AU2002217287A1 - Benzo(f) isoindol derivatives and their use as ep4 receptor ligands - Google Patents

Benzo(f) isoindol derivatives and their use as ep4 receptor ligands

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Publication number
AU2002217287A1
AU2002217287A1 AU2002217287A AU1728702A AU2002217287A1 AU 2002217287 A1 AU2002217287 A1 AU 2002217287A1 AU 2002217287 A AU2002217287 A AU 2002217287A AU 1728702 A AU1728702 A AU 1728702A AU 2002217287 A1 AU2002217287 A1 AU 2002217287A1
Authority
AU
Australia
Prior art keywords
benzo
receptor ligands
isoindol
derivatives
isoindol derivatives
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU2002217287A
Other languages
English (en)
Inventor
Stephen Vernon Frye
Gerard Martin Paul Giblin
Susan Roomans
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Glaxo Group Ltd
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Publication of AU2002217287A1 publication Critical patent/AU2002217287A1/en
Abandoned legal-status Critical Current

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    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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AU2002217287A 2000-12-21 2001-12-20 Benzo(f) isoindol derivatives and their use as ep4 receptor ligands Abandoned AU2002217287A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB0031295 2000-12-21
GBGB0031295.9A GB0031295D0 (en) 2000-12-21 2000-12-21 Naphthalene derivatives
PCT/GB2001/005706 WO2002050033A1 (en) 2000-12-21 2001-12-20 Benzo(f) isoindol derivatives and their use as ep4 receptor ligands

Publications (1)

Publication Number Publication Date
AU2002217287A1 true AU2002217287A1 (en) 2002-07-01

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AU2002217287A Abandoned AU2002217287A1 (en) 2000-12-21 2001-12-20 Benzo(f) isoindol derivatives and their use as ep4 receptor ligands

Country Status (6)

Country Link
US (2) US7173047B2 (enExample)
EP (1) EP1343759A1 (enExample)
JP (1) JP4398150B2 (enExample)
AU (1) AU2002217287A1 (enExample)
GB (1) GB0031295D0 (enExample)
WO (1) WO2002050033A1 (enExample)

Families Citing this family (26)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HN2001000224A (es) 2000-10-19 2002-06-13 Pfizer Compuestos de imidazol condensado con arilo o heteroarilo como agentes anti - inflamatorios y analgesicos.
GB0103269D0 (en) * 2001-02-09 2001-03-28 Glaxo Group Ltd Napthalene derivatives
BR0309200A (pt) 2002-04-12 2005-02-22 Pfizer Uso de ligandos receptores ep4 no tratamento de doenças envolvidas com a il-6
WO2004073589A2 (en) * 2003-02-24 2004-09-02 Bayer Healthcare Ag Diagnostics and therapeutics for diseases associated with g-protein coupled receptor prostaglandin e2 ep4 (prostaglandin e2 ep4)
JP2007533723A (ja) * 2004-04-20 2007-11-22 ファイザー・プロダクツ・インク α２δリガンドを含む組合せ
ATE533766T1 (de) 2005-05-19 2011-12-15 Merck Canada Inc Chinolinderivate als ep4-antagonisten
UY30121A1 (es) 2006-02-03 2007-08-31 Glaxo Group Ltd Nuevos compuestos
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