ATE509941T1 - Cycloalkylcarbonylaminosäureester-derivat und herstellungsverfahren dafür - Google Patents
Cycloalkylcarbonylaminosäureester-derivat und herstellungsverfahren dafürInfo
- Publication number
- ATE509941T1 ATE509941T1 AT07706501T AT07706501T ATE509941T1 AT E509941 T1 ATE509941 T1 AT E509941T1 AT 07706501 T AT07706501 T AT 07706501T AT 07706501 T AT07706501 T AT 07706501T AT E509941 T1 ATE509941 T1 AT E509941T1
- Authority
- AT
- Austria
- Prior art keywords
- acid ester
- groups
- ester derivative
- cycloalkylcarbonylaminosic
- production
- Prior art date
Links
- 239000002253 acid Substances 0.000 title abstract 3
- 150000002148 esters Chemical class 0.000 title abstract 3
- 238000004519 manufacturing process Methods 0.000 title abstract 2
- 125000000217 alkyl group Chemical group 0.000 abstract 2
- 125000004432 carbon atom Chemical group C* 0.000 abstract 2
- 125000005169 cycloalkylcarbonylamino group Chemical group 0.000 abstract 2
- 102000004171 Cathepsin K Human genes 0.000 abstract 1
- 108090000625 Cathepsin K Proteins 0.000 abstract 1
- 125000003342 alkenyl group Chemical group 0.000 abstract 1
- 125000001118 alkylidene group Chemical group 0.000 abstract 1
- 125000000304 alkynyl group Chemical group 0.000 abstract 1
- 125000002029 aromatic hydrocarbon group Chemical group 0.000 abstract 1
- 125000004122 cyclic group Chemical group 0.000 abstract 1
- -1 cycloalkane carboxamide Chemical class 0.000 abstract 1
- 125000000623 heterocyclic group Chemical group 0.000 abstract 1
- 239000000543 intermediate Substances 0.000 abstract 1
- 239000002994 raw material Substances 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C07K5/06008—Dipeptides with the first amino acid being neutral
- C07K5/06078—Dipeptides with the first amino acid being neutral and aromatic or cycloaliphatic
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Genetics & Genomics (AREA)
- Biochemistry (AREA)
- Biophysics (AREA)
- General Health & Medical Sciences (AREA)
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Molecular Biology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2006003508 | 2006-01-11 | ||
| JP2006343582 | 2006-12-20 | ||
| PCT/JP2007/050154 WO2007080884A1 (ja) | 2006-01-11 | 2007-01-10 | シクロアルキルカルボニルアミノ酸エステル誘導体及びその製造方法 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ATE509941T1 true ATE509941T1 (de) | 2011-06-15 |
Family
ID=38256289
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT07706501T ATE509941T1 (de) | 2006-01-11 | 2007-01-10 | Cycloalkylcarbonylaminosäureester-derivat und herstellungsverfahren dafür |
Country Status (6)
| Country | Link |
|---|---|
| US (1) | US8829209B2 (de) |
| EP (1) | EP2036920B1 (de) |
| AT (1) | ATE509941T1 (de) |
| AU (1) | AU2007205578B2 (de) |
| CA (1) | CA2636765C (de) |
| WO (1) | WO2007080884A1 (de) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP4012239B2 (ja) | 2006-01-11 | 2007-11-21 | 生化学工業株式会社 | オキサゾロン誘導体 |
| JP4047365B2 (ja) * | 2006-01-11 | 2008-02-13 | 生化学工業株式会社 | シクロアルカンカルボキサミド誘導体及びその製造方法 |
| JP3975226B2 (ja) * | 2006-01-11 | 2007-09-12 | 生化学工業株式会社 | シクロアルキルカルボニルアミノ酸誘導体及びその製造方法 |
| ATE509941T1 (de) | 2006-01-11 | 2011-06-15 | Seikagaku Kogyo Co Ltd | Cycloalkylcarbonylaminosäureester-derivat und herstellungsverfahren dafür |
| WO2009132453A1 (en) * | 2008-04-28 | 2009-11-05 | Neuromed Pharmaceuticals Ltd. | Cyclylamine derivatives as calcium channel blockers |
| IT1394304B1 (it) * | 2009-05-21 | 2012-06-06 | Malesci Sas | Processo per la preparazione di ibodutant (men15596) e relativi intermedi |
| WO2014199644A1 (ja) * | 2013-06-14 | 2014-12-18 | 生化学工業株式会社 | α-オキソアシルアミノカプロラクタム誘導体 |
Family Cites Families (25)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CS231227B1 (en) | 1982-10-01 | 1984-10-15 | Evzen Kasafirek | 2,5-pierazindion derivatives |
| ZA897515B (en) | 1988-10-07 | 1990-06-27 | Merrell Dow Pharma | Novel peptidase inhibitors |
| JP2701932B2 (ja) | 1989-04-10 | 1998-01-21 | サントリー株式会社 | タンパク質分解酵素阻害剤 |
| JPH04202170A (ja) | 1990-11-29 | 1992-07-22 | Taisho Pharmaceut Co Ltd | トリペプチド誘導体 |
| EP0729972A1 (de) * | 1995-02-28 | 1996-09-04 | F. Hoffmann-La Roche Ag | Tetrahydronaphthalin-Peptidderivate |
| US6162828A (en) * | 1995-03-31 | 2000-12-19 | Takeda Chemical Industries, Ltd. | Cysteine protease inhibitor |
| JPH09165360A (ja) | 1995-03-31 | 1997-06-24 | Takeda Chem Ind Ltd | システインプロテアーゼ阻害剤 |
| EP0835349B1 (de) | 1995-06-29 | 1999-09-22 | Minnesota Mining And Manufacturing Company | Retroreflektierender markierungskörper für nasse umgebungsbedingungen |
| EP0804180A4 (de) | 1995-10-30 | 2001-09-05 | Smithkline Beecham Corp | Verfahren zur cathepsinhemmung |
| AU3359697A (en) | 1996-07-08 | 1998-02-02 | Yamanouchi Pharmaceutical Co., Ltd. | Bone resorption inhibitors |
| DE69923676T2 (de) | 1998-04-23 | 2006-01-12 | Novartis Ag | Bestimmte heteroaryl substituierte thiol inhibitoren von endothelin wechselnden enzymen |
| IL138246A0 (en) | 1998-04-23 | 2001-10-31 | Novartis Ag | Certain thiol inhibitors of endothelin-converting enzyme |
| JP3892187B2 (ja) | 1998-11-12 | 2007-03-14 | 生化学工業株式会社 | 環状アミド誘導体 |
| US6117870A (en) * | 1998-11-12 | 2000-09-12 | Fujirebio Kabushiki Kaisha | Cyclic amide derivatives |
| JP2003524614A (ja) | 1998-12-22 | 2003-08-19 | 田辺製薬株式会社 | α4β1媒介細胞接着のインヒビター |
| JP2001139534A (ja) | 1999-11-16 | 2001-05-22 | Yoshimitsu Nagao | バリン誘導体およびその用途 |
| GB0003111D0 (en) | 2000-02-10 | 2000-03-29 | Novartis Ag | Organic compounds |
| SV2003000617A (es) * | 2000-08-31 | 2003-01-13 | Lilly Co Eli | Inhibidores de la proteasa peptidomimetica ref. x-14912m |
| AU2002258794A1 (en) * | 2001-04-10 | 2003-10-20 | Transtech Pharma, Inc. | Probes, systems and methods for drug discovery |
| PT1430045E (pt) * | 2001-09-21 | 2007-01-31 | Novartis Ag | Derivados de pirano como inibidores de ace e nep |
| JP4202170B2 (ja) | 2003-03-28 | 2008-12-24 | 三菱電機株式会社 | 空気調和装置 |
| US20050192279A1 (en) * | 2004-02-10 | 2005-09-01 | Kent Barbay | Pyridazinones as antagonists of alpha4 integrins |
| JP3975226B2 (ja) * | 2006-01-11 | 2007-09-12 | 生化学工業株式会社 | シクロアルキルカルボニルアミノ酸誘導体及びその製造方法 |
| JP4047365B2 (ja) * | 2006-01-11 | 2008-02-13 | 生化学工業株式会社 | シクロアルカンカルボキサミド誘導体及びその製造方法 |
| ATE509941T1 (de) | 2006-01-11 | 2011-06-15 | Seikagaku Kogyo Co Ltd | Cycloalkylcarbonylaminosäureester-derivat und herstellungsverfahren dafür |
-
2007
- 2007-01-10 AT AT07706501T patent/ATE509941T1/de not_active IP Right Cessation
- 2007-01-10 US US12/087,619 patent/US8829209B2/en not_active Expired - Fee Related
- 2007-01-10 CA CA2636765A patent/CA2636765C/en not_active Expired - Fee Related
- 2007-01-10 AU AU2007205578A patent/AU2007205578B2/en not_active Ceased
- 2007-01-10 WO PCT/JP2007/050154 patent/WO2007080884A1/ja not_active Ceased
- 2007-01-10 EP EP07706501A patent/EP2036920B1/de not_active Not-in-force
Also Published As
| Publication number | Publication date |
|---|---|
| EP2036920B1 (de) | 2011-05-18 |
| AU2007205578B2 (en) | 2012-06-28 |
| US20090137799A1 (en) | 2009-05-28 |
| WO2007080884A1 (ja) | 2007-07-19 |
| AU2007205578A1 (en) | 2007-07-19 |
| CA2636765A1 (en) | 2007-07-19 |
| CA2636765C (en) | 2014-03-18 |
| EP2036920A4 (de) | 2009-07-29 |
| US8829209B2 (en) | 2014-09-09 |
| EP2036920A1 (de) | 2009-03-18 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| ATE509941T1 (de) | Cycloalkylcarbonylaminosäureester-derivat und herstellungsverfahren dafür | |
| EP1541561A4 (de) | Pyrazolderivate und verfahren zu deren herstellung | |
| NZ601567A (en) | Process for production of delta-9-tetrahydrocannabinol | |
| CR10250A (es) | Derivados de amida y su aplicación para el tratamiento de enfermedades relacionadas con proteína-g | |
| MX2010008361A (es) | Derivados de arilamida oxazepinopirimidona sustituidos. | |
| GB0719180D0 (en) | New process | |
| GB0601744D0 (en) | Organic compounds | |
| MX2011008501A (es) | Compuestos heterociclicos fusionados que contienen nitrogeno y su uso como inhibidores de la produccion de beta-amiloide. | |
| MX2009008781A (es) | Derivados de ciclohexano espirociclicos. | |
| AR066023A1 (es) | Compuestos heterociclicos nitrogenados, su preparacion y su utilizacion como medicamentos antibacterianos | |
| PL2229356T3 (pl) | 1,2-Dipodstawione pochodne 4-benzyloamino-pirolidyny jako inhibitory CETP użyteczne do leczenia chorób, takich jak hiperlipidemia lub stwardnienie tętnic | |
| CN111727190A (zh) | 一种吡啶基咪唑并苯并二氮杂卓丙酸酯化合物及其合成和应用 | |
| ATE517869T1 (de) | Herstellung substituierter morphinan-6-one und salzen und zwischenprodukten davon | |
| ATE510844T1 (de) | Cycloalkylcarbonylaminosäure-derivat und herstellungsverfahren dafür | |
| MX2010008360A (es) | Derivados de oxazepinopirimidona heteroarilamida sustituidos. | |
| NZ586187A (en) | Processes for the synthesis of sinomenine derivatives and their intermediate | |
| ATE501103T1 (de) | Organische verbindungen | |
| MY148769A (en) | Process for the synthesis of derivatives of 3-amino-tetrahydrofuran-3-carboxylic acid and use thereof as medicaments | |
| NO20071319L (no) | Fremgangsmate for fremstilling av isotiazolderivater. | |
| MY156304A (en) | 5-hydroxymethyl-oxazolidin-2-one derivatives for treating bacterial intestinal diseases | |
| MXPA03011682A (es) | Derivados sustituidos de n-acil -anilina, su preparacion y su uso como medicamento. | |
| WO2010094666A3 (en) | Fungicidal n-(phenylcycloalkyl)carboxamide, n-(benzylcycloalkyl)carboxamide and thiocarboxamide derivatives | |
| TW200738693A (en) | Substituted biaryls, process for their manufacture and use thereof as medicaments | |
| EP1486500A4 (de) | 10-(3-cyclo propyl amino methyl-1-pyrrolidinyl) pyridobenzoxazin carbonsäure derivat mit wirkung gegen resistente bakterien | |
| GB2470170A (en) | Dithienothiophene derivatives |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| RER | Ceased as to paragraph 5 lit. 3 law introducing patent treaties |