AU2001294953A1 - Triterpenes having fungicidal activity against yeast - Google Patents

Triterpenes having fungicidal activity against yeast

Info

Publication number
AU2001294953A1
AU2001294953A1 AU2001294953A AU9495301A AU2001294953A1 AU 2001294953 A1 AU2001294953 A1 AU 2001294953A1 AU 2001294953 A AU2001294953 A AU 2001294953A AU 9495301 A AU9495301 A AU 9495301A AU 2001294953 A1 AU2001294953 A1 AU 2001294953A1
Authority
AU
Australia
Prior art keywords
betulin
alkyl
allobetulin
hydrogen
hydroxy
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU2001294953A
Other languages
English (en)
Inventor
Robert M. Carlson
Raj Karim
Pavel A. Krasutsky
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
University of Minnesota
Original Assignee
University of Minnesota
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by University of Minnesota filed Critical University of Minnesota
Publication of AU2001294953A1 publication Critical patent/AU2001294953A1/en
Abandoned legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J63/00Steroids in which the cyclopenta(a)hydrophenanthrene skeleton has been modified by expansion of only one ring by one or two atoms
    • C07J63/008Expansion of ring D by one atom, e.g. D homo steroids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10Antimycotics

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Oncology (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Steroid Compounds (AREA)
AU2001294953A 2000-09-29 2001-10-01 Triterpenes having fungicidal activity against yeast Abandoned AU2001294953A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US23775600P 2000-09-29 2000-09-29
US60237756 2000-09-29
PCT/US2001/030761 WO2002026761A1 (en) 2000-09-29 2001-10-01 Triterpenes having fungicidal activity against yeast

Publications (1)

Publication Number Publication Date
AU2001294953A1 true AU2001294953A1 (en) 2002-04-08

Family

ID=22895030

Family Applications (1)

Application Number Title Priority Date Filing Date
AU2001294953A Abandoned AU2001294953A1 (en) 2000-09-29 2001-10-01 Triterpenes having fungicidal activity against yeast

Country Status (6)

Country Link
US (1) US6642217B2 (ja)
EP (1) EP1322661A1 (ja)
JP (1) JP2004509972A (ja)
AU (1) AU2001294953A1 (ja)
CA (1) CA2424013A1 (ja)
WO (1) WO2002026761A1 (ja)

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US9556222B2 (en) 2012-06-15 2017-01-31 Reata Pharmaceuticals, Inc. A-ring epoxidized triterpenoid-based anti-inflammation modulators and methods of use thereof
ITMI20121109A1 (it) * 2012-06-25 2013-12-26 Rode Pharma S R L Composizione comprendente acido gascardico o un suo derivato e relativo uso come coadiuvante per antibiotici
US9278912B2 (en) 2012-09-10 2016-03-08 Reata Pharmaceuticals, Inc. C13-hydroxy derivatives of oleanolic acid and methods of use thereof
MY180903A (en) 2012-09-10 2020-12-11 Reata Pharmaceuticals Inc C17-alkanediyl and alkenediyl derivatives of oleanolic acid and methods of use thereof
US9512094B2 (en) 2012-09-10 2016-12-06 Reata Pharmaceuticals, Inc. C17-heteroaryl derivatives of oleanolic acid and methods of use thereof
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CN104387440A (zh) * 2014-11-07 2015-03-04 上海应用技术学院 一种白桦脂醇氨基酸酯化合物及其制备方法和用途
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RU2638160C1 (ru) * 2017-03-20 2017-12-12 Федеральное государственное бюджетное научное учреждение "Федеральный исследовательский центр "Красноярский научный центр Сибирского отделения Российской академии наук" (ФИЦ КНЦ СО РАН, КНЦ СО РАН) Способ получения дисукцината бетулинола
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CN107019660B (zh) 2017-04-27 2018-05-11 养生堂(上海)化妆品研发有限公司 保湿化妆品组合物
CN107049865B (zh) * 2017-04-27 2018-03-27 养生堂(上海)化妆品研发有限公司 护肤化妆品组合物
RU2660649C1 (ru) * 2017-10-18 2018-07-09 федеральное государственное бюджетное образовательное учреждение высшего образования "Приволжский исследовательский медицинский университет" Министерства здравоохранения Российской Федерации Способ получения соли 3,28-дифосфата бетулина
JP7358353B2 (ja) 2018-01-04 2023-10-10 アムリット・リサーチ・リミテッド ベツリン含有白樺樹皮抽出物およびその製剤
RU2658838C1 (ru) * 2018-02-22 2018-06-25 Федеральное государственное бюджетное научное учреждение "Федеральный исследовательский центр "Красноярский научный центр Сибирского отделения Российской академии наук" (ФИЦ КНЦ СО РАН, КНЦ СО РАН) Способ получения сукцината аллобетулина
RU2665578C1 (ru) * 2018-04-26 2018-08-31 Федеральное государственное бюджетное научное учреждение "Федеральный исследовательский центр "Красноярский научный центр Сибирского отделения Российской академии наук" (ФИЦ КНЦ СО РАН, КНЦ СО РАН) Способ получения дициннамата бетулина
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CN109498621B (zh) * 2018-12-28 2021-02-26 青岛大学附属医院 一种妇科用复方硝酸咪康唑组合物
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Also Published As

Publication number Publication date
US20020128210A1 (en) 2002-09-12
US6642217B2 (en) 2003-11-04
EP1322661A1 (en) 2003-07-02
WO2002026761A1 (en) 2002-04-04
CA2424013A1 (en) 2002-04-04
JP2004509972A (ja) 2004-04-02

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Legal Events

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MK4 Application lapsed section 142(2)(d) - no continuation fee paid for the application