ATE222587T1 - TROPAN-2-ALDOXIMDERIVATE ALS NEUROTRANSMITTER ßREUPTAKEß INHIBITOREN - Google Patents
TROPAN-2-ALDOXIMDERIVATE ALS NEUROTRANSMITTER ßREUPTAKEß INHIBITORENInfo
- Publication number
- ATE222587T1 ATE222587T1 AT95915869T AT95915869T ATE222587T1 AT E222587 T1 ATE222587 T1 AT E222587T1 AT 95915869 T AT95915869 T AT 95915869T AT 95915869 T AT95915869 T AT 95915869T AT E222587 T1 ATE222587 T1 AT E222587T1
- Authority
- AT
- Austria
- Prior art keywords
- pct
- inhibitors
- ßreuptakeß
- tropan
- neurotransmitters
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D451/00—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
- C07D451/02—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/26—Psychostimulants, e.g. nicotine, cocaine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DK44794 | 1994-04-19 | ||
DK133894 | 1994-11-24 | ||
PCT/EP1995/001358 WO1995028401A1 (en) | 1994-04-19 | 1995-04-12 | Tropane-2-aldoxine derivatives as neurotransmitter reuptake inhibitors |
Publications (1)
Publication Number | Publication Date |
---|---|
ATE222587T1 true ATE222587T1 (de) | 2002-09-15 |
Family
ID=26064021
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AT95915869T ATE222587T1 (de) | 1994-04-19 | 1995-04-12 | TROPAN-2-ALDOXIMDERIVATE ALS NEUROTRANSMITTER ßREUPTAKEß INHIBITOREN |
Country Status (25)
Country | Link |
---|---|
US (1) | US5736556A (de) |
EP (1) | EP0756596B1 (de) |
JP (1) | JP2899418B2 (de) |
KR (1) | KR100210417B1 (de) |
CN (1) | CN1043763C (de) |
AT (1) | ATE222587T1 (de) |
AU (1) | AU690257B2 (de) |
BG (1) | BG63259B1 (de) |
BR (1) | BR9507489A (de) |
CA (1) | CA2187309C (de) |
CZ (1) | CZ284379B6 (de) |
DE (1) | DE69527839T2 (de) |
DK (1) | DK0756596T3 (de) |
EE (1) | EE03877B1 (de) |
FI (1) | FI965074A0 (de) |
GE (1) | GEP19991749B (de) |
HU (1) | HU215830B (de) |
LV (1) | LV11738B (de) |
NO (1) | NO964180L (de) |
NZ (1) | NZ284075A (de) |
PL (1) | PL183025B1 (de) |
RU (1) | RU2134264C1 (de) |
SK (1) | SK280875B6 (de) |
UA (1) | UA49801C2 (de) |
WO (1) | WO1995028401A1 (de) |
Families Citing this family (21)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
TR199800628T2 (xx) * | 1995-10-13 | 1998-07-21 | Neurosearch A/S | 8-Azabisiklo$3.2.1]okt-2-en t�revleri, bunlar�n haz�rlanmas� ve kullan�m�. |
US6241963B1 (en) * | 1995-10-19 | 2001-06-05 | The Trustees Of The University Of Pennsylvania | Dopamine and serotonin transporter ligands and imaging agents |
DK0858461T3 (da) * | 1995-11-02 | 2003-01-27 | Neurosearch As | Kondenserede tropanderivater som neurotransmittergenoptagelsesinhibitorer |
US5948933A (en) | 1997-07-11 | 1999-09-07 | Organix, Inc. | Tropane analogs and methods for inhibition of monoamine transport |
CN1077574C (zh) | 1996-02-22 | 2002-01-09 | 神经研究公司 | 托烷衍生物,其制备和应用 |
US6232326B1 (en) | 1998-07-14 | 2001-05-15 | Jodi A. Nelson | Treatment for schizophrenia and other dopamine system dysfunctions |
US20040229908A1 (en) * | 1999-07-13 | 2004-11-18 | Jodi Nelson | Compositions and methods for the treatment of Parkinson's disease and tardive dyskinesias |
US6417177B1 (en) | 1999-07-13 | 2002-07-09 | Alpha Research Group, Llc | Chloroquine derivatives for the treatment of Parkinson's disease |
US6667314B2 (en) | 2000-05-26 | 2003-12-23 | Pfizer, Inc. | Tropane derivatives useful in therapy |
DK1526134T3 (da) * | 2000-05-26 | 2008-11-17 | Pfizer | Triazolyltropanderivater som CCR5-modulatorer |
JP2005508872A (ja) * | 2001-05-23 | 2005-04-07 | ニューロサーチ、アクティーゼルスカブ | トロパン誘導体及びこれをモノアミン神経伝達物質再取り込み阻害剤として使用する方法 |
US6610849B2 (en) * | 2001-06-28 | 2003-08-26 | Boehringer Ingelheim Pharma Kg | Process for the manufacture of tropenol |
AU2002365288A1 (en) * | 2001-11-30 | 2003-06-10 | Neurosearch A/S | Tropane derivatives having dopamine reuptake inhibitor activity for the treatment of ischemic diseases |
DE10200943A1 (de) * | 2002-01-12 | 2003-07-24 | Boehringer Ingelheim Pharma | Verfahren zur Herstellung von Scopinestern |
AU2003265233B2 (en) * | 2002-03-28 | 2008-05-08 | Organix, Inc. | Tropane compounds |
JP4874107B2 (ja) | 2003-10-03 | 2012-02-15 | ファイザー・インク | Hiv及び炎症の治療のためのccr5受容体拮抗活性を有するイミダゾピリジン置換トロパン誘導体 |
WO2005039580A1 (en) | 2003-10-16 | 2005-05-06 | Boehringer Ingelheim International Gmbh | Pharmaceutical composition comprising a monoamine neurotransmitter re-uptake inhibitor and an acetylcholinesterase inhibitor |
JP2007519646A (ja) * | 2004-01-22 | 2007-07-19 | ノイロサーチ アクティーゼルスカブ | 体重の持続的低減のための化合物 |
EP1708707A1 (de) * | 2004-01-22 | 2006-10-11 | Neurosearch A/S | Pharmazeutische zusammensetzung mit einem monoamin-neurotransmitter-wiederaufnahmehemmer und einem n-methyl-d-aspartat (nmda)-rezeptorantagonisten |
WO2006075976A1 (fr) * | 2005-01-14 | 2006-07-20 | Private Enterprise 'slavyanskaya Klinika' | Utilisation d'un anesthesique local pour corriger un comportement alimentaire humain, et procede d'utilisation associe |
EP1779851A1 (de) | 2005-10-31 | 2007-05-02 | Boehringer Ingelheim Pharma GmbH & Co.KG | Behandlung von Diabetes |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AU671163B2 (en) * | 1992-12-23 | 1996-08-15 | Neurosearch A/S | Alkyl substituted heterocyclic compounds |
AU672052B2 (en) * | 1992-12-23 | 1996-09-19 | Neurosearch A/S | Antidepressant and antiparkinsonian compounds |
-
1995
- 1995-04-12 AT AT95915869T patent/ATE222587T1/de not_active IP Right Cessation
- 1995-04-12 CA CA002187309A patent/CA2187309C/en not_active Expired - Fee Related
- 1995-04-12 SK SK1288-96A patent/SK280875B6/sk unknown
- 1995-04-12 GE GEAP19953459A patent/GEP19991749B/en unknown
- 1995-04-12 NZ NZ284075A patent/NZ284075A/en unknown
- 1995-04-12 KR KR1019960705823A patent/KR100210417B1/ko not_active IP Right Cessation
- 1995-04-12 BR BR9507489A patent/BR9507489A/pt not_active Application Discontinuation
- 1995-04-12 EP EP95915869A patent/EP0756596B1/de not_active Expired - Lifetime
- 1995-04-12 UA UA96103884A patent/UA49801C2/uk unknown
- 1995-04-12 DE DE69527839T patent/DE69527839T2/de not_active Expired - Lifetime
- 1995-04-12 AU AU22575/95A patent/AU690257B2/en not_active Ceased
- 1995-04-12 DK DK95915869T patent/DK0756596T3/da active
- 1995-04-12 CN CN95193151A patent/CN1043763C/zh not_active Expired - Fee Related
- 1995-04-12 JP JP7526700A patent/JP2899418B2/ja not_active Expired - Fee Related
- 1995-04-12 US US08/722,010 patent/US5736556A/en not_active Expired - Lifetime
- 1995-04-12 RU RU96121937A patent/RU2134264C1/ru active
- 1995-04-12 EE EE9600132A patent/EE03877B1/xx not_active IP Right Cessation
- 1995-04-12 WO PCT/EP1995/001358 patent/WO1995028401A1/en active IP Right Grant
- 1995-04-12 PL PL95316876A patent/PL183025B1/pl unknown
- 1995-04-12 CZ CZ962982A patent/CZ284379B6/cs not_active IP Right Cessation
- 1995-04-12 HU HU9602707A patent/HU215830B/hu not_active IP Right Cessation
-
1996
- 1996-10-02 NO NO964180A patent/NO964180L/no not_active Application Discontinuation
- 1996-10-02 BG BG100883A patent/BG63259B1/bg unknown
- 1996-11-11 LV LVP-96-428A patent/LV11738B/en unknown
- 1996-12-17 FI FI965074A patent/FI965074A0/fi active IP Right Revival
Also Published As
Similar Documents
Publication | Publication Date | Title |
---|---|---|
ATE222587T1 (de) | TROPAN-2-ALDOXIMDERIVATE ALS NEUROTRANSMITTER ßREUPTAKEß INHIBITOREN | |
DK0711280T3 (da) | Perhydroisoindolderivater, fremstilling af disse forbindelser og farmaceutiske præparater indeholdende disse forbindelser | |
BR9610960A (pt) | Derivados de 8-azabiciclo [3.2.1] oct -2- eno sua preparação e uso | |
FI964340A (fi) | Uudet asykliset ja sykliset amidit hermoston välittäjäaineen vapautumisen tehostimina | |
ES2173195T3 (es) | Derivados de antraciclina. | |
CA2112061A1 (en) | Alkyl substituted heterocyclic compounds | |
DE69633289D1 (de) | 4-acylamino(halogen)alkyl-chinolin derivate, deren herstellung und deren verwendung als melatonin-agonisten | |
BR9607841A (pt) | Método para a preparação de estéres de anidroeggonina |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
UEP | Publication of translation of european patent specification | ||
REN | Ceased due to non-payment of the annual fee |