AU2004220410A1 - Process for the preparation of a cyano-isobenzofuran - Google Patents

Process for the preparation of a cyano-isobenzofuran Download PDF

Info

Publication number
AU2004220410A1
AU2004220410A1 AU2004220410A AU2004220410A AU2004220410A1 AU 2004220410 A1 AU2004220410 A1 AU 2004220410A1 AU 2004220410 A AU2004220410 A AU 2004220410A AU 2004220410 A AU2004220410 A AU 2004220410A AU 2004220410 A1 AU2004220410 A1 AU 2004220410A1
Authority
AU
Australia
Prior art keywords
fluorophenyl
dihydro
isobenzofurancarbonitrile
hydroxymethyl
bis
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU2004220410A
Other languages
English (en)
Inventor
Giovanni Cotticelli
Leone Dall'asta
Gianluca Di Lernia
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Adorkem Technology SpA
Original Assignee
Adorkem Technology SpA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Adorkem Technology SpA filed Critical Adorkem Technology SpA
Publication of AU2004220410A1 publication Critical patent/AU2004220410A1/en
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/87—Benzo [c] furans; Hydrogenated benzo [c] furans
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Furan Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
AU2004220410A 2003-03-13 2004-03-09 Process for the preparation of a cyano-isobenzofuran Abandoned AU2004220410A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
ITMI2003A000479 2003-03-13
IT000479A ITMI20030479A1 (it) 2003-03-13 2003-03-13 Procedimento per la preparazione di un ciano-isobenzofurano.
PCT/EP2004/002522 WO2004080988A1 (en) 2003-03-13 2004-03-09 Process for the preparation of a cyano-isobenzofuran

Publications (1)

Publication Number Publication Date
AU2004220410A1 true AU2004220410A1 (en) 2004-09-23

Family

ID=32983208

Family Applications (1)

Application Number Title Priority Date Filing Date
AU2004220410A Abandoned AU2004220410A1 (en) 2003-03-13 2004-03-09 Process for the preparation of a cyano-isobenzofuran

Country Status (13)

Country Link
US (1) US7411077B2 (cg-RX-API-DMAC10.html)
EP (1) EP1601662A1 (cg-RX-API-DMAC10.html)
JP (1) JP2006520351A (cg-RX-API-DMAC10.html)
KR (1) KR20050108376A (cg-RX-API-DMAC10.html)
CN (1) CN1761658A (cg-RX-API-DMAC10.html)
AU (1) AU2004220410A1 (cg-RX-API-DMAC10.html)
BR (1) BRPI0408732A (cg-RX-API-DMAC10.html)
CA (1) CA2514458A1 (cg-RX-API-DMAC10.html)
HR (1) HRP20050893A2 (cg-RX-API-DMAC10.html)
IT (1) ITMI20030479A1 (cg-RX-API-DMAC10.html)
MX (1) MXPA05008411A (cg-RX-API-DMAC10.html)
WO (1) WO2004080988A1 (cg-RX-API-DMAC10.html)
ZA (1) ZA200505592B (cg-RX-API-DMAC10.html)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8969379B2 (en) 2004-09-17 2015-03-03 Eisai R&D Management Co., Ltd. Pharmaceutical compositions of 4-(3-chloro-4-(cyclopropylaminocarbonyl)aminophenoxy)-7=methoxy-6-quinolinecarboxide
WO2008059514A2 (en) * 2006-07-31 2008-05-22 Cadila Healthcare Limited Process for preparing escitalopram
EP3808181A1 (en) 2014-12-30 2021-04-21 Dow AgroSciences LLC Use of picolinamide compounds as fungicides
PL3481201T3 (pl) 2016-07-07 2021-03-22 Corteva Agriscience Llc Sposoby wytwarzania 4-alkoksy-3-(acylo lub alkilo)oksypikolinamidów
CN108929245A (zh) * 2017-05-25 2018-12-04 万全万特制药江苏有限公司 艾司西酞普兰工艺杂质的制备方法
CN108947869A (zh) * 2017-05-25 2018-12-07 万全万特制药江苏有限公司 一种艾司西酞普兰工艺杂质的制备方法
CN120097946B (zh) * 2025-02-28 2026-06-19 浙江工业大学 一种应用脱水膜强化5-氰二醇盐酸盐醚化制西酞普兰溴酸盐的方法

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1526331A (en) * 1976-01-14 1978-09-27 Kefalas As Phthalanes
JP3526581B2 (ja) * 1997-07-08 2004-05-17 ハー・ルンドベック・アクティーゼルスカブ シタロプラムの製造方法
UA62985C2 (en) * 1997-11-10 2004-01-15 Lunnbeck As H A method for the preparation of citalopram
CN1286687A (zh) * 1997-11-11 2001-03-07 H·隆德贝克有限公司 制备西酞普兰的方法
US6310222B1 (en) * 1999-11-01 2001-10-30 Sumika Fine Chemicals Co., Ltd. Production method of 5-phthalancarbonitrile compound, intermediate therefor and production method of the intermediate
JP3641420B2 (ja) * 1999-11-01 2005-04-20 住友化学株式会社 ５−フタランカルボニトリル化合物の製造方法、その中間体およびその製造方法
JP3735026B2 (ja) * 2000-02-17 2006-01-11 住友化学株式会社 シタロプラムの製造方法、およびその中間体とその製造方法
US6433196B1 (en) * 2000-02-17 2002-08-13 Sumika Fine Chemicals Co., Ltd. Production method of citalopram, intermediate therefor and production method of the intermediate

Also Published As

Publication number Publication date
HRP20050893A2 (en) 2005-12-31
BRPI0408732A (pt) 2006-03-07
JP2006520351A (ja) 2006-09-07
MXPA05008411A (es) 2005-10-05
KR20050108376A (ko) 2005-11-16
US20060183925A1 (en) 2006-08-17
ZA200505592B (en) 2006-09-27
EP1601662A1 (en) 2005-12-07
CA2514458A1 (en) 2004-09-23
CN1761658A (zh) 2006-04-19
US7411077B2 (en) 2008-08-12
WO2004080988A1 (en) 2004-09-23
ITMI20030479A1 (it) 2004-09-14

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Legal Events

Date Code Title Description
MK4 Application lapsed section 142(2)(d) - no continuation fee paid for the application