IL188932A0 - Sphingosine kinase inhibitors and methods of their use - Google Patents

Sphingosine kinase inhibitors and methods of their use

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Publication number
IL188932A0
IL188932A0 IL188932A IL18893208A IL188932A0 IL 188932 A0 IL188932 A0 IL 188932A0 IL 188932 A IL188932 A IL 188932A IL 18893208 A IL18893208 A IL 18893208A IL 188932 A0 IL188932 A0 IL 188932A0
Authority
IL
Israel
Prior art keywords
methods
kinase inhibitors
sphingosine kinase
sphingosine
inhibitors
Prior art date
Application number
IL188932A
Other languages
English (en)
Original Assignee
Apogee Biotechnology Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Apogee Biotechnology Corp filed Critical Apogee Biotechnology Corp
Publication of IL188932A0 publication Critical patent/IL188932A0/en

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    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
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    • C07C233/64—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings
    • C07C233/67—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by singly-bound oxygen atoms
    • C07C233/75—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by singly-bound oxygen atoms with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by a carbon atom of a six-membered aromatic ring
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  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Immunology (AREA)
  • Diabetes (AREA)
  • Pulmonology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Rheumatology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Hematology (AREA)
  • Urology & Nephrology (AREA)
  • Cardiology (AREA)
  • Dermatology (AREA)
  • Endocrinology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pain & Pain Management (AREA)
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  • Orthopedic Medicine & Surgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Obesity (AREA)
  • Emergency Medicine (AREA)
  • Transplantation (AREA)
  • Neurosurgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
IL188932A 2005-08-04 2008-01-22 Sphingosine kinase inhibitors and methods of their use IL188932A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US70560805P 2005-08-04 2005-08-04
PCT/US2006/030327 WO2007019251A2 (en) 2005-08-04 2006-08-03 Sphingosine kinase inhibitors and methods of their use

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IL188932A0 true IL188932A0 (en) 2008-04-13

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US (2) US20070032531A1 (enExample)
EP (1) EP1928848A2 (enExample)
JP (1) JP2009503107A (enExample)
AU (1) AU2006278592A1 (enExample)
CA (1) CA2617788A1 (enExample)
IL (1) IL188932A0 (enExample)
WO (1) WO2007019251A2 (enExample)

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US8324237B2 (en) * 2005-05-20 2012-12-04 Smith Charles D Methods for the treatment and prevention of inflammatory diseases
US8709015B2 (en) * 2008-03-10 2014-04-29 DePuy Synthes Products, LLC Bilateral vertebral body derotation system
EP2107054A1 (en) * 2008-04-01 2009-10-07 Università Degli Studi Di Milano - Bicocca Antiproliferative compounds and therapeutic uses thereof
DE102008029734A1 (de) 2008-06-23 2009-12-24 Merck Patent Gmbh Thiazolyl-piperidinderivate
EP2166094A1 (en) 2008-09-23 2010-03-24 Ecole Normale Superieure De Lyon Methods for prolonging the health benefits triggered by a dietary restriction using a sphingosine kinase inhibitor
PE20120834A1 (es) 2009-03-23 2012-07-25 Glenmark Pharmaceuticals Sa Derivados de furopirimidindiona como moduladores de trpa1
GB0905525D0 (en) * 2009-03-31 2009-05-13 Univ Leiden Compounds and uses
AU2010333338A1 (en) * 2009-12-14 2012-08-02 Merck Patent Gmbh Sphingosine kinase inhibitors
NZ601967A (en) 2010-03-12 2015-03-27 Omeros Corp Pde10 inhibitors and related compositions and methods
CN103038231B (zh) * 2010-03-17 2016-04-20 泰纬生命科技股份有限公司 Hec1活性调节剂及其方法
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