ATE407932T1 - Wasserlösliches triazolfungizid - Google Patents

Wasserlösliches triazolfungizid

Info

Publication number
ATE407932T1
ATE407932T1 AT02701569T AT02701569T ATE407932T1 AT E407932 T1 ATE407932 T1 AT E407932T1 AT 02701569 T AT02701569 T AT 02701569T AT 02701569 T AT02701569 T AT 02701569T AT E407932 T1 ATE407932 T1 AT E407932T1
Authority
AT
Austria
Prior art keywords
water soluble
triazole fungicide
soluble triazole
group
fungicide
Prior art date
Application number
AT02701569T
Other languages
English (en)
Inventor
Makoto Mori
Yoshiko Kagoshima
Takuya Uchida
Toshiyuki Konosu
Takahiro Shibayama
Original Assignee
Daiichi Sankyo Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Daiichi Sankyo Co Ltd filed Critical Daiichi Sankyo Co Ltd
Application granted granted Critical
Publication of ATE407932T1 publication Critical patent/ATE407932T1/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10Antimycotics
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D249/00Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/081,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/06Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/06Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/14Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/06Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/547Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6515Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having three nitrogen atoms as the only ring hetero atoms
    • C07F9/6518Five-membered rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/547Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6558Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing at least two different or differently substituted hetero rings neither condensed among themselves nor condensed with a common carbocyclic ring or ring system
    • C07F9/65586Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing at least two different or differently substituted hetero rings neither condensed among themselves nor condensed with a common carbocyclic ring or ring system at least one of the hetero rings does not contain nitrogen as ring hetero atom

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Oncology (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Communicable Diseases (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicinal Preparation (AREA)
AT02701569T 2001-02-22 2002-02-20 Wasserlösliches triazolfungizid ATE407932T1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP2001046890 2001-02-22

Publications (1)

Publication Number Publication Date
ATE407932T1 true ATE407932T1 (de) 2008-09-15

Family

ID=18908429

Family Applications (1)

Application Number Title Priority Date Filing Date
AT02701569T ATE407932T1 (de) 2001-02-22 2002-02-20 Wasserlösliches triazolfungizid

Country Status (22)

Country Link
US (1) US7230023B2 (de)
EP (1) EP1362856B1 (de)
KR (1) KR100851800B1 (de)
CN (2) CN100349569C (de)
AT (1) ATE407932T1 (de)
AU (1) AU2002234892C9 (de)
BR (1) BR0207534A (de)
CA (1) CA2439001C (de)
CZ (1) CZ20032218A3 (de)
DE (1) DE60228821D1 (de)
ES (1) ES2314028T3 (de)
HU (1) HUP0303249A3 (de)
IL (1) IL157440A0 (de)
MX (1) MXPA03007588A (de)
NO (1) NO326520B1 (de)
NZ (1) NZ527693A (de)
PL (1) PL363523A1 (de)
PT (1) PT1362856E (de)
RU (1) RU2276670C2 (de)
SK (1) SK10592003A3 (de)
WO (1) WO2002066465A1 (de)
ZA (1) ZA200306547B (de)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2003264533A1 (en) * 2002-09-20 2004-04-08 Sankyo Company, Limited Water-soluble triazole compound
ATE492523T1 (de) * 2004-08-05 2011-01-15 Sumitomo Chemical Co Verfahren zur herstellung von halogensubstituiertem benzoldimethanol
KR100738228B1 (ko) 2006-02-22 2007-07-12 한국화학연구원 아졸계 항균제 화합물 및 그의 제조방법
TW200817424A (en) 2006-08-04 2008-04-16 Daiichi Sankyo Co Ltd Benzylphenyl glucopyranoside derivatives
JP2010505811A (ja) 2006-10-04 2010-02-25 ファイザー・プロダクツ・インク カルシウム受容体アンタゴニストとしてのピリド[4,3−d]ピリミジン−4(3H)−オン誘導体
EP2326180B1 (de) * 2008-08-12 2013-10-16 Merck Sharp & Dohme Corp. Antimykotika
CN104877001B (zh) * 2008-08-12 2020-07-03 西尼克斯公司 抗真菌制剂
CN103508981A (zh) * 2012-06-18 2014-01-15 北京美倍他药物研究有限公司 新的哌嗪衍生物及其医药用途
CN107556294A (zh) * 2016-06-30 2018-01-09 陕西合成药业股份有限公司 一种新型抗真菌感染药物及其制备方法和用途
AU2020396543A1 (en) 2019-12-06 2022-06-16 Celgene Corporation Processes for preparing 2-(4-chlorophenyl)-N-((2-(2,6-dioxopiperidin-3-yl)-1-oxoisoindolin-5-yl)methyl)-2,2-difluoroacetamide

Family Cites Families (32)

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GB2104065B (en) * 1981-06-04 1985-11-06 Ciba Geigy Ag Heterocyclyl-substituted mandelic acid compounds and mandelonitriles and their use for combating microorganisms
CS228931B2 (cs) 1981-06-06 1984-05-14 Pfizer Způsob výroby 2-(2,4-difluorfenyl)-l,3-bis(lH-l,2,4-triazol-l-yl)propan- -2-oiu
EP0069442B1 (de) 1981-06-06 1985-02-20 Pfizer Limited Fungizide Mittel, Verfahren zu deren Herstellung, und diese enthaltende pharmazeutische Zusammenstellungen
JPS6214766A (ja) 1985-07-11 1987-01-23 Tokyu Foods:Kk 肉そばの製造法
RU2039050C1 (ru) * 1989-09-26 1995-07-09 Такеда Кемикал Индастриз ЛТД Производные 1,2,4-триазола, оптически инертные или имеющие r- или s-конфигурацию c-2 и c-3 асимметричных центров, или их соли, обладающие фунгицидной активностью, и способ их получения
GB9002375D0 (en) 1990-02-02 1990-04-04 Pfizer Ltd Triazole antifungal agents
NO913302L (no) * 1990-08-26 1992-03-02 Sankyo Co Anti-fungale triazolderivater, samt fremstilling og anvendelse derav
KR920019763A (ko) * 1991-04-26 1992-11-19 모리다 가즈라 아졸 화합물, 그의 제조방법 및 용도
JP3050982B2 (ja) 1991-12-13 2000-06-12 富山化学工業株式会社 新規なトリアゾール誘導体およびその塩
US5622944A (en) * 1992-06-12 1997-04-22 Affymax Technologies N.V. Testosterone prodrugs for improved drug delivery
JPH05345768A (ja) 1992-06-13 1993-12-27 Nippon Nohyaku Co Ltd 新規トリアゾール化合物及び該化合物を有効成分とする抗真菌剤
TW297813B (de) * 1993-09-24 1997-02-11 Takeda Pharm Industry Co Ltd
JP3635686B2 (ja) 1994-08-10 2005-04-06 エーザイ株式会社 抗真菌剤及びその製造方法
NZ270418A (en) * 1994-02-07 1997-09-22 Eisai Co Ltd Polycyclic triazole & imidazole derivatives, antifungal compositions
JPH09505083A (ja) 1994-03-12 1997-05-20 ユーハン・コーポレーション トリアゾール化合物およびその製造方法
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ATE206410T1 (de) * 1995-04-06 2001-10-15 Sankyo Co Triazole als fungizide mittel.
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JP3638438B2 (ja) 1997-12-26 2005-04-13 エスエス製薬株式会社 トリアゾール誘導体またはその塩、その製造方法及び当該化合物を有効成分とする医薬
WO1999045008A1 (en) 1998-03-06 1999-09-10 F. Hoffmann-La Roche Ag 3-[4-(4-cyanophenyl)thiazol-2-y)]-1-(1h-1,2,4-triazol-1-yl)-butan-2-ol derivatives having antifungal activity
US6265584B1 (en) * 1998-05-22 2001-07-24 Bristol-Myers Squibb Company Water soluble prodrugs of azole compounds
AU1177200A (en) 1998-11-10 2000-05-29 Meiji Seika Kaisha Ltd. Novel imidazo(5,1-B)thiazole derivatives and fungicides containing the same as the active ingredient
AU1915500A (en) * 1998-11-20 2000-06-13 Bristol-Myers Squibb Company Water soluble prodrugs of azole compounds
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Also Published As

Publication number Publication date
CN1720913A (zh) 2006-01-18
CA2439001C (en) 2010-05-04
HUP0303249A2 (hu) 2004-01-28
AU2002234892C1 (en) 2005-06-02
PL363523A1 (en) 2004-11-29
AU2002234892A1 (en) 2003-02-27
NO20033723D0 (no) 2003-08-21
CN1503795A (zh) 2004-06-09
CZ20032218A3 (cs) 2004-03-17
DE60228821D1 (de) 2008-10-23
CA2439001A1 (en) 2002-08-29
RU2276670C2 (ru) 2006-05-20
ES2314028T3 (es) 2009-03-16
HK1058037A1 (en) 2004-04-30
HUP0303249A3 (en) 2007-03-28
SK10592003A3 (sk) 2004-05-04
NZ527693A (en) 2004-10-29
MXPA03007588A (es) 2003-12-04
AU2002234892B2 (en) 2005-01-06
ZA200306547B (en) 2004-09-01
IL157440A0 (en) 2004-03-28
NO326520B1 (no) 2008-12-22
WO2002066465A1 (en) 2002-08-29
NO20033723L (no) 2003-10-21
EP1362856A1 (de) 2003-11-19
CN100430390C (zh) 2008-11-05
US20040198790A1 (en) 2004-10-07
CN100349569C (zh) 2007-11-21
RU2003125879A (ru) 2005-03-20
KR100851800B1 (ko) 2008-08-13
PT1362856E (pt) 2008-12-16
US7230023B2 (en) 2007-06-12
KR20030080030A (ko) 2003-10-10
AU2002234892C9 (en) 2006-01-05
EP1362856A4 (de) 2004-11-24
EP1362856B1 (de) 2008-09-10
BR0207534A (pt) 2004-07-20

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