AU2006245416B2 - Anhydrous crystalline forms of N-[1-(2-ethoxyethyl)-5-(N-ethyl-N-methylamino)-7-(4-methylpyridin-2-yl-amino)-1H-pyrazolo[4,3-d]pyrimidine-3-carbonyl]methanesulfonamide - Google Patents

Anhydrous crystalline forms of N-[1-(2-ethoxyethyl)-5-(N-ethyl-N-methylamino)-7-(4-methylpyridin-2-yl-amino)-1H-pyrazolo[4,3-d]pyrimidine-3-carbonyl]methanesulfonamide Download PDF

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AU2006245416B2
AU2006245416B2 AU2006245416A AU2006245416A AU2006245416B2 AU 2006245416 B2 AU2006245416 B2 AU 2006245416B2 AU 2006245416 A AU2006245416 A AU 2006245416A AU 2006245416 A AU2006245416 A AU 2006245416A AU 2006245416 B2 AU2006245416 B2 AU 2006245416B2
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ethoxyethyl
pyrazolo
ethyl
methylpyridin
methanesulfonamide
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AU2006245416A1 (en
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David Andrew Entwistle
Peter Vallance Marshall
Stefan Colin John Taylor
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Pfizer Inc
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Pfizer Inc
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
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AU2006245416A 2005-05-12 2006-05-03 Anhydrous crystalline forms of N-[1-(2-ethoxyethyl)-5-(N-ethyl-N-methylamino)-7-(4-methylpyridin-2-yl-amino)-1H-pyrazolo[4,3-d]pyrimidine-3-carbonyl]methanesulfonamide Ceased AU2006245416B2 (en)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US68044505P 2005-05-12 2005-05-12
US60/680,445 2005-05-12
US68171105P 2005-05-17 2005-05-17
US60/681,711 2005-05-17
PCT/IB2006/001233 WO2006120552A2 (en) 2005-05-12 2006-05-03 ANHYDROUS CRYSTALLINE FORMS OF N-[1-(2-ETHOXYETHYL)-5-(N-ETHYL-N-METHYLAMINO)-7-(4-METHYLPYRIDIN-2-yl-AMINO)-1H-PYRAZOLO[4,3-d]PYRIMIDINE-3-CARBONYL]METHANESULFONAMIDE

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AU2006245416A1 AU2006245416A1 (en) 2006-11-16
AU2006245416B2 true AU2006245416B2 (en) 2012-02-23

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AU2006245416A Ceased AU2006245416B2 (en) 2005-05-12 2006-05-03 Anhydrous crystalline forms of N-[1-(2-ethoxyethyl)-5-(N-ethyl-N-methylamino)-7-(4-methylpyridin-2-yl-amino)-1H-pyrazolo[4,3-d]pyrimidine-3-carbonyl]methanesulfonamide

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US (3) US8227475B2 (https=)
EP (1) EP1881985B1 (https=)
JP (2) JP4271695B2 (https=)
KR (1) KR100939890B1 (https=)
AT (1) ATE493413T1 (https=)
AU (1) AU2006245416B2 (https=)
BR (1) BRPI0609225A2 (https=)
CA (1) CA2608018C (https=)
CR (1) CR9505A (https=)
CY (1) CY1111171T1 (https=)
DE (1) DE602006019231D1 (https=)
DK (1) DK1881985T3 (https=)
EA (1) EA012577B1 (https=)
IL (1) IL186693A (https=)
MA (1) MA29447B1 (https=)
MX (1) MX2007013215A (https=)
NO (1) NO20075258L (https=)
NZ (1) NZ564187A (https=)
PL (1) PL1881985T3 (https=)
PT (1) PT1881985E (https=)
TN (1) TNSN07414A1 (https=)
TW (1) TWI380986B (https=)
WO (1) WO2006120552A2 (https=)

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