiolabeled tracers and precursors thereof

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