AU2004270741B2 - Gapped oligomeric compounds having linked bicyclic sugar moieties at the termini - Google Patents

Gapped oligomeric compounds having linked bicyclic sugar moieties at the termini Download PDF

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Publication number
AU2004270741B2
AU2004270741B2 AU2004270741A AU2004270741A AU2004270741B2 AU 2004270741 B2 AU2004270741 B2 AU 2004270741B2 AU 2004270741 A AU2004270741 A AU 2004270741A AU 2004270741 A AU2004270741 A AU 2004270741A AU 2004270741 B2 AU2004270741 B2 AU 2004270741B2
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Prior art keywords
oligomeric compound
independently
nucleoside
nucleosides
bridge
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AU2004270741A
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AU2004270741A1 (en
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Michael T. Migawa
Eric E. Swayze
Tradeusz Krzysztof Wyrzykiewicz
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Ionis Pharmaceuticals Inc
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Isis Pharmaceuticals Inc
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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H21/00Compounds containing two or more mononucleotide units having separate phosphate or polyphosphate groups linked by saccharide radicals of nucleoside groups, e.g. nucleic acids
    • C07H21/04Compounds containing two or more mononucleotide units having separate phosphate or polyphosphate groups linked by saccharide radicals of nucleoside groups, e.g. nucleic acids with deoxyribosyl as saccharide radical
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

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  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Genetics & Genomics (AREA)
  • Biotechnology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
AU2004270741A 2003-09-09 2004-09-09 Gapped oligomeric compounds having linked bicyclic sugar moieties at the termini Ceased AU2004270741B2 (en)

Applications Claiming Priority (9)

Application Number Priority Date Filing Date Title
US50171903P 2003-09-09 2003-09-09
US60/501,719 2003-09-09
US56803904P 2004-05-03 2004-05-03
US60/568,039 2004-05-03
US56848904P 2004-05-06 2004-05-06
US60/568,489 2004-05-06
US10/872,106 US20050053981A1 (en) 2003-09-09 2004-06-18 Gapped oligomeric compounds having linked bicyclic sugar moieties at the termini
US10/872,106 2004-06-18
PCT/US2004/029650 WO2005023825A2 (en) 2003-09-09 2004-09-09 Gapped oligomeric compounds having linked bicyclic sugar moieties at the termini

Publications (2)

Publication Number Publication Date
AU2004270741A1 AU2004270741A1 (en) 2005-03-17
AU2004270741B2 true AU2004270741B2 (en) 2011-02-24

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AU2004270741A Ceased AU2004270741B2 (en) 2003-09-09 2004-09-09 Gapped oligomeric compounds having linked bicyclic sugar moieties at the termini

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US (2) US20050053981A1 (enExample)
EP (1) EP1670810A4 (enExample)
JP (1) JP2007505138A (enExample)
AU (1) AU2004270741B2 (enExample)
CA (1) CA2538174A1 (enExample)
WO (1) WO2005023825A2 (enExample)

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