AU2001234273A1 - Thiazolopyrimidines and their use as modulators of chemokine receptor activity - Google Patents

Thiazolopyrimidines and their use as modulators of chemokine receptor activity

Info

Publication number
AU2001234273A1
AU2001234273A1 AU2001234273A AU3427301A AU2001234273A1 AU 2001234273 A1 AU2001234273 A1 AU 2001234273A1 AU 2001234273 A AU2001234273 A AU 2001234273A AU 3427301 A AU3427301 A AU 3427301A AU 2001234273 A1 AU2001234273 A1 AU 2001234273A1
Authority
AU
Australia
Prior art keywords
thiazolopyrimidines
modulators
chemokine receptor
receptor activity
compounds
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU2001234273A
Other languages
English (en)
Inventor
Roger Bonnert
Peter Cage
Fraser Hunt
Robert Jewell
Iain Walters
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
AstraZeneca AB
Original Assignee
AstraZeneca AB
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by AstraZeneca AB filed Critical AstraZeneca AB
Publication of AU2001234273A1 publication Critical patent/AU2001234273A1/en
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/06—Antipsoriatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Dermatology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Pulmonology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
AU2001234273A 2000-02-11 2001-02-07 Thiazolopyrimidines and their use as modulators of chemokine receptor activity Abandoned AU2001234273A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB0003025 2000-02-11
GB0003025A GB2359081A (en) 2000-02-11 2000-02-11 Pharmaceutically active thiazolopyrimidines
PCT/SE2001/000247 WO2001058907A1 (en) 2000-02-11 2001-02-07 Thiazolopyrimidines and their use as modulators of chemokine receptor activity

Publications (1)

Publication Number Publication Date
AU2001234273A1 true AU2001234273A1 (en) 2001-08-20

Family

ID=9885290

Family Applications (1)

Application Number Title Priority Date Filing Date
AU2001234273A Abandoned AU2001234273A1 (en) 2000-02-11 2001-02-07 Thiazolopyrimidines and their use as modulators of chemokine receptor activity

Country Status (8)

Country Link
US (1) US6958343B2 (cg-RX-API-DMAC7.html)
EP (1) EP1257556B1 (cg-RX-API-DMAC7.html)
JP (1) JP2003522192A (cg-RX-API-DMAC7.html)
AT (1) ATE269340T1 (cg-RX-API-DMAC7.html)
AU (1) AU2001234273A1 (cg-RX-API-DMAC7.html)
DE (1) DE60103856T2 (cg-RX-API-DMAC7.html)
GB (1) GB2359081A (cg-RX-API-DMAC7.html)
WO (1) WO2001058907A1 (cg-RX-API-DMAC7.html)

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GB2359551A (en) * 2000-02-23 2001-08-29 Astrazeneca Uk Ltd Pharmaceutically active pyrimidine derivatives
SE0003828D0 (sv) 2000-10-20 2000-10-20 Astrazeneca Ab Novel compounds
SE0101082D0 (sv) * 2001-03-27 2001-03-27 Astrazeneca Ab Novel use
SE0101322D0 (sv) 2001-04-12 2001-04-12 Astrazeneca Ab Novel compounds
SE0102716D0 (sv) * 2001-08-14 2001-08-14 Astrazeneca Ab Novel compounds
DE60304718T2 (de) 2002-08-06 2007-04-26 Astrazeneca Ab Kondensierte pyridine und pyrimidine mit tie2 (tek) aktivität
GB0221829D0 (en) * 2002-09-20 2002-10-30 Astrazeneca Ab Novel compound
GB0221828D0 (en) * 2002-09-20 2002-10-30 Astrazeneca Ab Novel compound
GB0328243D0 (en) * 2003-12-05 2004-01-07 Astrazeneca Ab Methods
UA90707C2 (en) 2005-04-06 2010-05-25 Астразенека Аб Novel 5-substituted 7-amino-[1,3]thiazolo[4,5-d]pyrimidine derivatives
AR053347A1 (es) 2005-04-06 2007-05-02 Astrazeneca Ab Derivados de [1,3]tiazolo[4,5-d]pirimidin-2(3h)-ona 5,7-sustituidos
TW200820973A (en) 2006-09-29 2008-05-16 Astrazeneca Ab Novel compounds 480
EP2069365A4 (en) * 2006-09-29 2011-11-02 Astrazeneca Ab NOVEL [1, 3] THIAZOLO [4,5-D] PYRIMIDIN-2 (3H) -AMINE 5,7-DISUBSTITUTED DERIVATIVES AND THEIR USE IN THERAPY
US9040538B2 (en) * 2009-05-21 2015-05-26 Universite Laval Pyrimidines as novel therapeutic agents

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Also Published As

Publication number Publication date
DE60103856T2 (de) 2005-07-14
US20030032642A1 (en) 2003-02-13
US6958343B2 (en) 2005-10-25
EP1257556B1 (en) 2004-06-16
DE60103856D1 (de) 2004-07-22
EP1257556A1 (en) 2002-11-20
WO2001058907A1 (en) 2001-08-16
JP2003522192A (ja) 2003-07-22
ATE269340T1 (de) 2004-07-15
GB0003025D0 (en) 2000-03-29
GB2359081A (en) 2001-08-15

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