AU2001240561A1 - Novel positive allosteric ampa receptor modulators (paarm), method for the production and use thereof as medicaments - Google Patents
Novel positive allosteric ampa receptor modulators (paarm), method for the production and use thereof as medicamentsInfo
- Publication number
- AU2001240561A1 AU2001240561A1 AU2001240561A AU4056101A AU2001240561A1 AU 2001240561 A1 AU2001240561 A1 AU 2001240561A1 AU 2001240561 A AU2001240561 A AU 2001240561A AU 4056101 A AU4056101 A AU 4056101A AU 2001240561 A1 AU2001240561 A1 AU 2001240561A1
- Authority
- AU
- Australia
- Prior art keywords
- paarm
- medicaments
- production
- receptor modulators
- positive allosteric
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/06—Peri-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Neurosurgery (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Neurology (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Biomedical Technology (AREA)
- Public Health (AREA)
- Psychiatry (AREA)
- Urology & Nephrology (AREA)
- Heart & Thoracic Surgery (AREA)
- Hospice & Palliative Care (AREA)
- Vascular Medicine (AREA)
- Cardiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE10004572A DE10004572A1 (de) | 2000-02-02 | 2000-02-02 | Neue positive allosterische AMPA-Rezeptor Modulatoren (PAARM), Verfahren zu deren Herstellung und deren Verwendung als Arzneimittel |
DE10004572 | 2000-02-02 | ||
PCT/EP2001/000960 WO2001057045A1 (de) | 2000-02-02 | 2001-01-30 | Neue positive allosterische ampa-rezeptor modulatoren (paarm), verfahren zu deren herstellung und deren verwendung als arzneimittel |
Publications (1)
Publication Number | Publication Date |
---|---|
AU2001240561A1 true AU2001240561A1 (en) | 2001-08-14 |
Family
ID=7629599
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AU2001240561A Abandoned AU2001240561A1 (en) | 2000-02-02 | 2001-01-30 | Novel positive allosteric ampa receptor modulators (paarm), method for the production and use thereof as medicaments |
Country Status (16)
Country | Link |
---|---|
US (3) | US6525045B2 (ja) |
EP (1) | EP1265904B1 (ja) |
JP (1) | JP4891510B2 (ja) |
AR (1) | AR027352A1 (ja) |
AT (1) | ATE277054T1 (ja) |
AU (1) | AU2001240561A1 (ja) |
CA (1) | CA2399377C (ja) |
CO (1) | CO5261505A1 (ja) |
DE (2) | DE10004572A1 (ja) |
DK (1) | DK1265904T3 (ja) |
ES (1) | ES2228817T3 (ja) |
MX (1) | MXPA02007460A (ja) |
PT (1) | PT1265904E (ja) |
TR (1) | TR200402650T4 (ja) |
UY (1) | UY26566A1 (ja) |
WO (1) | WO2001057045A1 (ja) |
Families Citing this family (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE10004572A1 (de) * | 2000-02-02 | 2001-08-09 | Boehringer Ingelheim Pharma | Neue positive allosterische AMPA-Rezeptor Modulatoren (PAARM), Verfahren zu deren Herstellung und deren Verwendung als Arzneimittel |
SK13632002A3 (sk) * | 2000-03-21 | 2003-02-04 | Smithkline Beecham Corporation | C1-6-alkyl-4-amino-azepán-3-ónové zlúčeniny, spôsob ich prípravy, farmaceutický prostriedok s ich obsahom, ich použitie a medziprodukty |
NZ529308A (en) * | 2001-04-05 | 2005-03-24 | Collagenex Pharm Inc | Tetracycline compounds comprising a tetracycline and a controlled release agent to provide delivery at a dose below that required for antibiotic activity |
US20030100552A1 (en) | 2001-05-17 | 2003-05-29 | Boehringer Ingelheim Pharma Kg | Positive allosteric AMPA receptor modulators (PAARM), processes for preparing them, and their use as pharmaceutical compositions |
DE10123952A1 (de) * | 2001-05-17 | 2002-11-21 | Boehringer Ingelheim Pharma | Neue positive allosterische AMPA-Rezeptor Modulatoren (PAARM), Verfahren zu deren Herstellung und deren Verwendung als Arzneimittel |
US7199118B2 (en) | 2001-10-10 | 2007-04-03 | Neurosearch A/S | Benzothiazine derivatives, their preparation and use |
US7815391B2 (en) * | 2004-07-23 | 2010-10-19 | Kauppila Richard W | Structural member joints |
WO2006034196A1 (en) * | 2004-09-17 | 2006-03-30 | Lifelike Biomatic Inc. | Compositions for enhancing memory and methods therefor |
EA022476B1 (ru) * | 2008-05-05 | 2016-01-29 | Лонца Лтд. | Индолсульфонильные защищенные соединения и способ их получения |
US20110218190A1 (en) * | 2008-11-10 | 2011-09-08 | The Regents Of The University Of California | Therapeutic uses of ampa receptor modulators for treatment of motor dysfunction |
AU2014277952A1 (en) | 2013-06-13 | 2016-01-28 | Veroscience Llc | Compositions and methods for treating metabolic disorders |
Family Cites Families (12)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB8724566D0 (en) * | 1987-10-20 | 1987-11-25 | Roussel Lab Ltd | Chemical compounds |
US4994452A (en) * | 1989-11-28 | 1991-02-19 | Hoechst-Roussel Pharmaceuticals Inc. | Hexahydro-1H-quino[4,3,2-ef][1,4]benzoxazepines and related compounds |
CA2130096A1 (fr) * | 1992-04-15 | 1993-10-28 | Jean-Claude Aloup | Derives d'acide 3,4-dihydro-2h-1,2,4-benzothiadiazine 1,1-dioxyde-3-carboxylique, leur preparation et les medicaments les contenant |
RU2145606C1 (ru) * | 1994-05-24 | 2000-02-20 | Ф.Хоффманн-Ля Рош Аг | Трициклические дикарбонильные производные и лекарственный препарат на их основе |
US5891871A (en) * | 1996-03-21 | 1999-04-06 | Cocensys, Inc. | Substituted 2,3-benzodiazepin-4-ones and the use thereof |
AU4345297A (en) * | 1996-09-17 | 1998-04-14 | Regents Of The University Of California, The | Benzothiadiazide derivatives and their use as allosteric up-modulators of the ampa receptor |
US5968928A (en) * | 1996-09-19 | 1999-10-19 | Warner-Lambert Company | Excitatory amino acid antagonists: fused-azacyclic quinoxalinediones and immunoassays thereof |
US5969138A (en) * | 1996-11-01 | 1999-10-19 | Mitsui Chemicals, Inc. | Pyrrolidinone derivatives |
US5985871A (en) * | 1997-12-24 | 1999-11-16 | Cortex Pharmaceuticals, Inc. | Benzoxazine compounds for enhancing synaptic response |
RU2214405C2 (ru) * | 1998-02-18 | 2003-10-20 | НьюроСёрч А/С | Новые соединения и их применение в качестве положительных модуляторов амра-рецепторов |
US6096744A (en) * | 1998-05-04 | 2000-08-01 | Warner-Lambert Company | Sulfonamide derivatives of substituted quinoxaline 2,3-diones as glutamate receptor antagonists |
DE10004572A1 (de) * | 2000-02-02 | 2001-08-09 | Boehringer Ingelheim Pharma | Neue positive allosterische AMPA-Rezeptor Modulatoren (PAARM), Verfahren zu deren Herstellung und deren Verwendung als Arzneimittel |
-
2000
- 2000-02-02 DE DE10004572A patent/DE10004572A1/de not_active Withdrawn
-
2001
- 2001-01-30 DE DE50103760T patent/DE50103760D1/de not_active Expired - Lifetime
- 2001-01-30 DK DK01911553T patent/DK1265904T3/da active
- 2001-01-30 EP EP01911553A patent/EP1265904B1/de not_active Expired - Lifetime
- 2001-01-30 AT AT01911553T patent/ATE277054T1/de active
- 2001-01-30 AU AU2001240561A patent/AU2001240561A1/en not_active Abandoned
- 2001-01-30 ES ES01911553T patent/ES2228817T3/es not_active Expired - Lifetime
- 2001-01-30 TR TR2004/02650T patent/TR200402650T4/xx unknown
- 2001-01-30 WO PCT/EP2001/000960 patent/WO2001057045A1/de active IP Right Grant
- 2001-01-30 UY UY26566A patent/UY26566A1/es not_active Application Discontinuation
- 2001-01-30 MX MXPA02007460A patent/MXPA02007460A/es active IP Right Grant
- 2001-01-30 PT PT01911553T patent/PT1265904E/pt unknown
- 2001-01-30 JP JP2001557876A patent/JP4891510B2/ja not_active Expired - Fee Related
- 2001-01-30 CA CA002399377A patent/CA2399377C/en not_active Expired - Fee Related
- 2001-01-31 CO CO01007094A patent/CO5261505A1/es not_active Application Discontinuation
- 2001-01-31 US US09/774,864 patent/US6525045B2/en not_active Expired - Lifetime
- 2001-02-02 AR ARP010100494A patent/AR027352A1/es not_active Suspension/Interruption
-
2003
- 2003-01-06 US US10/336,876 patent/US20030158181A1/en not_active Abandoned
- 2003-01-06 US US10/336,865 patent/US6800623B2/en not_active Expired - Lifetime
Also Published As
Publication number | Publication date |
---|---|
MXPA02007460A (es) | 2003-01-28 |
CO5261505A1 (es) | 2003-03-31 |
TR200402650T4 (tr) | 2004-11-22 |
DE50103760D1 (de) | 2004-10-28 |
UY26566A1 (es) | 2001-08-27 |
AR027352A1 (es) | 2003-03-26 |
EP1265904A1 (de) | 2002-12-18 |
CA2399377A1 (en) | 2001-08-09 |
WO2001057045A1 (de) | 2001-08-09 |
ES2228817T3 (es) | 2005-04-16 |
US20030158183A1 (en) | 2003-08-21 |
DK1265904T3 (da) | 2004-10-25 |
US20030158181A1 (en) | 2003-08-21 |
JP2003522180A (ja) | 2003-07-22 |
JP4891510B2 (ja) | 2012-03-07 |
DE10004572A1 (de) | 2001-08-09 |
PT1265904E (pt) | 2004-11-30 |
EP1265904B1 (de) | 2004-09-22 |
US20020013313A1 (en) | 2002-01-31 |
ATE277054T1 (de) | 2004-10-15 |
US6800623B2 (en) | 2004-10-05 |
US6525045B2 (en) | 2003-02-25 |
CA2399377C (en) | 2008-12-16 |
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