AU2006329007A1 - Nicotinic acid derivatives as modulators of metabotropic glutamate receptors - Google Patents

Nicotinic acid derivatives as modulators of metabotropic glutamate receptors Download PDF

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Publication number
AU2006329007A1
AU2006329007A1 AU2006329007A AU2006329007A AU2006329007A1 AU 2006329007 A1 AU2006329007 A1 AU 2006329007A1 AU 2006329007 A AU2006329007 A AU 2006329007A AU 2006329007 A AU2006329007 A AU 2006329007A AU 2006329007 A1 AU2006329007 A1 AU 2006329007A1
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Prior art keywords
pyridin
chloro
methyl
methanone
piperidin
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Abandoned
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AU2006329007A
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Inventor
Ralf Glatthar
David Orain
Carsten Spanka
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Novartis AG
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Novartis AG
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  • Chemical & Material Sciences (AREA)
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  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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  • Pharmacology & Pharmacy (AREA)
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  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Urology & Nephrology (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
  • Psychology (AREA)
  • Vascular Medicine (AREA)
  • Hospice & Palliative Care (AREA)
  • Obesity (AREA)
  • Child & Adolescent Psychology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Addiction (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Ophthalmology & Optometry (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Dermatology (AREA)
  • Nutrition Science (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyridine Compounds (AREA)
AU2006329007A 2005-12-20 2006-12-18 Nicotinic acid derivatives as modulators of metabotropic glutamate receptors Abandoned AU2006329007A1 (en)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
EP05027934.8 2005-12-20
EP05027934 2005-12-20
EP06120424.4 2006-09-11
EP06120424 2006-09-11
PCT/EP2006/012181 WO2007071358A1 (en) 2005-12-20 2006-12-18 Nicotinic acid derivatives as modulators of metabotropic glutamate receptors

Publications (1)

Publication Number Publication Date
AU2006329007A1 true AU2006329007A1 (en) 2007-06-28

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AU2006329007A Abandoned AU2006329007A1 (en) 2005-12-20 2006-12-18 Nicotinic acid derivatives as modulators of metabotropic glutamate receptors

Country Status (12)

Country Link
US (1) US20090005363A1 (enExample)
EP (1) EP1966144A1 (enExample)
JP (1) JP2009519986A (enExample)
KR (1) KR20080076962A (enExample)
AR (1) AR058554A1 (enExample)
AU (1) AU2006329007A1 (enExample)
BR (1) BRPI0620066A2 (enExample)
CA (1) CA2627630A1 (enExample)
PE (1) PE20071171A1 (enExample)
RU (1) RU2008129622A (enExample)
TW (1) TW200732323A (enExample)
WO (1) WO2007071358A1 (enExample)

Cited By (1)

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AU2007296964B2 (en) * 2006-09-11 2012-05-31 Novartis Ag Nicotinic acid derivatives as modulators of metabotropic glutanate receptors

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CA2695331A1 (en) * 2007-08-03 2009-02-12 F. Hoffmann-La Roche Ag Pyridinecarboxamide and benzamide derivatives as taar1 ligands
WO2009047303A2 (en) * 2007-10-12 2009-04-16 Novartis Ag Metabotropic glutamate receptor modulators for the treatment of pervasive developmental disorder
MX2010003913A (es) * 2007-10-12 2010-04-27 Novartis Ag Moduladores de los receptores de glutamato metabotropicos para el tratamiento de enfermedades de parkinson.
WO2010000763A2 (en) * 2008-06-30 2010-01-07 Novartis Ag Combination products
ES2551557T3 (es) * 2008-12-19 2015-11-19 Boehringer Ingelheim International Gmbh Pirimidin-4-carboxamidas cíclicas como antagonistas del receptor CCR2 para el tratamiento de inflamaciones, asma y EPOC
EP2942346B1 (en) 2009-02-17 2020-05-06 Syntrix Biosystems, Inc. Pyridinecarboxamides as cxcr2 modulators
EP2456438A2 (en) 2009-07-23 2012-05-30 Novartis AG Use of azabicycloalkyl derivatives or pyrrolidine-2-one derivatives
SG178867A1 (en) 2009-08-24 2012-04-27 Neuralstem Inc Synthesis of a neurostimulative piperazine
CA2774981A1 (en) * 2009-09-21 2011-03-24 Vanderbilt University O-benzyl nicotinamide analogs as mglur5 positive allosteric modulators
TWI558398B (zh) 2009-09-22 2016-11-21 諾華公司 菸鹼乙醯膽鹼受體α７活化劑之用途
WO2011048150A1 (en) 2009-10-20 2011-04-28 Novartis Ag Use of 1h-quinazoline-2,4-diones
PL2513093T3 (pl) 2009-12-17 2015-03-31 Centrexion Therapeutics Corp Nowi antagoniści receptora CCR2 i ich zastosowanie
KR20130122531A (ko) * 2010-05-24 2013-11-07 벤더르빌트 유니버시티 Ｍｇｌｕｒ５ 양성 알로스테릭 조절물로서 치환된 ６­메틸니코틴아미드
CA2800970A1 (en) 2010-06-24 2011-12-29 Novartis Ag Use of 1h-quinazoline-2,4-diones
AU2011293612B2 (en) 2010-08-23 2015-11-26 Syntrix Biosystems Inc. Aminopyridine- and aminopyrimidinecarboxamides as CXCR2 modulators
AR084515A1 (es) * 2010-12-22 2013-05-22 Merz Pharma Gmbh & Co Kgaa Derivados heterociclicos nitrogenados, composiciones farmaceuticas que los contienen y uso de los mismos en el tratamiento de enfermedades asociadas al sistema nervioso central tales como parkinson y alzheimer, entre otras
WO2012085166A1 (en) * 2010-12-22 2012-06-28 Merz Pharma Gmbh & Co. Kgaa Metabotropic glutamate receptor modulators
US20140171448A1 (en) 2011-01-27 2014-06-19 Novartis Ag Use of nicotinic acetylcholine receptor alpha 7 activators
CA2846503A1 (en) 2011-09-07 2013-03-14 Novartis Ag Use of 1h-quinazoline-2,4-diones for use in the prevention or treatment of photosensitive epilepsy
MX358696B (es) * 2011-12-22 2018-08-31 Connexios Life Sciences Pvt Ltd Derivados de aza adamantano y lo usos de los mismos.
MX379289B (es) 2013-01-15 2025-03-10 Novartis Ag Uso de agonistas del receptor nicotinico de acetilcolina alfa 7.
JP6137336B2 (ja) 2013-01-15 2017-05-31 ノバルティス アーゲー ナルコレプシーの処置のためのアルファ７ニコチン性受容体アゴニストの使用
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US20090005363A1 (en) 2009-01-01
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CA2627630A1 (en) 2007-06-28
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BRPI0620066A2 (pt) 2011-11-01
AR058554A1 (es) 2008-02-13

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