AU2007279311A1 - Antagonists of endothelial differentiation gene subfamily 3 (Edg-3, S1P3) receptors for prevention and treatment of ocular disorders - Google Patents
Antagonists of endothelial differentiation gene subfamily 3 (Edg-3, S1P3) receptors for prevention and treatment of ocular disorders Download PDFInfo
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- AU2007279311A1 AU2007279311A1 AU2007279311A AU2007279311A AU2007279311A1 AU 2007279311 A1 AU2007279311 A1 AU 2007279311A1 AU 2007279311 A AU2007279311 A AU 2007279311A AU 2007279311 A AU2007279311 A AU 2007279311A AU 2007279311 A1 AU2007279311 A1 AU 2007279311A1
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Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/16—Amides, e.g. hydroxamic acids
- A61K31/17—Amides, e.g. hydroxamic acids having the group >N—C(O)—N< or >N—C(S)—N<, e.g. urea, thiourea, carmustine
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
- A61K31/426—1,3-Thiazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A61P27/06—Antiglaucoma agents or miotics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
Landscapes
- Health & Medical Sciences (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Epidemiology (AREA)
- General Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Ophthalmology & Optometry (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US83308006P | 2006-07-25 | 2006-07-25 | |
| US60/833,080 | 2006-07-25 | ||
| PCT/US2007/074351 WO2008014338A2 (en) | 2006-07-25 | 2007-07-25 | Antagonists of endothelial differentiation gene subfamily 3 (edg-3, s1p3) receptors for prevention and treatment of ocular disorders |
Publications (1)
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|---|---|
| AU2007279311A1 true AU2007279311A1 (en) | 2008-01-31 |
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
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| AU2007279311A Abandoned AU2007279311A1 (en) | 2006-07-25 | 2007-07-25 | Antagonists of endothelial differentiation gene subfamily 3 (Edg-3, S1P3) receptors for prevention and treatment of ocular disorders |
Country Status (11)
| Country | Link |
|---|---|
| US (2) | US20080025973A1 (https=) |
| EP (1) | EP2068856A2 (https=) |
| JP (1) | JP2009544734A (https=) |
| KR (1) | KR20090033886A (https=) |
| CN (1) | CN101505744A (https=) |
| AU (1) | AU2007279311A1 (https=) |
| BR (1) | BRPI0714593A2 (https=) |
| CA (1) | CA2657480A1 (https=) |
| MX (1) | MX2009000907A (https=) |
| WO (1) | WO2008014338A2 (https=) |
| ZA (1) | ZA200900316B (https=) |
Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
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| CN101014329B (zh) | 2004-07-16 | 2010-09-08 | 杏林制药株式会社 | 用于对器官或组织的移植的排异反应或骨髓移植的移植物抗宿主反应预防或治疗的药物组合物 |
| EP1806338B1 (en) | 2004-10-12 | 2016-01-20 | Kyorin Pharmaceutical Co., Ltd. | Process for producing 2-amino-2-[2-[4-(3-benzyloxy-phenylthio)-2-chlorophenyl[ethyl]-1,3-propanediol hydrochloride and hydrates thereof. and intermediates the production thereof |
| SI1932522T1 (sl) * | 2005-10-07 | 2012-08-31 | Kyorin Seiyaku Kk | Terapevtsko sredstvo za jetrno bolezen, ki vsebuje 2-amino-1,3- propandiolni derivat kot aktivno sestavino |
| TWI389683B (zh) * | 2006-02-06 | 2013-03-21 | Kyorin Seiyaku Kk | A therapeutic agent for an inflammatory bowel disease or an inflammatory bowel disease treatment using a 2-amino-1,3-propanediol derivative as an active ingredient |
| MX2009001457A (es) * | 2006-08-08 | 2009-02-19 | Kyorin Seiyaku Kk | Derivados de aminoalcohol e inmunosupresores que contienen lo mismo como ingrediente activo. |
| JP5188972B2 (ja) * | 2006-08-08 | 2013-04-24 | 杏林製薬株式会社 | アミノリン酸エステル誘導体及びそれらを有効成分とするｓ１ｐ受容体調節剤 |
| WO2009099174A1 (ja) | 2008-02-07 | 2009-08-13 | Kyorin Pharmaceutical Co., Ltd. | アミノアルコール誘導体を有効成分とする炎症性腸疾患の治療剤又は予防剤 |
| WO2009117335A2 (en) * | 2008-03-17 | 2009-09-24 | Allergan, Inc. | S1p3 receptor inhibitors for treating inflammation |
| US20120071448A1 (en) * | 2009-05-05 | 2012-03-22 | Allergan, Inc. | S1P3 Receptor Inhibitors for Treating Conditions of the Eye |
| US20110039900A1 (en) * | 2009-08-11 | 2011-02-17 | Allergan, Inc. | Isothiozoles for treating conditions of the eye |
| BR112012006965A2 (pt) * | 2009-09-30 | 2017-08-29 | Stiefel Res Australia Pty Ltd | Cosmético sob a forma de espuma |
| CN102146411B (zh) * | 2011-01-06 | 2013-01-02 | 中国人民解放军第三军医大学第三附属医院 | 新型双功能抗瘢痕和组织纤维化寡聚核苷酸药物 |
Family Cites Families (15)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU8107694A (en) * | 1993-11-17 | 1995-06-06 | Byk Nederland Bv | Use of substituted thiazolidine derivatives in the treatment of raised intraocular pressure |
| US5545626A (en) * | 1994-01-19 | 1996-08-13 | The Trustees Of Columbia University In The City Of New York | Method of treating glaucoma with oligonucleotides |
| US5750652A (en) * | 1994-01-21 | 1998-05-12 | Yale University | Deltex proteins |
| WO2001058468A1 (en) * | 2000-02-09 | 2001-08-16 | Connetics Corporation | Use of relaxin to treat diseases related to vasoconstriction |
| JP2001261575A (ja) * | 2000-03-13 | 2001-09-26 | General Hospital Corp | 血管収縮を調節する方法とその組成物 |
| JP2002332278A (ja) * | 2001-05-08 | 2002-11-22 | Human Science Shinko Zaidan | Ｅｄｇ受容体拮抗作用を有する複素環誘導体 |
| WO2003092584A2 (en) * | 2002-04-30 | 2003-11-13 | Alcon, Inc. | Agents which regulate, inhibit, or modulate the activity and/or expression of connective tissue growth factor (ctgf) as a unique means to both lower intraocular pressure and treat glaucomatous retinopathies/optic neuropathies |
| CA2533587A1 (en) * | 2002-07-30 | 2004-02-05 | University Of Virginia Patent Foundation | Compounds active in sphingosine 1-phosphate signaling |
| AU2003258433A1 (en) * | 2002-08-28 | 2004-03-19 | Merck Frosst Canada Ltd | Oxazolidin-2-one and thiazolidin-2-one derivatives for use as ep4 receptor agonists in the treatment of glaucoma |
| FR2845003A1 (fr) * | 2002-09-30 | 2004-04-02 | Merck Sante Sas | Utilisation de derives de thiazolidinedione comme inhibiteurs de l'aldose reductase |
| CN100418948C (zh) * | 2003-07-15 | 2008-09-17 | 麦克公司 | 羟基吡啶cgrp受体抗拮抗剂 |
| JP2005247691A (ja) * | 2004-03-01 | 2005-09-15 | Toa Eiyo Ltd | Ｓ１ｐ３受容体拮抗薬 |
| JP2008522977A (ja) * | 2004-12-06 | 2008-07-03 | ユニバーシティ オブ バージニア パテント ファンデーション | スフィンゴシン＝１−リン酸のアリールアミドアナログ |
| US8546452B2 (en) * | 2005-10-12 | 2013-10-01 | Toa Eiyo Ltd. | S1P3 receptor antagonist |
| CN101460458A (zh) * | 2006-02-15 | 2009-06-17 | 阿勒根公司 | 具有1－磷酸－鞘氨醇(s1p)受体拮抗剂生物活性的带芳基或者杂芳基基团的吲哚－3－羧酸的酰胺、酯、硫代酰胺和硫羟酸酯化合物 |
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2007
- 2007-07-25 EP EP07813352A patent/EP2068856A2/en not_active Withdrawn
- 2007-07-25 MX MX2009000907A patent/MX2009000907A/es not_active Application Discontinuation
- 2007-07-25 CA CA002657480A patent/CA2657480A1/en not_active Abandoned
- 2007-07-25 ZA ZA200900316A patent/ZA200900316B/xx unknown
- 2007-07-25 CN CNA2007800311386A patent/CN101505744A/zh active Pending
- 2007-07-25 BR BRPI0714593-4A patent/BRPI0714593A2/pt not_active IP Right Cessation
- 2007-07-25 AU AU2007279311A patent/AU2007279311A1/en not_active Abandoned
- 2007-07-25 JP JP2009521989A patent/JP2009544734A/ja active Pending
- 2007-07-25 WO PCT/US2007/074351 patent/WO2008014338A2/en not_active Ceased
- 2007-07-25 KR KR1020097002077A patent/KR20090033886A/ko not_active Ceased
- 2007-07-25 US US11/828,137 patent/US20080025973A1/en not_active Abandoned
-
2010
- 2010-03-29 US US12/749,331 patent/US20100183629A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| US20080025973A1 (en) | 2008-01-31 |
| WO2008014338A2 (en) | 2008-01-31 |
| CA2657480A1 (en) | 2008-01-31 |
| BRPI0714593A2 (pt) | 2013-05-07 |
| MX2009000907A (es) | 2009-02-04 |
| EP2068856A2 (en) | 2009-06-17 |
| ZA200900316B (en) | 2010-05-26 |
| JP2009544734A (ja) | 2009-12-17 |
| WO2008014338A3 (en) | 2008-12-24 |
| US20100183629A1 (en) | 2010-07-22 |
| CN101505744A (zh) | 2009-08-12 |
| KR20090033886A (ko) | 2009-04-06 |
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| Date | Code | Title | Description |
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| MK4 | Application lapsed section 142(2)(d) - no continuation fee paid for the application |