ATE455776T1 - Nikotinische alpha-7-rezeptorliganden gegen erkrankungen des zns - Google Patents
Nikotinische alpha-7-rezeptorliganden gegen erkrankungen des znsInfo
- Publication number
- ATE455776T1 ATE455776T1 AT05854897T AT05854897T ATE455776T1 AT E455776 T1 ATE455776 T1 AT E455776T1 AT 05854897 T AT05854897 T AT 05854897T AT 05854897 T AT05854897 T AT 05854897T AT E455776 T1 ATE455776 T1 AT E455776T1
- Authority
- AT
- Austria
- Prior art keywords
- receptor ligands
- cns diseases
- nicotinic alpha
- ligands against
- against cns
- Prior art date
Links
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D453/00—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
- C07D453/02—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/439—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom the ring forming part of a bridged ring system, e.g. quinuclidine
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P21/00—Drugs for disorders of the muscular or neuromuscular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A61P25/32—Alcohol-abuse
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A61P25/34—Tobacco-abuse
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US63777104P | 2004-12-22 | 2004-12-22 | |
PCT/US2005/046256 WO2006069097A2 (en) | 2004-12-22 | 2005-12-21 | Nicotinic alpha-7 receptor ligands and preparation and uses thereof |
Publications (1)
Publication Number | Publication Date |
---|---|
ATE455776T1 true ATE455776T1 (de) | 2010-02-15 |
Family
ID=36177987
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AT05854897T ATE455776T1 (de) | 2004-12-22 | 2005-12-21 | Nikotinische alpha-7-rezeptorliganden gegen erkrankungen des zns |
Country Status (15)
Country | Link |
---|---|
US (2) | US7625924B2 (de) |
EP (1) | EP1828179B1 (de) |
JP (1) | JP2008525464A (de) |
KR (1) | KR20070087674A (de) |
CN (1) | CN101124224A (de) |
AT (1) | ATE455776T1 (de) |
AU (1) | AU2005319248A1 (de) |
BR (1) | BRPI0517494A (de) |
CA (1) | CA2591817A1 (de) |
DE (1) | DE602005019094D1 (de) |
ES (1) | ES2342675T3 (de) |
MX (1) | MX2007007328A (de) |
PL (1) | PL1828179T3 (de) |
RU (1) | RU2418797C2 (de) |
WO (1) | WO2006069097A2 (de) |
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US8252321B2 (en) | 2004-09-13 | 2012-08-28 | Chrono Therapeutics, Inc. | Biosynchronous transdermal drug delivery for longevity, anti-aging, fatigue management, obesity, weight loss, weight management, delivery of nutraceuticals, and the treatment of hyperglycemia, alzheimer's disease, sleep disorders, parkinson's disease, aids, epilepsy, attention deficit disorder, nicotine addiction, cancer, headache and pain control, asthma, angina, hypertension, depression, cold, flu and the like |
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KR101122469B1 (ko) * | 2007-04-02 | 2012-07-12 | 파킨슨즈 인스티튜트 | 처치 치료의 부작용을 감소시키기 위한 방법 및 조성물 |
SA08290475B1 (ar) * | 2007-08-02 | 2013-06-22 | Targacept Inc | (2s، 3r)-n-(2-((3-بيردينيل)ميثيل)-1-آزا بيسيكلو[2، 2، 2]أوكت-3-يل)بنزو فيوران-2-كربوكساميد، وصور أملاحه الجديدة وطرق استخدامه |
CA2701126A1 (en) * | 2007-10-01 | 2009-04-09 | Comentis, Inc. | 4-substituted quinuclidine derivatives, methods of production, and pharmaceutical uses thereof |
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PL2346833T3 (pl) * | 2008-10-13 | 2013-08-30 | Hoffmann La Roche | Wolny od soli diazoniowych sposób wytwarzania indazolowego związku pośredniego w syntezie bicyklicznych amidów kwasów 5-(trifluormetoksy)-1H-3-indazolokarboksylowych |
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KR101928505B1 (ko) * | 2011-01-28 | 2018-12-12 | 에스케이바이오팜 주식회사 | 피리돈 유도체 및 이를 포함하는 약학적 조성물 |
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WO2016007630A1 (en) | 2014-07-11 | 2016-01-14 | Alpharmagen, Llc | Quinuclidine compounds for modulating alpha7 -nicotinic acetylcholine receptor activity |
US10213586B2 (en) | 2015-01-28 | 2019-02-26 | Chrono Therapeutics Inc. | Drug delivery methods and systems |
AU2016228779A1 (en) | 2015-03-12 | 2017-09-07 | Chrono Therapeutics Inc. | Craving input and support system |
JP2018516973A (ja) * | 2015-06-10 | 2018-06-28 | フォーラム・ファーマシューティカルズ・インコーポレイテッドForum Pharmaceuticals Inc. | α7−ニコチン性アセチルコリン受容体のアゴニストとしてのアミノベンゾイソオキサゾール化合物 |
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AU2018205529B2 (en) | 2017-01-06 | 2023-08-10 | Morningside Venture Investments Limited | Transdermal drug delivery devices and methods |
CA3101966A1 (en) | 2018-05-29 | 2019-12-05 | Morningside Venture Investments Limited | Drug delivery methods and systems |
CN111808907B (zh) * | 2019-10-09 | 2021-07-09 | 北京原基华毅生物科技有限公司 | 调整觉醒的物质及方法 |
WO2023230540A2 (en) * | 2022-05-25 | 2023-11-30 | Katholieke Universiteit Leuven | Indazole derivatives for treating trpm3-mediated disorders |
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-
2005
- 2005-12-21 MX MX2007007328A patent/MX2007007328A/es active IP Right Grant
- 2005-12-21 AT AT05854897T patent/ATE455776T1/de active
- 2005-12-21 DE DE602005019094T patent/DE602005019094D1/de active Active
- 2005-12-21 PL PL05854897T patent/PL1828179T3/pl unknown
- 2005-12-21 RU RU2007128062/04A patent/RU2418797C2/ru not_active IP Right Cessation
- 2005-12-21 WO PCT/US2005/046256 patent/WO2006069097A2/en active Application Filing
- 2005-12-21 CN CNA2005800485590A patent/CN101124224A/zh active Pending
- 2005-12-21 KR KR1020077016683A patent/KR20070087674A/ko not_active Application Discontinuation
- 2005-12-21 AU AU2005319248A patent/AU2005319248A1/en not_active Abandoned
- 2005-12-21 CA CA002591817A patent/CA2591817A1/en not_active Abandoned
- 2005-12-21 JP JP2007548401A patent/JP2008525464A/ja active Pending
- 2005-12-21 BR BRPI0517494-5A patent/BRPI0517494A/pt not_active IP Right Cessation
- 2005-12-21 EP EP05854897A patent/EP1828179B1/de not_active Not-in-force
- 2005-12-21 US US11/312,831 patent/US7625924B2/en not_active Expired - Fee Related
- 2005-12-21 ES ES05854897T patent/ES2342675T3/es active Active
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Also Published As
Publication number | Publication date |
---|---|
EP1828179B1 (de) | 2010-01-20 |
ES2342675T3 (es) | 2010-07-12 |
US20100016351A1 (en) | 2010-01-21 |
BRPI0517494A (pt) | 2008-10-14 |
WO2006069097A3 (en) | 2006-10-05 |
CN101124224A (zh) | 2008-02-13 |
US7625924B2 (en) | 2009-12-01 |
PL1828179T3 (pl) | 2010-08-31 |
KR20070087674A (ko) | 2007-08-28 |
DE602005019094D1 (de) | 2010-03-11 |
EP1828179A2 (de) | 2007-09-05 |
WO2006069097A2 (en) | 2006-06-29 |
MX2007007328A (es) | 2007-07-25 |
RU2418797C2 (ru) | 2011-05-20 |
AU2005319248A1 (en) | 2006-06-29 |
US20060167039A1 (en) | 2006-07-27 |
JP2008525464A (ja) | 2008-07-17 |
CA2591817A1 (en) | 2006-06-29 |
RU2007128062A (ru) | 2009-01-27 |
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