AU2002316421B2 - N-heterocyclic inhibitors of TNF-ALPHA expression - Google Patents

N-heterocyclic inhibitors of TNF-ALPHA expression Download PDF

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Publication number
AU2002316421B2
AU2002316421B2 AU2002316421A AU2002316421A AU2002316421B2 AU 2002316421 B2 AU2002316421 B2 AU 2002316421B2 AU 2002316421 A AU2002316421 A AU 2002316421A AU 2002316421 A AU2002316421 A AU 2002316421A AU 2002316421 B2 AU2002316421 B2 AU 2002316421B2
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Prior art keywords
hydrogen
alkyl
substituted
compound
methyl
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AU2002316421A1 (en
Inventor
Gulzar Ahmed
David J. Diller
Ian Henderson
Katerina Leftheris
Axel Metzger
James Wen
Stephen T. Wrobleski
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Bristol Myers Squibb Co
Pharmacopeia LLC
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Bristol Myers Squibb Co
Pharmacopeia Inc
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AU2002316421A 2001-06-26 2002-06-26 N-heterocyclic inhibitors of TNF-ALPHA expression Ceased AU2002316421B2 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US30102001P 2001-06-26 2001-06-26
US60/301,020 2001-06-26
PCT/US2002/020341 WO2003002544A1 (en) 2001-06-26 2002-06-26 N-heterocyclic inhibitors of tnf-alpha expression

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AU2002316421A1 AU2002316421A1 (en) 2003-05-15
AU2002316421B2 true AU2002316421B2 (en) 2008-05-15

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EP (1) EP1406875B1 (enExample)
JP (1) JP4510442B2 (enExample)
AU (1) AU2002316421B2 (enExample)
CA (1) CA2451128A1 (enExample)
HU (1) HUP0401711A3 (enExample)
WO (1) WO2003002544A1 (enExample)

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AU2002316421B2 (en) * 2001-06-26 2008-05-15 Bristol-Myers Squibb Company N-heterocyclic inhibitors of TNF-ALPHA expression
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TWI329105B (en) 2002-02-01 2010-08-21 Rigel Pharmaceuticals Inc 2,4-pyrimidinediamine compounds and their uses
PL219736B1 (pl) 2002-04-23 2015-07-31 Bristol Myers Squibb Co Pochodna pirolotriazynoaniliny, kompozycja farmaceutyczna i jej zastosowanie
ATE418546T1 (de) 2002-04-23 2009-01-15 Bristol Myers Squibb Co Als kinase inhibitoren geeignete arylketonpyrrolotriazin-verbindungen
IL166241A0 (en) 2002-07-29 2006-01-15 Rigel Pharmaceuticals Inc Method of treating or preventing autoimmune diseases with 2,4-pyrimidinedinediamine compounds
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