AU2006278592A1 - Sphingosine kinase inhibitors and methods of their use - Google Patents
Sphingosine kinase inhibitors and methods of their use Download PDFInfo
- Publication number
- AU2006278592A1 AU2006278592A1 AU2006278592A AU2006278592A AU2006278592A1 AU 2006278592 A1 AU2006278592 A1 AU 2006278592A1 AU 2006278592 A AU2006278592 A AU 2006278592A AU 2006278592 A AU2006278592 A AU 2006278592A AU 2006278592 A1 AU2006278592 A1 AU 2006278592A1
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- Prior art keywords
- phenyl
- chloro
- alkyl
- thiazol
- thiazole
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- C07C233/64—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings
- C07C233/67—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by singly-bound oxygen atoms
- C07C233/75—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by singly-bound oxygen atoms with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by a carbon atom of a six-membered aromatic ring
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- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Immunology (AREA)
- Diabetes (AREA)
- Pulmonology (AREA)
- Physical Education & Sports Medicine (AREA)
- Rheumatology (AREA)
- Ophthalmology & Optometry (AREA)
- Hematology (AREA)
- Urology & Nephrology (AREA)
- Cardiology (AREA)
- Dermatology (AREA)
- Endocrinology (AREA)
- Heart & Thoracic Surgery (AREA)
- Pain & Pain Management (AREA)
- Vascular Medicine (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Obesity (AREA)
- Emergency Medicine (AREA)
- Transplantation (AREA)
- Neurosurgery (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US70560805P | 2005-08-04 | 2005-08-04 | |
| US60/705,608 | 2005-08-04 | ||
| PCT/US2006/030327 WO2007019251A2 (en) | 2005-08-04 | 2006-08-03 | Sphingosine kinase inhibitors and methods of their use |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AU2006278592A1 true AU2006278592A1 (en) | 2007-02-15 |
Family
ID=37433959
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AU2006278592A Abandoned AU2006278592A1 (en) | 2005-08-04 | 2006-08-03 | Sphingosine kinase inhibitors and methods of their use |
Country Status (7)
| Country | Link |
|---|---|
| US (2) | US20070032531A1 (enExample) |
| EP (1) | EP1928848A2 (enExample) |
| JP (1) | JP2009503107A (enExample) |
| AU (1) | AU2006278592A1 (enExample) |
| CA (1) | CA2617788A1 (enExample) |
| IL (1) | IL188932A0 (enExample) |
| WO (1) | WO2007019251A2 (enExample) |
Families Citing this family (40)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US8324237B2 (en) * | 2005-05-20 | 2012-12-04 | Smith Charles D | Methods for the treatment and prevention of inflammatory diseases |
| US8709015B2 (en) * | 2008-03-10 | 2014-04-29 | DePuy Synthes Products, LLC | Bilateral vertebral body derotation system |
| EP2107054A1 (en) * | 2008-04-01 | 2009-10-07 | Università Degli Studi Di Milano - Bicocca | Antiproliferative compounds and therapeutic uses thereof |
| DE102008029734A1 (de) | 2008-06-23 | 2009-12-24 | Merck Patent Gmbh | Thiazolyl-piperidinderivate |
| EP2166094A1 (en) | 2008-09-23 | 2010-03-24 | Ecole Normale Superieure De Lyon | Methods for prolonging the health benefits triggered by a dietary restriction using a sphingosine kinase inhibitor |
| PE20120834A1 (es) | 2009-03-23 | 2012-07-25 | Glenmark Pharmaceuticals Sa | Derivados de furopirimidindiona como moduladores de trpa1 |
| GB0905525D0 (en) * | 2009-03-31 | 2009-05-13 | Univ Leiden | Compounds and uses |
| AU2010333338A1 (en) * | 2009-12-14 | 2012-08-02 | Merck Patent Gmbh | Sphingosine kinase inhibitors |
| NZ601967A (en) | 2010-03-12 | 2015-03-27 | Omeros Corp | Pde10 inhibitors and related compositions and methods |
| CN103038231B (zh) * | 2010-03-17 | 2016-04-20 | 泰纬生命科技股份有限公司 | Hec1活性调节剂及其方法 |
| KR101847669B1 (ko) * | 2010-08-16 | 2018-05-24 | 알러간, 인코포레이티드 | 알파-2b 아드레날린성 수용체 효현제로 조절 t 세포를 활성화시키는 방법 |
| AU2012221800B2 (en) | 2011-02-23 | 2016-10-27 | Lupin Limited | Heteroaryl derivatives as alpha7 nAChR modulators |
| US9687477B2 (en) * | 2011-06-01 | 2017-06-27 | The Curators Of The University Of Missouri | Modulation of sphingosine 1-phosphate metabolizing enzymes for the treatment of negative-strand RNA virus infections |
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| EP3223807B1 (en) * | 2014-11-24 | 2021-09-15 | The Board of Trustees of the University of Illinois | Method of preventing or treating a pulmonary disease or condition |
| CA2980801A1 (en) | 2015-04-24 | 2016-10-27 | Omeros Corporation | Pde10 inhibitors and related compositions and methods |
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| KR102732033B1 (ko) | 2019-07-26 | 2024-11-20 | 아주대학교산학협력단 | Tlr7 및 tlr9의 신호전달 경로를 억제하는 신규한 소분자 화합물 및 그 용도 |
| WO2021066608A1 (ko) * | 2019-10-02 | 2021-04-08 | 주식회사 클로소사이언스 | 항노화 유전자 klotho의 발현을 유도하는 화합물 및 이의 용도 |
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| US8324237B2 (en) * | 2005-05-20 | 2012-12-04 | Smith Charles D | Methods for the treatment and prevention of inflammatory diseases |
| US20060270631A1 (en) * | 2005-05-26 | 2006-11-30 | Smith Charles D | Methods for the treatment and prevention of angiogenic diseases |
-
2006
- 2006-08-03 CA CA002617788A patent/CA2617788A1/en not_active Abandoned
- 2006-08-03 WO PCT/US2006/030327 patent/WO2007019251A2/en not_active Ceased
- 2006-08-03 EP EP06800721A patent/EP1928848A2/en not_active Withdrawn
- 2006-08-03 AU AU2006278592A patent/AU2006278592A1/en not_active Abandoned
- 2006-08-03 JP JP2008525195A patent/JP2009503107A/ja active Pending
- 2006-08-03 US US11/462,153 patent/US20070032531A1/en not_active Abandoned
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2008
- 2008-01-22 IL IL188932A patent/IL188932A0/en unknown
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2009
- 2009-11-30 US US12/627,812 patent/US20100137315A1/en not_active Abandoned
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|---|---|
| US20100137315A1 (en) | 2010-06-03 |
| WO2007019251A2 (en) | 2007-02-15 |
| WO2007019251A9 (en) | 2007-04-19 |
| IL188932A0 (en) | 2008-04-13 |
| EP1928848A2 (en) | 2008-06-11 |
| US20070032531A1 (en) | 2007-02-08 |
| WO2007019251A3 (en) | 2007-05-31 |
| JP2009503107A (ja) | 2009-01-29 |
| CA2617788A1 (en) | 2007-02-15 |
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